PL112867B1 - Process for preparing novel derivatives of kanamycin - Google Patents

Process for preparing novel derivatives of kanamycin Download PDF

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Publication number
PL112867B1
PL112867B1 PL1977215139A PL21513977A PL112867B1 PL 112867 B1 PL112867 B1 PL 112867B1 PL 1977215139 A PL1977215139 A PL 1977215139A PL 21513977 A PL21513977 A PL 21513977A PL 112867 B1 PL112867 B1 PL 112867B1
Authority
PL
Poland
Prior art keywords
groups
group
kanamycin
product
acid
Prior art date
Application number
PL1977215139A
Other languages
English (en)
Polish (pl)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of PL112867B1 publication Critical patent/PL112867B1/pl

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/22Cyclohexane rings, substituted by nitrogen atoms
    • C07H15/222Cyclohexane rings substituted by at least two nitrogen atoms
    • C07H15/226Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
    • C07H15/234Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Biotechnology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
PL1977215139A 1976-04-14 1977-04-13 Process for preparing novel derivatives of kanamycin PL112867B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB15421/76A GB1530201A (en) 1976-04-14 1976-04-14 Process for the preparation of aminoglycoside antibiotics and intermediates therefor

Publications (1)

Publication Number Publication Date
PL112867B1 true PL112867B1 (en) 1980-11-29

Family

ID=10058845

Family Applications (2)

Application Number Title Priority Date Filing Date
PL1977215139A PL112867B1 (en) 1976-04-14 1977-04-13 Process for preparing novel derivatives of kanamycin
PL19737277A PL197372A1 (pl) 1976-04-14 1977-04-13 Sposob wytwarzania pochodnych kanamycyny

Family Applications After (1)

Application Number Title Priority Date Filing Date
PL19737277A PL197372A1 (pl) 1976-04-14 1977-04-13 Sposob wytwarzania pochodnych kanamycyny

Country Status (28)

Country Link
JP (2) JPS52139044A (member.php)
AR (1) AR219074A1 (member.php)
AT (1) AT356267B (member.php)
AU (1) AU497416B2 (member.php)
BE (1) BE853564A (member.php)
BG (2) BG28072A4 (member.php)
CA (1) CA1083568A (member.php)
CH (1) CH622528A5 (member.php)
CS (1) CS202570B2 (member.php)
DD (2) DD135496A5 (member.php)
DE (1) DE2716533C3 (member.php)
DK (1) DK164277A (member.php)
EG (1) EG12909A (member.php)
ES (1) ES457793A1 (member.php)
FI (1) FI771144A7 (member.php)
FR (1) FR2348223A1 (member.php)
GB (1) GB1530201A (member.php)
GR (1) GR68936B (member.php)
IE (1) IE45030B1 (member.php)
IL (1) IL51775A (member.php)
LU (1) LU77108A1 (member.php)
NL (1) NL7703567A (member.php)
NZ (1) NZ183733A (member.php)
PH (1) PH14029A (member.php)
PL (2) PL112867B1 (member.php)
PT (1) PT66422B (member.php)
RO (2) RO79969A (member.php)
ZA (1) ZA771944B (member.php)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2924659A1 (de) * 1979-06-19 1981-01-22 Bayer Ag Pseudotrisaccharide, ihre herstellung und verwendung als arzneimittel
JPS61191642U (member.php) * 1985-05-20 1986-11-28
IT1225484B (it) * 1987-11-27 1990-11-14 Pierrel Spa Procedimento di sintesi dell'amikacina
CN101481397B (zh) * 2009-01-23 2012-10-31 北京大学 一种新的卡那霉素a衍生物及其制备方法和用途
WO2012064266A1 (en) 2010-11-04 2012-05-18 Albireo Ab Ibat inhibitors for the treatment of liver diseases
KR102560954B1 (ko) 2014-06-25 2023-07-31 이에이 파마 가부시키가이샤 고형 제제 및 그의 착색 방지 또는 착색 감소 방법
US20170143738A1 (en) 2014-06-25 2017-05-25 Ea Pharma Co., Ltd. Solid formulation and method for stabilizing the same
EP3012252A1 (en) 2014-10-24 2016-04-27 Ferring BV Crystal modifications of elobixibat
US10786529B2 (en) 2016-02-09 2020-09-29 Albireo Ab Oral cholestyramine formulation and use thereof
US10441604B2 (en) 2016-02-09 2019-10-15 Albireo Ab Cholestyramine pellets and methods for preparation thereof
US10441605B2 (en) 2016-02-09 2019-10-15 Albireo Ab Oral cholestyramine formulation and use thereof
US11007142B2 (en) 2018-08-09 2021-05-18 Albireo Ab Oral cholestyramine formulation and use thereof
US10722457B2 (en) 2018-08-09 2020-07-28 Albireo Ab Oral cholestyramine formulation and use thereof

Also Published As

Publication number Publication date
PT66422A (en) 1977-05-01
LU77108A1 (member.php) 1979-01-18
RO79969B (ro) 1983-01-30
JPS52139044A (en) 1977-11-19
JPS5549587B2 (member.php) 1980-12-12
AT356267B (de) 1980-04-25
PT66422B (en) 1978-09-18
DE2716533A1 (de) 1977-11-03
GR68936B (member.php) 1982-03-29
IL51775A0 (en) 1977-05-31
PH14029A (en) 1980-12-12
DD130661A5 (de) 1978-04-19
BG28072A4 (bg) 1980-02-25
CS202570B2 (en) 1981-01-30
DE2716533B2 (de) 1981-04-30
GB1530201A (en) 1978-10-25
AU2372177A (en) 1978-10-05
ATA261477A (de) 1979-09-15
DE2716533C3 (de) 1982-05-13
FR2348223A1 (fr) 1977-11-10
ZA771944B (en) 1978-03-29
PL197372A1 (pl) 1979-06-18
ES457793A1 (es) 1978-08-01
IE45030B1 (en) 1982-06-02
IL51775A (en) 1980-07-31
FI771144A7 (member.php) 1977-10-15
CH622528A5 (en) 1981-04-15
RO79969A (ro) 1983-02-01
AU497416B2 (en) 1978-12-14
IE45030L (en) 1977-10-14
DK164277A (da) 1977-10-15
CA1083568A (en) 1980-08-12
JPS535141A (en) 1978-01-18
EG12909A (en) 1979-12-31
BE853564A (fr) 1977-10-13
BG27759A3 (bg) 1979-12-12
JPS5421326B2 (member.php) 1979-07-30
AR219074A1 (es) 1980-07-31
NZ183733A (en) 1979-12-11
DD135496A5 (de) 1979-05-09
NL7703567A (nl) 1977-10-18
RO74431A (ro) 1981-08-30

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