PL3486233T3 - Słabo rozpuszczalny kompleks lub jego solwat, kompozycja farmaceutyczna i jej zastosowanie - Google Patents

Słabo rozpuszczalny kompleks lub jego solwat, kompozycja farmaceutyczna i jej zastosowanie

Info

Publication number
PL3486233T3
PL3486233T3 PL18777940T PL18777940T PL3486233T3 PL 3486233 T3 PL3486233 T3 PL 3486233T3 PL 18777940 T PL18777940 T PL 18777940T PL 18777940 T PL18777940 T PL 18777940T PL 3486233 T3 PL3486233 T3 PL 3486233T3
Authority
PL
Poland
Prior art keywords
solvate
application
pharmaceutical composition
poorly soluble
soluble complex
Prior art date
Application number
PL18777940T
Other languages
English (en)
Inventor
Shanchun ZHANG
Yihua Wang
Jiashi PENG
Kaisheng CHENG
Xiao Wang
Shu Gao
Hongzhang Sun
Xiaorong LU
Original Assignee
Fruithy Holdings Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fruithy Holdings Limited filed Critical Fruithy Holdings Limited
Publication of PL3486233T3 publication Critical patent/PL3486233T3/pl

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/235—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group
    • A61K31/24—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group having an amino or nitro group
    • A61K31/245—Amino benzoic acid types, e.g. procaine, novocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
    • A61K47/542—Carboxylic acids, e.g. a fatty acid or an amino acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00—Anaesthetics
    • A61P23/02—Local anaesthetics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C65/00—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C65/01—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups
    • C07C65/105—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups polycyclic
    • C07C65/11—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing hydroxy or O-metal groups polycyclic with carboxyl groups on a condensed ring system containing two rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Anesthesiology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)
PL18777940T 2017-03-27 2018-03-26 Słabo rozpuszczalny kompleks lub jego solwat, kompozycja farmaceutyczna i jej zastosowanie PL3486233T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN201710188001 2017-03-27
EP18777940.0A EP3486233B1 (en) 2017-03-27 2018-03-26 Poorly soluble complex or solvate thereof, pharmaceutical composition, and application thereof
PCT/CN2018/080424 WO2018177232A1 (zh) 2017-03-27 2018-03-26 难溶性复合物或其溶剂合物、药物组合物及其应用

Publications (1)

Publication Number Publication Date
PL3486233T3 true PL3486233T3 (pl) 2021-06-28

Family

ID=63675241

Family Applications (1)

Application Number Title Priority Date Filing Date
PL18777940T PL3486233T3 (pl) 2017-03-27 2018-03-26 Słabo rozpuszczalny kompleks lub jego solwat, kompozycja farmaceutyczna i jej zastosowanie

Country Status (18)

Country Link
US (1) US11084790B2 (pl)
EP (1) EP3486233B1 (pl)
JP (1) JP6923122B2 (pl)
KR (1) KR102248445B1 (pl)
CN (1) CN109996787B (pl)
AU (1) AU2018241564B2 (pl)
CA (1) CA3049220C (pl)
DK (1) DK3486233T3 (pl)
EA (1) EA039449B1 (pl)
ES (1) ES2866401T3 (pl)
HU (1) HUE053472T2 (pl)
MY (1) MY199896A (pl)
PH (1) PH12019501560B1 (pl)
PL (1) PL3486233T3 (pl)
PT (1) PT3486233T (pl)
SG (1) SG11201906132UA (pl)
TW (1) TWI740045B (pl)
WO (1) WO2018177232A1 (pl)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN110483372A (zh) * 2018-05-14 2019-11-22 南京诺瑞特医药科技有限公司 布比卡因的盐
CN111983052B (zh) * 2020-07-24 2023-03-31 合肥诺明药物安全研究有限公司 一种hyr-pb21有效成分血药浓度的定量分析方法
KR102741835B1 (ko) 2022-03-11 2024-12-12 한국한의약진흥원 등검은말벌독에 함유된 세로토닌의 안정성을 유지하기 위한 조성물
CN118566394A (zh) * 2024-08-01 2024-08-30 山东省食品药品检验研究院 一种曲安奈德混悬注射液的流通池溶出度测定方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003099293A1 (en) 2002-05-23 2003-12-04 Danmarks Farmaceutiske Universitet Pharmacologically active salts
US20070110804A1 (en) * 2003-06-20 2007-05-17 Royer Biomedical, Inc. Drug polymer complexes
BRPI0515372B8 (pt) * 2004-09-17 2021-05-25 Durect Corp composição líquida para fornecer anestesia local prolongada após administração a um indivíduo, e, uso de bupivacaína, acetato isobutirato de sacarose e álcool benzílico
US8920843B2 (en) 2007-11-07 2014-12-30 Svip5 Llc Slow release of organic salts of local anesthetics for pain relief
SI2398468T1 (sl) 2009-02-17 2017-03-31 Krka, D.D., Novo Mesto Farmacevtske sestave, ki obsegajo prasugrel ali njegove farmacevtsko sprejemljive kislinske adicijske soli in postopek za njihovo pripravo
CZ2009762A3 (cs) 2009-11-16 2011-05-25 Zentiva, K. S. Nové soli 5-[2-cyklopropyl-1-(2-fluorfenyl)-2-oxoethyl]-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl acetátu známého pod nechráneným názvem prasugrel a zpusob jejich výroby
CN104370934B (zh) * 2013-08-13 2018-04-06 上海科胜药物研发有限公司 一种普拉格雷盐及其制备方法
WO2017036408A1 (zh) * 2015-09-01 2017-03-09 四川海思科制药有限公司 S-(-)-1-丙基-2',6'-二甲苯胺甲酰基哌啶晶体及其缓释制剂
CN110325179A (zh) * 2016-12-26 2019-10-11 塞尔利克斯生物私人有限公司 用于治疗慢性疼痛的组合物和方法

