DE3786118D1 - Aminoalkylthio-triazolopyridin- oder triazolochinolinderivate, verfahren zu ihrer herstellung, diese enthaltende arzneimittel, brauchbar als antalgikum. - Google Patents

Aminoalkylthio-triazolopyridin- oder triazolochinolinderivate, verfahren zu ihrer herstellung, diese enthaltende arzneimittel, brauchbar als antalgikum.

Info

Publication number
DE3786118D1
DE3786118D1 DE8787401585T DE3786118T DE3786118D1 DE 3786118 D1 DE3786118 D1 DE 3786118D1 DE 8787401585 T DE8787401585 T DE 8787401585T DE 3786118 T DE3786118 T DE 3786118T DE 3786118 D1 DE3786118 D1 DE 3786118D1
Authority
DE
Germany
Prior art keywords
heterocycle
phenyl
ring
lower alkyl
atoms
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE8787401585T
Other languages
English (en)
Other versions
DE3786118T2 (de
Inventor
Nicole Bru-Magniez
Jean-Marie Teulon
Michele Launay
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
UNION PHARMA SCIENT APPL
UPSA SAS
Original Assignee
UNION PHARMA SCIENT APPL
UPSA SAS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by UNION PHARMA SCIENT APPL, UPSA SAS filed Critical UNION PHARMA SCIENT APPL
Application granted granted Critical
Publication of DE3786118D1 publication Critical patent/DE3786118D1/de
Publication of DE3786118T2 publication Critical patent/DE3786118T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DE87401585T 1986-07-23 1987-07-07 Aminoalkylthio-Triazolopyridin- oder Triazolochinolinderivate, Verfahren zu ihrer Herstellung, diese enthaltende Arzneimittel, brauchbar als Antalgikum. Expired - Fee Related DE3786118T2 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8610709A FR2601952B1 (fr) 1986-07-23 1986-07-23 Nouveaux derives amino alkyl thio de triazolopyridine ou triazoloquinoline, leurs procedes de preparation, medicaments les contenant, utiles notamment comme antalgiques

Publications (2)

Publication Number Publication Date
DE3786118D1 true DE3786118D1 (de) 1993-07-15
DE3786118T2 DE3786118T2 (de) 1993-10-28

Family

ID=9337681

Family Applications (1)

Application Number Title Priority Date Filing Date
DE87401585T Expired - Fee Related DE3786118T2 (de) 1986-07-23 1987-07-07 Aminoalkylthio-Triazolopyridin- oder Triazolochinolinderivate, Verfahren zu ihrer Herstellung, diese enthaltende Arzneimittel, brauchbar als Antalgikum.

Country Status (18)

