DK382987A - Aminoalkylthioderivater af triazolopyridin eller triazoloquinolin og syreadditionssalte deraf samt deres fremstilling og anvendelse - Google Patents

Aminoalkylthioderivater af triazolopyridin eller triazoloquinolin og syreadditionssalte deraf samt deres fremstilling og anvendelse

Info

Publication number
DK382987A
DK382987A DK382987A DK382987A DK382987A DK 382987 A DK382987 A DK 382987A DK 382987 A DK382987 A DK 382987A DK 382987 A DK382987 A DK 382987A DK 382987 A DK382987 A DK 382987A
Authority
DK
Denmark
Prior art keywords
heterocycle
phenyl
acid addition
addition salts
ring
Prior art date
Application number
DK382987A
Other languages
English (en)
Other versions
DK382987D0 (da
DK170472B1 (da
Inventor
Nicole Bru-Magniez
Jean-Marie Teulon
Michele Launay
Original Assignee
Carpibem
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Carpibem filed Critical Carpibem
Publication of DK382987D0 publication Critical patent/DK382987D0/da
Publication of DK382987A publication Critical patent/DK382987A/da
Application granted granted Critical
Publication of DK170472B1 publication Critical patent/DK170472B1/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DK382987A 1986-07-23 1987-07-22 Aminoalkylthioderivater af triazolopyridin eller triazoloquinolin og syreadditionssalte deraf samt deres fremstilling og farmaceutisk præparat og lægemiddel indeholdende dem DK170472B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8610709 1986-07-23
FR8610709A FR2601952B1 (fr) 1986-07-23 1986-07-23 Nouveaux derives amino alkyl thio de triazolopyridine ou triazoloquinoline, leurs procedes de preparation, medicaments les contenant, utiles notamment comme antalgiques

Publications (3)

Publication Number Publication Date
DK382987D0 DK382987D0 (da) 1987-07-22
DK382987A true DK382987A (da) 1988-01-24
DK170472B1 DK170472B1 (da) 1995-09-11

Family

ID=9337681

Family Applications (2)

Application Number Title Priority Date Filing Date
DK382987A DK170472B1 (da) 1986-07-23 1987-07-22 Aminoalkylthioderivater af triazolopyridin eller triazoloquinolin og syreadditionssalte deraf samt deres fremstilling og farmaceutisk præparat og lægemiddel indeholdende dem
DK084093A DK170533B1 (da) 1986-07-23 1993-07-14 4-(2,4-Difluorphenyl)-piperazin eller et syreadditionssalt deraf samt farmaceutisk præparat og lægemiddel indeholdende mindst én af disse forbindelser

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK084093A DK170533B1 (da) 1986-07-23 1993-07-14 4-(2,4-Difluorphenyl)-piperazin eller et syreadditionssalt deraf samt farmaceutisk præparat og lægemiddel indeholdende mindst én af disse forbindelser

Country Status (18)