Also Published As

Publication number Publication date
TW201940170A (zh) 2019-10-16
PT3486233T (pt) 2021-03-18
US20210087144A1 (en) 2021-03-25
CN109996787B (zh) 2022-07-05
WO2018177232A1 (zh) 2018-10-04
KR102248445B1 (ko) 2021-05-04
JP2020515513A (ja) 2020-05-28
SG11201906132UA (en) 2019-10-30
HUE053472T2 (hu) 2021-06-28
EP3486233A4 (en) 2020-04-08
CN109996787A (zh) 2019-07-09
CA3049220A1 (en) 2018-10-04
EP3486233B1 (en) 2021-01-27
JP6923122B2 (ja) 2021-08-18
EP3486233A1 (en) 2019-05-22
EA039449B1 (ru) 2022-01-28
PH12019501560A1 (en) 2020-02-24
PH12019501560B1 (en) 2023-09-27
AU2018241564A1 (en) 2019-05-30
EA201990419A1 (ru) 2019-09-30
CA3049220C (en) 2022-03-29
DK3486233T3 (da) 2021-03-15
US11084790B2 (en) 2021-08-10
MY199896A (en) 2023-11-28
AU2018241564B2 (en) 2020-07-02
KR20190101980A (ko) 2019-09-02
TWI740045B (zh) 2021-09-21
ES2866401T3 (es) 2021-10-19

Similar Documents

Publication Publication Date Title
ZA201802125B (en) Pharmaceutical composition and application thereof
IL269061A (en) A pharmaceutical preparation containing Selexifag
IL271986B1 (en) pharmaceutical preparation
PT3606511T (pt) Composição farmacêutica compreendendo mesilato de lenvatinib
ZA201804692B (en) Quinazolinone derivative, preparation method therefor, pharmaceutical composition, and applications
IL273339A (en) Griseofulbin compound and its medical use
GB201709141D0 (en) Pharmaceutical formulation
EP3381925A4 (en) Deuterium-modified brigatinib derivatives, pharmaceutical compositions comprising same, and use thereof
IL262929B1 (en) Preparations for treatment, methods of their preparation and their uses
GB201712159D0 (en) Pharmaceutical composition
IL248773B (en) History -6,1-Naphthyridine-5,4-Dione and pharmaceutical preparations containing them
HUE068810T2 (hu) Gyógyászati készítmény
IL272419A (en) Pharmaceutical composition
GB201719447D0 (en) Pharmaceutical composition
EP3486233A4 (en) POORLY SOLUBLE COMPLEX OR SOLVATE THEREOF, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF
PL3658122T3 (pl) Kompozycja farmaceutyczna zawierająca sakubitryl i walsartan
PL3646867T3 (pl) Kompozycja farmaceutyczna
EP3647325A4 (en) PHARMACEUTICAL COMPOSITION OF PCSK-9 ANTIBODIES AND USES THEREOF
IL257621B (en) A catechol derivative and a pharmaceutical preparation that includes it
ZA202000959B (en) Adamantylmethylamine derivative and use thereof as pharmaceutical
ZA201903341B (en) Pharmaceutical compositions and uses thereof
GB201713920D0 (en) Pharmaceutical compositions and uses thereof
HK40020689A (en) Pharmaceutical compositions and uses thereof
GB201812022D0 (en) Pharmaceutical methods and compositions
GB201708328D0 (en) Pharmaceutical composition