PH23791A - Novel aminoalkylthio derivatives of triazolophiridine or triazoloquinoline,the processes for their preparation and pharmaceutical composition thereof - Google Patents

Novel aminoalkylthio derivatives of triazolophiridine or triazoloquinoline,the processes for their preparation and pharmaceutical composition thereof

Info

Publication number
PH23791A
PH23791A PH35574A PH35574A PH23791A PH 23791 A PH23791 A PH 23791A PH 35574 A PH35574 A PH 35574A PH 35574 A PH35574 A PH 35574A PH 23791 A PH23791 A PH 23791A
Authority
PH
Philippines
Prior art keywords
heterocycle
phenyl
ring
lower alkyl
atoms
Prior art date
Application number
PH35574A
Other languages
English (en)
Inventor
Nicole Bru-Magniez
Jean-Marie Teulon
Michele Launay
Original Assignee
Carpibem
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Carpibem filed Critical Carpibem
Publication of PH23791A publication Critical patent/PH23791A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PH35574A 1986-07-23 1987-07-22 Novel aminoalkylthio derivatives of triazolophiridine or triazoloquinoline,the processes for their preparation and pharmaceutical composition thereof PH23791A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8610709A FR2601952B1 (fr) 1986-07-23 1986-07-23 Nouveaux derives amino alkyl thio de triazolopyridine ou triazoloquinoline, leurs procedes de preparation, medicaments les contenant, utiles notamment comme antalgiques

Publications (1)

Publication Number Publication Date
PH23791A true PH23791A (en) 1989-11-03

Family

ID=9337681

Family Applications (1)

Application Number Title Priority Date Filing Date
PH35574A PH23791A (en) 1986-07-23 1987-07-22 Novel aminoalkylthio derivatives of triazolophiridine or triazoloquinoline,the processes for their preparation and pharmaceutical composition thereof

Country Status (18)

Country Link
US (1) US4886805A (da)
EP (1) EP0254623B1 (da)
JP (1) JP2535355B2 (da)
KR (1) KR960000358B1 (da)
AT (1) ATE90349T1 (da)
AU (1) AU601452B2 (da)
CA (2) CA1334968C (da)
DE (1) DE3786118T2 (da)
DK (2) DK170472B1 (da)
ES (1) ES2058134T3 (da)
FR (1) FR2601952B1 (da)
IE (1) IE60116B1 (da)
IL (1) IL83206A0 (da)
LV (1) LV10716B (da)
NZ (1) NZ221141A (da)
PH (1) PH23791A (da)
PT (1) PT85387B (da)
ZA (1) ZA875424B (da)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2687147A1 (fr) * 1992-02-11 1993-08-13 Union Pharma Scient Appl Nouveaux derives d'alpha-amino n-pyridyl benzene propanamide, leurs procedes de preparation, compositions pharmaceutiques les contenant.
DE4425144A1 (de) * 1994-07-15 1996-01-18 Basf Ag Triazolverbindungen und deren Verwendung
US6403593B1 (en) 1995-07-14 2002-06-11 Abbott Laboratories Triazole compounds and the use thereof
DE19728996A1 (de) 1997-07-07 1999-01-14 Basf Ag Triazolverbindungen und deren Verwendung
AR022230A1 (es) 1999-01-12 2002-09-04 Abbott Gmbh & Co Kg Compuestos de triazol, composicion farmaceutica que los comprende y uso de los mismos para preparar dicha composicion
US6989392B2 (en) 2002-06-18 2006-01-24 Abbott Laboratories 2-Aminoquinolines as melanin concentrating hormone receptor antagonists
PE20080403A1 (es) * 2006-07-14 2008-04-25 Amgen Inc Derivados heterociclicos fusionados y metodos de uso
US8217177B2 (en) 2006-07-14 2012-07-10 Amgen Inc. Fused heterocyclic derivatives and methods of use
US8198448B2 (en) 2006-07-14 2012-06-12 Amgen Inc. Fused heterocyclic derivatives and methods of use
EP1972628A1 (en) * 2007-03-21 2008-09-24 Schwarz Pharma Ag Indolizines and aza-analog derivatives thereof as CNS active compounds
FR2941229B1 (fr) * 2009-01-21 2012-11-30 Sanofi Aventis Nouveaux derives triazolo°4,3-a!pyridine, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de met
FR2933980B1 (fr) * 2008-07-18 2011-07-29 Sanofi Aventis Nouveaux derives triazolo°4,3-a!pyridine, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de met
PE20110560A1 (es) * 2008-07-18 2011-08-29 Sanofi Aventis NUEVOS DERIVADOS DE TRIAZOLO[4,3-a]PIRIDINA, SU PROCEDIMIENTO DE PREPARACION, SU APLICACION COMO MEDICAMENTOS, COMPOSICIONES FARMACEUTICAS Y NUEVA UTILIZACION PARTICULARMENTE COMO INHIBIDORES DE MET
MX339302B (es) 2011-09-15 2016-05-19 Novartis Ag 3-(quinolin-6-il-tio)-[1,2,4]-triazolo-[4,3-a]-piridinas 6-sustituidas como cinasas de tirosina.
GB201321742D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
CN105541702B (zh) * 2016-01-27 2019-10-22 宜春学院 类卢扎朵仑结构的芳胺基烷基硫类化合物及其制备方法
KR102230681B1 (ko) 2019-10-17 2021-03-22 주식회사 포스코건설 태그유닛 및 이를 포함하는 진동측정장치

