PT1030852E - Derivados de oxazolidinona e composicoes farmaceuticas - Google Patents

Derivados de oxazolidinona e composicoes farmaceuticas

Info

Publication number
PT1030852E
PT1030852E PT98956200T PT98956200T PT1030852E PT 1030852 E PT1030852 E PT 1030852E PT 98956200 T PT98956200 T PT 98956200T PT 98956200 T PT98956200 T PT 98956200T PT 1030852 E PT1030852 E PT 1030852E
Authority
PT
Portugal
Prior art keywords
pharmaceutical compositions
oxazolidinone derivatives
organisms
compound
formula
Prior art date
Application number
PT98956200T
Other languages
English (en)
Portuguese (pt)
Inventor
Jackson B Hester Jr
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of PT1030852E publication Critical patent/PT1030852E/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
PT98956200T 1997-11-12 1998-10-30 Derivados de oxazolidinona e composicoes farmaceuticas PT1030852E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US6537697P 1997-11-12 1997-11-12

Publications (1)

Publication Number Publication Date
PT1030852E true PT1030852E (pt) 2004-02-27

Family

ID=22062294

Family Applications (1)

Application Number Title Priority Date Filing Date
PT98956200T PT1030852E (pt) 1997-11-12 1998-10-30 Derivados de oxazolidinona e composicoes farmaceuticas

Country Status (21)

Country Link
US (1) US5998406A (https=)
EP (1) EP1030852B1 (https=)
JP (1) JP2001522849A (https=)
KR (1) KR20010031953A (https=)
CN (1) CN1154644C (https=)
AT (1) ATE250054T1 (https=)
AU (1) AU739055B2 (https=)
BR (1) BR9813985A (https=)
CA (1) CA2303959A1 (https=)
DE (1) DE69818294T2 (https=)
DK (1) DK1030852T3 (https=)
ES (1) ES2207010T3 (https=)
HU (1) HUP0100470A3 (https=)
IL (1) IL136062A (https=)
NO (1) NO317291B1 (https=)
NZ (1) NZ504503A (https=)
PT (1) PT1030852E (https=)
RU (1) RU2215740C2 (https=)
SK (1) SK284577B6 (https=)
TR (1) TR200001330T2 (https=)
WO (1) WO1999024428A1 (https=)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1999064417A2 (en) 1998-06-05 1999-12-16 Astrazeneca Ab Oxazolidinone derivatives, process for their preparation and pharmaceutical compositions containing them
GB9928568D0 (en) 1999-12-03 2000-02-02 Zeneca Ltd Chemical compounds
DE19962924A1 (de) 1999-12-24 2001-07-05 Bayer Ag Substituierte Oxazolidinone und ihre Verwendung
KR100355345B1 (ko) * 2000-01-21 2002-10-12 한국과학기술연구원 티오펜환을 함유한 신규한 옥사졸리디논 유도체, 그의 제조방법 및 조성물
GB0009803D0 (en) 2000-04-25 2000-06-07 Astrazeneca Ab Chemical compounds
DE10129725A1 (de) 2001-06-20 2003-01-02 Bayer Ag Kombinationstherapie substituierter Oxazolidinone
DE60304360T2 (de) * 2002-08-12 2006-11-16 Pharmacia & Upjohn Co. Llc, Kalamazoo N-aryl-2-oxazolidinone und deren derivate
DE10300111A1 (de) * 2003-01-07 2004-07-15 Bayer Healthcare Ag Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid
MXPA06002188A (es) * 2003-08-25 2006-04-27 Warner Lambert Co Nuevos compuestos antimicrobianos de ariloxazolidinona.
DE10355461A1 (de) 2003-11-27 2005-06-23 Bayer Healthcare Ag Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung
KR100854211B1 (ko) * 2003-12-18 2008-08-26 동아제약주식회사 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물
CA2589250A1 (en) * 2004-11-29 2006-06-01 Pharmacia & Upjohn Company Llc Diazepine oxazolidinones as antibacterial agents
DE102004062475A1 (de) * 2004-12-24 2006-07-06 Bayer Healthcare Ag Feste, oral applizierbare pharmazeutische Darreichungsformen mit modifizierter Freisetzung
EP1685841A1 (en) * 2005-01-31 2006-08-02 Bayer Health Care Aktiengesellschaft Prevention and treatment of thromboembolic disorders
DE602006010702D1 (de) 2005-06-29 2010-01-07 Pharmacia & Upjohn Co Llc Homomorpholinoxazolidinone als antibakterielle mittel
DE102005045518A1 (de) 2005-09-23 2007-03-29 Bayer Healthcare Ag 2-Aminoethoxyessigsäure-Derivate und ihre Verwendung
DE102005047558A1 (de) * 2005-10-04 2008-02-07 Bayer Healthcare Ag Kombinationstherapie substituierter Oxazolidinone zur Prophylaxe und Behandlung von cerebralen Durchblutungsstörungen
DE102005047561A1 (de) 2005-10-04 2007-04-05 Bayer Healthcare Ag Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung
CA2624310C (en) 2005-10-04 2014-01-07 Bayer Healthcare Ag Polymorphic form of 5-chloro-n-({5s)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophenecarboxamide
KR20080110877A (ko) 2006-03-31 2008-12-19 재단법인 이쯔우 연구소 헤테로환을 갖는 신규 화합물
CN101883768A (zh) 2007-10-02 2010-11-10 财团法人乙卯研究所 具有7元杂环的噁唑烷酮衍生物
EP2635589A1 (en) 2010-11-03 2013-09-11 Wockhardt Limited Process for the preparation of phosphoric acid mono- (l-{4- [(s) -5- (acetylaminomethyl) - 2 - oxo - oxazolidin- 3 - yl]- 2, 6 - difluorophenyl} - 4 -methoxymethylpiperidin- 4 - yl) ester
WO2015173664A1 (en) 2014-05-14 2015-11-19 Wockhardt Limited Process for the preparation of (5s)-n-{3-[3,5-difluoro-4-(4-hydroxy-4-methoxymethyl-piperidin-1-yl)-phenyl]-2-oxo-oxazolidin-5-ylmethyl}-acetamide

