DK84093A - Mellemprodukt bestaaende af 4-(2,4-difluorphenyl)-piperazin eller et syreadditionssalt deraf samt farmaceutisk praeparat og laegemiddel indeholdende mindst en af disse forbindelser - Google Patents

Mellemprodukt bestaaende af 4-(2,4-difluorphenyl)-piperazin eller et syreadditionssalt deraf samt farmaceutisk praeparat og laegemiddel indeholdende mindst en af disse forbindelser

Info

Publication number
DK84093A
DK84093A DK084093A DK84093A DK84093A DK 84093 A DK84093 A DK 84093A DK 084093 A DK084093 A DK 084093A DK 84093 A DK84093 A DK 84093A DK 84093 A DK84093 A DK 84093A
Authority
DK
Denmark
Prior art keywords
piperazine
heterocycle
phenyl
ring
lower alkyl
Prior art date
Application number
DK084093A
Other languages
English (en)
Other versions
DK84093D0 (da
DK170533B1 (da
Inventor
Nicole Bru-Magniez
Jean-Marie Teulon
Michele Launay
Original Assignee
Union Pharma Scient Appl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Union Pharma Scient Appl filed Critical Union Pharma Scient Appl
Publication of DK84093D0 publication Critical patent/DK84093D0/da
Publication of DK84093A publication Critical patent/DK84093A/da
Application granted granted Critical
Publication of DK170533B1 publication Critical patent/DK170533B1/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK084093A 1986-07-23 1993-07-14 4-(2,4-Difluorphenyl)-piperazin eller et syreadditionssalt deraf samt farmaceutisk præparat og lægemiddel indeholdende mindst én af disse forbindelser DK170533B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8610709 1986-07-23
FR8610709A FR2601952B1 (fr) 1986-07-23 1986-07-23 Nouveaux derives amino alkyl thio de triazolopyridine ou triazoloquinoline, leurs procedes de preparation, medicaments les contenant, utiles notamment comme antalgiques

Publications (3)

Publication Number Publication Date
DK84093D0 DK84093D0 (da) 1993-07-14
DK84093A true DK84093A (da) 1993-07-14
DK170533B1 DK170533B1 (da) 1995-10-16

Family

ID=9337681

Family Applications (2)

Application Number Title Priority Date Filing Date
DK382987A DK170472B1 (da) 1986-07-23 1987-07-22 Aminoalkylthioderivater af triazolopyridin eller triazoloquinolin og syreadditionssalte deraf samt deres fremstilling og farmaceutisk præparat og lægemiddel indeholdende dem
DK084093A DK170533B1 (da) 1986-07-23 1993-07-14 4-(2,4-Difluorphenyl)-piperazin eller et syreadditionssalt deraf samt farmaceutisk præparat og lægemiddel indeholdende mindst én af disse forbindelser

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK382987A DK170472B1 (da) 1986-07-23 1987-07-22 Aminoalkylthioderivater af triazolopyridin eller triazoloquinolin og syreadditionssalte deraf samt deres fremstilling og farmaceutisk præparat og lægemiddel indeholdende dem

Country Status (18)