Country Link
US (1) US4886805A (da)
EP (1) EP0254623B1 (da)
JP (1) JP2535355B2 (da)
KR (1) KR960000358B1 (da)
AT (1) ATE90349T1 (da)
AU (1) AU601452B2 (da)
CA (2) CA1334968C (da)
DE (1) DE3786118T2 (da)
DK (2) DK170472B1 (da)
ES (1) ES2058134T3 (da)
FR (1) FR2601952B1 (da)
IE (1) IE60116B1 (da)
IL (1) IL83206A0 (da)
LV (1) LV10716B (da)
NZ (1) NZ221141A (da)
PH (1) PH23791A (da)
PT (1) PT85387B (da)
ZA (1) ZA875424B (da)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2687147A1 (fr) * 1992-02-11 1993-08-13 Union Pharma Scient Appl Nouveaux derives d'alpha-amino n-pyridyl benzene propanamide, leurs procedes de preparation, compositions pharmaceutiques les contenant.
DE4425144A1 (de) * 1994-07-15 1996-01-18 Basf Ag Triazolverbindungen und deren Verwendung
US6403593B1 (en) 1995-07-14 2002-06-11 Abbott Laboratories Triazole compounds and the use thereof
DE19728996A1 (de) 1997-07-07 1999-01-14 Basf Ag Triazolverbindungen und deren Verwendung
AR022230A1 (es) 1999-01-12 2002-09-04 Abbott Gmbh & Co Kg Compuestos de triazol, composicion farmaceutica que los comprende y uso de los mismos para preparar dicha composicion
US6989392B2 (en) 2002-06-18 2006-01-24 Abbott Laboratories 2-Aminoquinolines as melanin concentrating hormone receptor antagonists
US8198448B2 (en) 2006-07-14 2012-06-12 Amgen Inc. Fused heterocyclic derivatives and methods of use
PE20080403A1 (es) * 2006-07-14 2008-04-25 Amgen Inc Derivados heterociclicos fusionados y metodos de uso
US8217177B2 (en) 2006-07-14 2012-07-10 Amgen Inc. Fused heterocyclic derivatives and methods of use
EP1972628A1 (en) * 2007-03-21 2008-09-24 Schwarz Pharma Ag Indolizines and aza-analog derivatives thereof as CNS active compounds
AU2009272516A1 (en) * 2008-07-18 2010-01-21 Sanofi-Aventis Novel triazolo(4,3-a)pyridine derivatives, process for the preparation thereof, use thereof as medicaments, pharmaceutical compositions and novel use, in particular as MET inhibitors
FR2941229B1 (fr) * 2009-01-21 2012-11-30 Sanofi Aventis Nouveaux derives triazolo°4,3-a!pyridine, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de met
FR2933980B1 (fr) * 2008-07-18 2011-07-29 Sanofi Aventis Nouveaux derives triazolo°4,3-a!pyridine, leur procede de preparation, leur application a titre de medicaments, compositions pharmaceutiques et nouvelle utilisation notamment comme inhibiteurs de met
EP2755976B1 (en) 2011-09-15 2018-07-18 Novartis AG 6-substituted 3-(quinolin-6-ylthio)-[1,2,4]triazolo[4,3-a]pyridines as c-met tyrosine kinase inhibitors
GB201321742D0 (en) * 2013-12-09 2014-01-22 Ucb Pharma Sa Therapeutic agents
CN105541702B (zh) * 2016-01-27 2019-10-22 宜春学院 类卢扎朵仑结构的芳胺基烷基硫类化合物及其制备方法
KR102230681B1 (ko) 2019-10-17 2021-03-22 주식회사 포스코건설 태그유닛 및 이를 포함하는 진동측정장치

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3050525A (en) * 1960-12-14 1962-08-21 John B Bicking Certain derivatives of s-triazolo [4, 3-a]-pyridine
US4244953A (en) * 1979-10-24 1981-01-13 American Cyanamid Company Substituted 6-phenyl-5,6,7,8-tetrahydro-1,2,4-triazolo-[4,3-a]pyridines
US4340597A (en) * 1981-04-13 1982-07-20 Schering Corporation 1-Substituted-4-aryl-1,2,5,6-tetrahydro and hexahydropyridines
US4358453A (en) * 1982-01-08 1982-11-09 Schering Corporation 1,2,4-Triazolo[4,3-a]pyridines
US4358454A (en) * 1982-01-08 1982-11-09 Schering Corporation 1,3,4-Triazolo[1,5-a]pyridines
US4419516A (en) * 1982-06-16 1983-12-06 American Home Products Corporation Antiviral imidazo- and triazolo-pyridines
JPH0439094A (ja) * 1990-06-06 1992-02-10 Fuji Photo Film Co Ltd 直描型平版印刷用原版