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4801600A (en) * 1987-10-09 1989-01-31 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
CA1320730C (en) * 1987-10-16 1993-07-27 The Du Pont Merck Pharmaceutical Company Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents
ES2059467T3 (es) * 1987-10-21 1994-11-16 Du Pont Merck Pharma Derivados de aminometil-oxooxazolidinil-etenilbenceno utiles como agentes antibacterianos.
US4948801A (en) * 1988-07-29 1990-08-14 E. I. Du Pont De Nemours And Company Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents
JP2865211B2 (ja) * 1988-09-15 1999-03-08 ファルマシア・アンド・アップジョン・カンパニー ５’―インドリニル―５β―アミドメチルオキサゾリジン―２―オン類、３―（縮合環置換）フェニル―５β―アミドメチルオキサゾリジン―２―オン類および３―（窒素原子置換）フェニル―５β―アミドメチルオキサゾリジン―２―オン類
EP0610265B1 (en) * 1991-11-01 1996-12-27 PHARMACIA & UPJOHN COMPANY Substituted aryl- and heteroarylphenyloxazolidinones useful as antibacterial agents
SK283420B6 (sk) * 1992-05-08 2003-07-01 Pharmacia & Upjohn Company Antimikrobiálne oxazolidinóny obsahujúce substituované diazínové skupiny
CA2174107C (en) * 1993-11-22 2005-04-12 Steven J. Brickner Esters of substituted-hydroxyacetyl piperazine phenyl oxazolidinones
JPH0873455A (ja) * 1994-03-15 1996-03-19 Upjohn Co:The オキサゾリジノン誘導体及びこれを有効成分とする医薬組成物
GB9601666D0 (en) * 1996-01-27 1996-03-27 Zeneca Ltd Chemical compounds