Country Link
US (1) US4886805A (da)
EP (1) EP0254623B1 (da)
JP (1) JP2535355B2 (da)
KR (1) KR960000358B1 (da)
AT (1) ATE90349T1 (da)
AU (1) AU601452B2 (da)
CA (2) CA1334968C (da)
DE (1) DE3786118T2 (da)
DK (2) DK170472B1 (da)
ES (1) ES2058134T3 (da)
FR (1) FR2601952B1 (da)
IE (1) IE60116B1 (da)
IL (1) IL83206A0 (da)
LV (1) LV10716B (da)
NZ (1) NZ221141A (da)
PH (1) PH23791A (da)
PT (1) PT85387B (da)
ZA (1) ZA875424B (da)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2687147A1 (fr) * 1992-02-11 1993-08-13 Union Pharma Scient Appl Nouveaux derives d'alpha-amino n-pyridyl benzene propanamide, leurs procedes de preparation, compositions pharmaceutiques les contenant.
DE4425144A1 (de) * 1994-07-15 1996-01-18 Basf Ag Triazolverbindungen und deren Verwendung
US6403593B1 (en) 1995-07-14 2002-06-11 Abbott Laboratories Triazole compounds and the use thereof
DE19728996A1 (de) 1997-07-07 1999-01-14 Basf Ag Triazolverbindungen und deren Verwendung
AR022228A1 (es) 1999-01-12 2002-09-04 Abbott Gmbh & Co Kg Compuestos de triazol, composicion farmaceutica que los comprende y uso de los mismos para la preparar dicha composicion
US6989392B2 (en) 2002-06-18 2006-01-24 Abbott Laboratories 2-Aminoquinolines as melanin concentrating hormone receptor antagonists
PE20121506A1 (es) * 2006-07-14 2012-11-26 Amgen Inc Compuestos triazolopiridinas como inhibidores de c-met
US8198448B2 (en) 2006-07-14 2012-06-12 Amgen Inc. Fused heterocyclic derivatives and methods of use
US8217177B2 (en) 2006-07-14 2012-07-10 Amgen Inc. Fused heterocyclic derivatives and methods of use
EP1972628A1 (en) * 2007-03-21 2008-09-24 Schwarz Pharma Ag Indolizines and aza-analog derivatives thereof as CNS active compounds
EA201170222A1 (ru) * 2008-07-18 2011-08-30 Санофи-Авентис НОВЫЕ ПРОИЗВОДНЫЕ ТРИАЗОЛО[4,3-a]ПИРИДИНА, СПОСОБ ИХ ПОЛУЧЕНИЯ, ИХ ПРИМЕНЕНИЕ В КАЧЕСТВЕ ЛЕКАРСТВЕННЫХ СРЕДСТВ, ФАРМАЦЕВТИЧЕСКИЕ КОМПОЗИЦИИ И НОВОЕ ПРИМЕНЕНИЕ, В ЧАСТНОСТИ, В КАЧЕСТВЕ ИНГИБИТОРОВ МЕТ
FR2933980B1 (fr) * 2008-07-18 2011-07-29 Sanofi Aventis Nouveaux derives triazolo°4,3-a!pyridine, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de met
FR2941229B1 (fr) * 2009-01-21 2012-11-30 Sanofi Aventis Nouveaux derives triazolo°4,3-a!pyridine, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de met
ES2691650T3 (es) 2011-09-15 2018-11-28 Novartis Ag 3-(quinolin-6-il-tio)-[1,2,4]-triazolo-[4,3-a]-piridinas 6-sustituidas como inhibidores de tirosina quinasa c-Met
GB201321742D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
CN105541702B (zh) * 2016-01-27 2019-10-22 宜春学院 类卢扎朵仑结构的芳胺基烷基硫类化合物及其制备方法
KR102230681B1 (ko) 2019-10-17 2021-03-22 주식회사 포스코건설 태그유닛 및 이를 포함하는 진동측정장치

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3050525A (en) * 1960-12-14 1962-08-21 John B Bicking Certain derivatives of s-triazolo [4, 3-a]-pyridine
US4244953A (en) * 1979-10-24 1981-01-13 American Cyanamid Company Substituted 6-phenyl-5,6,7,8-tetrahydro-1,2,4-triazolo-[4,3-a]pyridines
US4340597A (en) * 1981-04-13 1982-07-20 Schering Corporation 1-Substituted-4-aryl-1,2,5,6-tetrahydro and hexahydropyridines
US4358454A (en) * 1982-01-08 1982-11-09 Schering Corporation 1,3,4-Triazolo[1,5-a]pyridines
US4358453A (en) * 1982-01-08 1982-11-09 Schering Corporation 1,2,4-Triazolo[4,3-a]pyridines
US4419516A (en) * 1982-06-16 1983-12-06 American Home Products Corporation Antiviral imidazo- and triazolo-pyridines
JPH0439094A (ja) * 1990-06-06 1992-02-10 Fuji Photo Film Co Ltd 直描型平版印刷用原版

Also Published As

Publication number Publication date
KR960000358B1 (ko) 1996-01-05
EP0254623B1 (fr) 1993-06-09
AU601452B2 (en) 1990-09-13
FR2601952B1 (fr) 1988-11-25
KR880001650A (ko) 1988-04-25
ZA875424B (en) 1988-04-27
DK84093D0 (da) 1993-07-14
IE60116B1 (en) 1994-06-01
JPS6335572A (ja) 1988-02-16
DK170472B1 (da) 1995-09-11
CA1334968C (en) 1995-03-28
FR2601952A1 (fr) 1988-01-29
DK382987A (da) 1988-01-24
DK170533B1 (da) 1995-10-16
DE3786118T2 (de) 1993-10-28
AU7616387A (en) 1988-01-28
EP0254623A1 (fr) 1988-01-27
JP2535355B2 (ja) 1996-09-18
PT85387B (pt) 1990-04-30
DK382987D0 (da) 1987-07-22
IL83206A0 (en) 1987-12-31
LV10716B (en) 1995-12-20
IE871880L (en) 1988-01-23
DE3786118D1 (de) 1993-07-15
PT85387A (fr) 1987-08-01
ATE90349T1 (de) 1993-06-15
PH23791A (en) 1989-11-03
CA1338908C (en) 1997-02-11
NZ221141A (en) 1990-05-28
LV10716A (lv) 1995-06-20
US4886805A (en) 1989-12-12
ES2058134T3 (es) 1994-11-01

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PBP Patent lapsed