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3050525A (en) * 1960-12-14 1962-08-21 John B Bicking Certain derivatives of s-triazolo [4, 3-a]-pyridine
US4244953A (en) * 1979-10-24 1981-01-13 American Cyanamid Company Substituted 6-phenyl-5,6,7,8-tetrahydro-1,2,4-triazolo-[4,3-a]pyridines
US4340597A (en) * 1981-04-13 1982-07-20 Schering Corporation 1-Substituted-4-aryl-1,2,5,6-tetrahydro and hexahydropyridines
US4358454A (en) * 1982-01-08 1982-11-09 Schering Corporation 1,3,4-Triazolo[1,5-a]pyridines
US4358453A (en) * 1982-01-08 1982-11-09 Schering Corporation 1,2,4-Triazolo[4,3-a]pyridines
US4419516A (en) * 1982-06-16 1983-12-06 American Home Products Corporation Antiviral imidazo- and triazolo-pyridines
JPH0439094A (ja) * 1990-06-06 1992-02-10 Fuji Photo Film Co Ltd 直描型平版印刷用原版

Also Published As

Publication number Publication date
DK84093D0 (da) 1993-07-14
ES2058134T3 (es) 1994-11-01
IE60116B1 (en) 1994-06-01
US4886805A (en) 1989-12-12
LV10716B (en) 1995-12-20
FR2601952A1 (fr) 1988-01-29
DK84093A (da) 1993-07-14
ZA875424B (en) 1988-04-27
JP2535355B2 (ja) 1996-09-18
DE3786118D1 (de) 1993-07-15
IE871880L (en) 1988-01-23
FR2601952B1 (fr) 1988-11-25
KR960000358B1 (ko) 1996-01-05
LV10716A (lv) 1995-06-20
CA1338908C (en) 1997-02-11
IL83206A0 (en) 1987-12-31
EP0254623B1 (fr) 1993-06-09
DK382987A (da) 1988-01-24
KR880001650A (ko) 1988-04-25
JPS6335572A (ja) 1988-02-16
DK382987D0 (da) 1987-07-22
NZ221141A (en) 1990-05-28
EP0254623A1 (fr) 1988-01-27
DK170472B1 (da) 1995-09-11
AU601452B2 (en) 1990-09-13
PT85387A (fr) 1987-08-01
ATE90349T1 (de) 1993-06-15
AU7616387A (en) 1988-01-28
PT85387B (pt) 1990-04-30
DE3786118T2 (de) 1993-10-28
CA1334968C (en) 1995-03-28
DK170533B1 (da) 1995-10-16