Also Published As

Publication number Publication date
EP0254623A1 (fr) 1988-01-27
IE871880L (en) 1988-01-23
PT85387A (fr) 1987-08-01
DK84093A (da) 1993-07-14
LV10716A (lv) 1995-06-20
DK382987D0 (da) 1987-07-22
AU7616387A (en) 1988-01-28
FR2601952A1 (fr) 1988-01-29
CA1334968C (en) 1995-03-28
ES2058134T3 (es) 1994-11-01
JPS6335572A (ja) 1988-02-16
DK84093D0 (da) 1993-07-14
DK170533B1 (da) 1995-10-16
FR2601952B1 (fr) 1988-11-25
NZ221141A (en) 1990-05-28
IL83206A0 (en) 1987-12-31
EP0254623B1 (fr) 1993-06-09
ATE90349T1 (de) 1993-06-15
IE60116B1 (en) 1994-06-01
KR960000358B1 (ko) 1996-01-05
PT85387B (pt) 1990-04-30
DE3786118T2 (de) 1993-10-28
CA1338908C (en) 1997-02-11
US4886805A (en) 1989-12-12
DE3786118D1 (de) 1993-07-15
LV10716B (en) 1995-12-20
AU601452B2 (en) 1990-09-13
PH23791A (en) 1989-11-03
DK170472B1 (da) 1995-09-11
ZA875424B (en) 1988-04-27
JP2535355B2 (ja) 1996-09-18
KR880001650A (ko) 1988-04-25

Similar Documents

Publication Publication Date Title
DK382987A (da) Aminoalkylthioderivater af triazolopyridin eller triazoloquinolin og syreadditionssalte deraf samt deres fremstilling og anvendelse
AR010331A1 (es) Compuestos derivados de 6-fenilpiridil-2-amina utiles como inhibidores nos, composiciones farmaceuticas que comprenden dichos compuestos, y metodosde tratamiento utilizando dichos compuestos.
NO953447D0 (no) Nye 4-aminopyridiner, fremgangsmåte for deres fremstilling samt legemidler inneholdende disse
ES2066875T3 (es) Aminoalquilindoles, procedimiento para su obtencion y preparados farmaceuticos que los contienen.
IE891797L (en) 4-amino quinolines and naphthyridines, process for their¹preparation and their use as medicines
HUP9802534A2 (hu) Neurotranszmitter újrafelvételt gátló kondenzált tropánszármazékok és előállításuk, e vegyületeket tartalmazó gyógyászati készítmények, valamint e vegyületek alkalmazása
KR850006400A (ko) 1,7-디아미노-1,4-디하이드로-4-옥소-3-(아자)퀴놀린-카복실산의 제조방법
DK12087D0 (da) Decahydroquinolinderivater, deres fremstilling og anvendelse samt praeparater med indhold deraf
ATE9336T1 (de) 3,1-benzoxazin-2-one, ihre herstellung und verwendung.
DK393486A (da) Dihydropyridin-derivater og fremgangsmaade til fremstilling deraf
NO850315L (no) Fremgangsmaate for fremstilling av metylendifosfonsyre-derivater med antireumatiske egenskaper
DE68913365T2 (de) 4-Amino-3-carboxynaphthyridin-Derivate, ihre Herstellung und pharmazeutische Zusammensetzungen.
KR850005433A (ko) 나프티리딘 및 피리도피리미딘 화합물의 제조방법
IL111375A (en) N-substituted azabicycloalkane derivatives and pharmaceutical compositions containing them
ES488370A0 (es) Un procedimiento para la preparacion de derivados de 2-hidroxinaftaleno.
SE7713968L (sv) Basiskt alkylerade ditiosalicylsyraamider, sett for framstellning derav samt anvendning derav som lekemedel
PT85300A (fr) Procede de preparation de nouveaux derives de la piperazine dione-2,6
IL69931A (en) N-(6-chloro-pyrazin-2-yl)-4-hydroxy-2h-1,2-benzothiazine-3-carboxamide-1,1-dioxides,their preparation and pharmaceutical compositions containing them
ATE33134T1 (de) 2-aminoethyl-pyridin oder pyrazin-derivate, ihre herstellung und diese enthaltende pharmazeutische zusammensetzungen.
ES2038780T3 (es) Procedimiento para la preparacion de nuevos compuestos triciclicos.
SE8003394L (sv) Nytt sett att framstella 6-(substituerad amino)-3-pyridazinylhydrazin
ATE28192T1 (de) 4-alkylimidazol-derivate, ihre herstellung und verwendung.

Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PBP Patent lapsed