Country Link
US (1) US4886805A (de)
EP (1) EP0254623B1 (de)
JP (1) JP2535355B2 (de)
KR (1) KR960000358B1 (de)
AT (1) ATE90349T1 (de)
AU (1) AU601452B2 (de)
CA (2) CA1334968C (de)
DE (1) DE3786118T2 (de)
DK (2) DK170472B1 (de)
ES (1) ES2058134T3 (de)
FR (1) FR2601952B1 (de)
IE (1) IE60116B1 (de)
IL (1) IL83206A0 (de)
LV (1) LV10716B (de)
NZ (1) NZ221141A (de)
PH (1) PH23791A (de)
PT (1) PT85387B (de)
ZA (1) ZA875424B (de)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2687147A1 (fr) * 1992-02-11 1993-08-13 Union Pharma Scient Appl Nouveaux derives d'alpha-amino n-pyridyl benzene propanamide, leurs procedes de preparation, compositions pharmaceutiques les contenant.
DE4425144A1 (de) * 1994-07-15 1996-01-18 Basf Ag Triazolverbindungen und deren Verwendung
US6403593B1 (en) 1995-07-14 2002-06-11 Abbott Laboratories Triazole compounds and the use thereof
DE19728996A1 (de) 1997-07-07 1999-01-14 Basf Ag Triazolverbindungen und deren Verwendung
AR022228A1 (es) 1999-01-12 2002-09-04 Abbott Gmbh & Co Kg Compuestos de triazol, composicion farmaceutica que los comprende y uso de los mismos para la preparar dicha composicion
US6989392B2 (en) 2002-06-18 2006-01-24 Abbott Laboratories 2-Aminoquinolines as melanin concentrating hormone receptor antagonists
PE20121506A1 (es) * 2006-07-14 2012-11-26 Amgen Inc Compuestos triazolopiridinas como inhibidores de c-met
US8198448B2 (en) 2006-07-14 2012-06-12 Amgen Inc. Fused heterocyclic derivatives and methods of use
US8217177B2 (en) 2006-07-14 2012-07-10 Amgen Inc. Fused heterocyclic derivatives and methods of use
EP1972628A1 (de) * 2007-03-21 2008-09-24 Schwarz Pharma Ag Indolizine und aza-analoge Derivate davon als CNS-aktive Verbindungen
EA201170222A1 (ru) * 2008-07-18 2011-08-30 Санофи-Авентис НОВЫЕ ПРОИЗВОДНЫЕ ТРИАЗОЛО[4,3-a]ПИРИДИНА, СПОСОБ ИХ ПОЛУЧЕНИЯ, ИХ ПРИМЕНЕНИЕ В КАЧЕСТВЕ ЛЕКАРСТВЕННЫХ СРЕДСТВ, ФАРМАЦЕВТИЧЕСКИЕ КОМПОЗИЦИИ И НОВОЕ ПРИМЕНЕНИЕ, В ЧАСТНОСТИ, В КАЧЕСТВЕ ИНГИБИТОРОВ МЕТ
FR2933980B1 (fr) * 2008-07-18 2011-07-29 Sanofi Aventis Nouveaux derives triazolo°4,3-a!pyridine, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de met
FR2941229B1 (fr) * 2009-01-21 2012-11-30 Sanofi Aventis Nouveaux derives triazolo°4,3-a!pyridine, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de met
ES2691650T3 (es) 2011-09-15 2018-11-28 Novartis Ag 3-(quinolin-6-il-tio)-[1,2,4]-triazolo-[4,3-a]-piridinas 6-sustituidas como inhibidores de tirosina quinasa c-Met
GB201321742D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
CN105541702B (zh) * 2016-01-27 2019-10-22 宜春学院 类卢扎朵仑结构的芳胺基烷基硫类化合物及其制备方法
KR102230681B1 (ko) 2019-10-17 2021-03-22 주식회사 포스코건설 태그유닛 및 이를 포함하는 진동측정장치

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3050525A (en) * 1960-12-14 1962-08-21 John B Bicking Certain derivatives of s-triazolo [4, 3-a]-pyridine
US4244953A (en) * 1979-10-24 1981-01-13 American Cyanamid Company Substituted 6-phenyl-5,6,7,8-tetrahydro-1,2,4-triazolo-[4,3-a]pyridines
US4340597A (en) * 1981-04-13 1982-07-20 Schering Corporation 1-Substituted-4-aryl-1,2,5,6-tetrahydro and hexahydropyridines
US4358454A (en) * 1982-01-08 1982-11-09 Schering Corporation 1,3,4-Triazolo[1,5-a]pyridines
US4358453A (en) * 1982-01-08 1982-11-09 Schering Corporation 1,2,4-Triazolo[4,3-a]pyridines
US4419516A (en) * 1982-06-16 1983-12-06 American Home Products Corporation Antiviral imidazo- and triazolo-pyridines
JPH0439094A (ja) * 1990-06-06 1992-02-10 Fuji Photo Film Co Ltd 直描型平版印刷用原版

Also Published As

Publication number Publication date
KR960000358B1 (ko) 1996-01-05
EP0254623B1 (de) 1993-06-09
AU601452B2 (en) 1990-09-13
FR2601952B1 (fr) 1988-11-25
KR880001650A (ko) 1988-04-25
ZA875424B (en) 1988-04-27
DK84093D0 (da) 1993-07-14
IE60116B1 (en) 1994-06-01
JPS6335572A (ja) 1988-02-16
DK170472B1 (da) 1995-09-11
CA1334968C (en) 1995-03-28
FR2601952A1 (fr) 1988-01-29
DK382987A (da) 1988-01-24
DK84093A (da) 1993-07-14
DK170533B1 (da) 1995-10-16
DE3786118T2 (de) 1993-10-28
AU7616387A (en) 1988-01-28
EP0254623A1 (de) 1988-01-27
JP2535355B2 (ja) 1996-09-18
PT85387B (pt) 1990-04-30
DK382987D0 (da) 1987-07-22
IL83206A0 (en) 1987-12-31
LV10716B (en) 1995-12-20
IE871880L (en) 1988-01-23
PT85387A (fr) 1987-08-01
ATE90349T1 (de) 1993-06-15
PH23791A (en) 1989-11-03
CA1338908C (en) 1997-02-11
NZ221141A (en) 1990-05-28
LV10716A (lv) 1995-06-20
US4886805A (en) 1989-12-12
ES2058134T3 (es) 1994-11-01

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Legal Events

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8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee