PL2589599T3 - Nowe hydroksy-6-heteroarylofenantrydyny i ich zastosowanie jako inhibitorów PDE4 - Google Patents

Nowe hydroksy-6-heteroarylofenantrydyny i ich zastosowanie jako inhibitorów PDE4

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Publication number
PL2589599T3
PL2589599T3 PL12196702T PL12196702T PL2589599T3 PL 2589599 T3 PL2589599 T3 PL 2589599T3 PL 12196702 T PL12196702 T PL 12196702T PL 12196702 T PL12196702 T PL 12196702T PL 2589599 T3 PL2589599 T3 PL 2589599T3
Authority
PL
Poland
Prior art keywords
heteroarylphenanthridines
pde4 inhibitors
novel hydroxy
hydroxy
novel
Prior art date
Application number
PL12196702T
Other languages
English (en)
Other versions
PL2589599T4 (pl
Inventor
Ulrich Kautz
Beate Schmidt
Dieter Flockerzi
Armin Hatzelmann
Christof Zitt
Johannes Barsig
Degenhard Marx
Hans-Peter Kley
Original Assignee
Takeda Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Gmbh filed Critical Takeda Gmbh
Publication of PL2589599T3 publication Critical patent/PL2589599T3/pl
Publication of PL2589599T4 publication Critical patent/PL2589599T4/pl

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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/473Quinolines; Isoquinolines ortho- or peri-condensed with carbocyclic ring systems, e.g. acridines, phenanthridines
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    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
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    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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PL12196702T 2004-03-03 2005-03-02 Nowe hydroksy-6-heteroarylofenantrydyny i ich zastosowanie jako inhibitorów PDE4 PL2589599T4 (pl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
EP04004973 2004-03-03
EP04106359 2004-12-07
EP05716889.0A EP1723135B1 (en) 2004-03-03 2005-03-02 Novel hydroxy-6-heroarylphenanthridines and their use as pde4 inhibitors
EP20120196702 EP2589599B1 (en) 2004-03-03 2005-03-02 Novel hydroxy-6-heteroarylphenanthridines and their use as PDE4 inhibitors

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