Also Published As

Publication number Publication date
AU1277899A (en) 1999-05-31
TR200001330T2 (tr) 2000-11-21
EP1030852B1 (en) 2003-09-17
IL136062A (en) 2004-02-08
CN1154644C (zh) 2004-06-23
EP1030852A1 (en) 2000-08-30
SK6182000A3 (en) 2000-12-11
NO317291B1 (no) 2004-10-04
HUP0100470A3 (en) 2002-08-28
NZ504503A (en) 2002-10-25
DE69818294D1 (de) 2003-10-23
DK1030852T3 (da) 2003-12-22
SK284577B6 (sk) 2005-07-01
ES2207010T3 (es) 2004-05-16
CN1271358A (zh) 2000-10-25
US5998406A (en) 1999-12-07
NO20002434D0 (no) 2000-05-11
DE69818294T2 (de) 2004-07-08
JP2001522849A (ja) 2001-11-20
HK1030373A1 (en) 2001-05-04
ATE250054T1 (de) 2003-10-15
RU2215740C2 (ru) 2003-11-10
NO20002434L (no) 2000-05-11
AU739055B2 (en) 2001-10-04
CA2303959A1 (en) 1999-05-20
WO1999024428A1 (en) 1999-05-20
HUP0100470A2 (hu) 2002-05-29
BR9813985A (pt) 2000-09-26
IL136062A0 (en) 2001-05-20
KR20010031953A (ko) 2001-04-16

Similar Documents

Publication Publication Date Title
PT1030852E (pt) Derivados de oxazolidinona e composicoes farmaceuticas
NO996269L (no) Kinolin-indol antimikrobielle midler, samt anvendelse og blandinger derav
ATE232862T1 (de) Oxazolidinon derivate und diese enthaltende pharmazeutische zusammensetzungen
FI950309A0 (fi) Proliiniamidijohdannaisia
SE9604786D0 (sv) New compounds
PA8451801A1 (es) Derivados de la 9-oxima eritromicina
DE69721679D1 (de) Antimikrobielle Zusammensetzung.
WO2001003685A3 (en) Novel prodrugs for antimicrobial amidines
PL358666A1 (en) 2-hydroxy-mutilin carbamate derivatives for antibacterial use
NZ333926A (en) Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
CA2386685A1 (en) Use of pleuromutilin derivatives for transdermal treatment of bacterial diseases
ATE203246T1 (de) Dialkyltiacumicine
ATE205505T1 (de) Basische oxazolinamid-derivate von ge2270 und ge2270-änlichen antibiotika
NO331012B1 (no) N-sulfonyl-4-metylenamino-3-hydroksy-2-pyridoner som antimikrobielle midler
ATE165101T1 (de) Basische prolinamid derivate von ge2270 und ge2270-ahnlichten antibiotika
DE60005517D1 (de) Kaliumkanal-blockierende mittel
DE60030300D1 (de) Topische behandlung zur vorbeugung von augeninfektionen
KR970703147A (ko) 동맥경화 억제제(Arteriosclerosis Depressant)
MY122570A (en) Benzamide derivatives and drugs containing the same
BG101996A (en) 9-n-ethylenederivatives of 9(s)-erythromycylamine
NZ503027A (en) Use of rifamycin derivative for treating mastitis in a domestic animal
ATE234320T1 (de) Beta,beta-disubstituierte derivate von 9-deoxo-9a-n-ethenyl-9a-aza-9a-homoerythromycin a
TR199700921T1 (xx) �nsanlarda g�r�len herpes-vir�s-8'in tedavisinde pensiklovir'in kullan�lmas�.
DE60011096D1 (de) Ester enthaltende zusammensetzungen zur behandlung von parasitischem befall in organismen
BR0215070A (pt) Métodos de tratamento de infecções bacterianas em cães e gatos