Similar Documents

Publication Publication Date Title
PH23791A (en) Novel aminoalkylthio derivatives of triazolophiridine or triazoloquinoline,the processes for their preparation and pharmaceutical composition thereof
HUP9802534A2 (hu) Neurotranszmitter újrafelvételt gátló kondenzált tropánszármazékok és előállításuk, e vegyületeket tartalmazó gyógyászati készítmények, valamint e vegyületek alkalmazása
IL95568A0 (en) N-substituted-4-pyrimidinamines and pyrimidinidiamines,process for their preparation and pharmaceutical compositions containing them
FI954105A (fi) Uusia 4-aminopyridiinejä, niiden valmistusmenetelmä sekä näitä yhdisteitä sisältäviä lääkkeitä
IL111355A0 (en) Pharmaceutical compositions containing aminoquinoline derivatives, certain such novel compounds and their preparation
ATE74352T1 (de) Dekahydrochinolinderivate, verfahren zu ihrer herstellung, zwischenprodukte zu ihrer herstellung, ihre verwendung als arzneimittel und diese enthaltende zubereitungen.
DE3869173D1 (de) Amino 5,6,7,8-tetrahydronaphtho(2,3b)furanderivate, verfahren zu ihrer herstellung und diese enthaltende arzneimittel.
AU5795694A (en) New bicyclic nitrogen compounds, process for preparing them and pharmaceutical compositions containing them
KR900003156A (ko) 진통제 화합물, 그의 제조방법 및 그를 함유하는 약학 조성물
DE3882438D1 (de) Alkansulfonanilid-derivate, verfahren zu deren herstellung und diese enthaltende pharmazeutische zusammensetzung.
AU2186288A (en) Novel amide compounds, process for preparing the same, and composition for activating gastric motor function containing the same
IL111375A (en) N-substituted azabicycloalkane derivatives and pharmaceutical compositions containing them
IE832581L (en) Piperidinedione derivatives, possessing anti-arrythmic¹activity, for protecting the myocardium, process for their¹preparation and pharmaceutical compositions containing said¹derivatives
ZA926277B (en) 1-(alkoxybenzyl)piperazine amide compounds, process for preparing them and pharmaceutical compositions containing them.
ES8103081A1 (es) Procedimiento para la obtencion de diazatriciclos
DK0410278T3 (da) Reninhæmmende aminooligohydroxyderivater
ES2000458A6 (es) Procedimiento para la obtencion de nuevos tieno-1,2-tiazolderivados y sales farmaceuticamente aceptables de los mismos
ZA874970B (en) Derivatives of 2,6-piperazinedione,their preparation processes and the pharmaceutical compositions containing them
ATE33134T1 (de) 2-aminoethyl-pyridin oder pyrazin-derivate, ihre herstellung und diese enthaltende pharmazeutische zusammensetzungen.
SE7905051L (sv) Nya sulfonamider
IL69931A (en) N-(6-chloro-pyrazin-2-yl)-4-hydroxy-2h-1,2-benzothiazine-3-carboxamide-1,1-dioxides,their preparation and pharmaceutical compositions containing them
ES8104248A1 (es) Procedimiento de preparacion de 6-amino-sustituidas-3-piri- dazinilhidrazinas y de sus sales de adicion acidas terapeu- ticamente aceptables
GB2133012B (en) Quinazolines process for their preparation and pharmaceutical compositions containing them
ES2006336A6 (es) Procedimiento de preparacion de nuevas acetamidas derivadas de la 2,3-dihidro-3-fenil-2-benzofuranona.
ES2058761T3 (es) Proceso para la preparacion de derivados de dibenzodioxazecina y dibenzodioxaazacicloundecina.