PE20151654A1 - Inhibidores de cdc7 - Google Patents
Inhibidores de cdc7Info
- Publication number
- PE20151654A1 PE20151654A1 PE2015001925A PE2015001925A PE20151654A1 PE 20151654 A1 PE20151654 A1 PE 20151654A1 PE 2015001925 A PE2015001925 A PE 2015001925A PE 2015001925 A PE2015001925 A PE 2015001925A PE 20151654 A1 PE20151654 A1 PE 20151654A1
- Authority
- PE
- Peru
- Prior art keywords
- cdc7 inhibitors
- cdc7
- inhibitors
- isoindolinone
- cancer
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Hematology (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Epidemiology (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201361782798P | 2013-03-14 | 2013-03-14 | |
US201361789108P | 2013-03-15 | 2013-03-15 |
Publications (1)
Publication Number | Publication Date |
---|---|
PE20151654A1 true PE20151654A1 (es) | 2015-11-12 |
Family
ID=50382704
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PE2015001925A PE20151654A1 (es) | 2013-03-14 | 2014-03-07 | Inhibidores de cdc7 |
Country Status (37)
Country | Link |
---|---|
US (1) | US9156824B2 (de) |
EP (1) | EP2970221B1 (de) |
JP (1) | JP6064079B2 (de) |
KR (1) | KR101718645B1 (de) |
CN (1) | CN105008351B (de) |
AP (1) | AP2015008734A0 (de) |
AU (1) | AU2014228374B2 (de) |
BR (1) | BR112015020466B1 (de) |
CA (1) | CA2900773C (de) |
CL (1) | CL2015002530A1 (de) |
CR (1) | CR20150416A (de) |
CY (1) | CY1119199T1 (de) |
DK (1) | DK2970221T3 (de) |
EA (1) | EA027012B1 (de) |
ES (1) | ES2639793T3 (de) |
GT (1) | GT201500263A (de) |
HK (1) | HK1212696A1 (de) |
HR (1) | HRP20171151T1 (de) |
HU (1) | HUE033482T2 (de) |
IL (1) | IL240962B (de) |
JO (1) | JO3383B1 (de) |
LT (1) | LT2970221T (de) |
ME (1) | ME02805B (de) |
MX (1) | MX363438B (de) |
MY (1) | MY188145A (de) |
NZ (1) | NZ710392A (de) |
PE (1) | PE20151654A1 (de) |
PH (1) | PH12015502091B1 (de) |
PL (1) | PL2970221T3 (de) |
PT (1) | PT2970221T (de) |
RS (1) | RS56122B1 (de) |
SG (1) | SG11201507541PA (de) |
SI (1) | SI2970221T1 (de) |
TN (1) | TN2015000349A1 (de) |
TW (1) | TWI622396B (de) |
UA (1) | UA116125C2 (de) |
WO (1) | WO2014143601A1 (de) |
Families Citing this family (26)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK2906555T3 (en) * | 2012-10-15 | 2017-02-06 | Pfizer Ireland Pharmaceuticals | Process for the preparation of voriconazole and analogs thereof |
CA2897200C (en) | 2013-01-14 | 2021-07-06 | Incyte Corporation | Bicyclic aromatic carboxamide compounds useful as pim kinase inhibitors |
ES2790419T3 (es) | 2013-01-15 | 2020-10-27 | Incyte Holdings Corp | Los compuestos de tiazolcarboxamidas y piridinacarboxamida útiles como inhibidores de quinasa de PIM |
ES2689526T3 (es) | 2013-03-14 | 2018-11-14 | Janssen Pharmaceutica Nv | Moduladores de P2X7 |
TWI599567B (zh) | 2013-03-14 | 2017-09-21 | 健生藥品公司 | P2x7調節劑 |
JO3509B1 (ar) | 2013-03-14 | 2020-07-05 | Janssen Pharmaceutica Nv | معدلات p2x7 |
JP6294953B2 (ja) | 2013-03-14 | 2018-03-14 | ヤンセン ファーマシューティカ エヌ.ベー. | P2x7調節物質 |
AU2014230814B2 (en) | 2013-03-14 | 2017-12-21 | Boehringer Ingelheim International Gmbh | Substituted 2-Aza-bicyclo[2.2.1]heptane-3-carboxylic acid (benzyl-cyano-methyl)-amides inhibitors of Cathepsin C |
TW201605866A (zh) | 2013-08-23 | 2016-02-16 | 英塞特公司 | 可用作pim激酶抑制劑之呋喃并-及噻吩并-吡啶甲醯胺化合物 |
WO2016010897A1 (en) | 2014-07-14 | 2016-01-21 | Incyte Corporation | Bicyclic heteroaromatic carboxamide compounds useful as pim kinase inhibitors |
US9580418B2 (en) | 2014-07-14 | 2017-02-28 | Incyte Corporation | Bicyclic aromatic carboxamide compounds useful as Pim kinase inhibitors |
EP3191492B1 (de) | 2014-09-12 | 2019-01-09 | Janssen Pharmaceutica NV | P2x7-modulatoren |
MY188382A (en) | 2014-09-12 | 2021-12-07 | Boehringer Ingelheim Int | Spirocyclic inhibitors of cathepsin c |
WO2016196244A1 (en) | 2015-05-29 | 2016-12-08 | Incyte Corporation | Pyridineamine compounds useful as pim kinase inhibitors |
TWI734699B (zh) | 2015-09-09 | 2021-08-01 | 美商英塞特公司 | Pim激酶抑制劑之鹽 |
TW201718546A (zh) | 2015-10-02 | 2017-06-01 | 英塞特公司 | 適用作pim激酶抑制劑之雜環化合物 |
CN110036006B (zh) * | 2016-09-22 | 2022-12-13 | 癌症研究科技有限公司 | 嘧啶酮衍生物的制备和用途 |
TW201924683A (zh) | 2017-12-08 | 2019-07-01 | 美商英塞特公司 | 用於治療骨髓增生性贅瘤的低劑量組合療法 |
CN108383771A (zh) * | 2018-01-08 | 2018-08-10 | 华东师范大学 | 手性3,3-二取代异吲哚啉-1-酮衍生物及其合成方法和应用 |
GB201807147D0 (en) | 2018-05-01 | 2018-06-13 | Oncologica Uk Ltd | Therapeutic combination |
NL2021185B1 (en) | 2018-06-26 | 2020-01-06 | Stichting Het Nederlands Kanker Inst Antoni Van Leeuwenhoek Ziekenhuis | Combination Therapy and Use Thereof for Treating Cancer |
MX2021003661A (es) | 2018-09-28 | 2021-08-19 | Janssen Pharmaceutica Nv | Moduladores de la monoacilglicerol lipasa. |
MA53721A (fr) | 2018-09-28 | 2021-09-15 | Janssen Pharmaceutica Nv | Modulateurs de la monoacylglycérol lipase |
US20220220125A1 (en) * | 2019-04-16 | 2022-07-14 | Janssen Pharmaceutica Nv | Fused isoindolin-1-one derivatives useful as grk2 inhibitors |
JP2022550767A (ja) | 2019-09-30 | 2022-12-05 | ヤンセン ファーマシューティカ エヌ.ベー. | 放射線標識されたmgl petリガンド |
EP4126860A1 (de) | 2020-03-26 | 2023-02-08 | Janssen Pharmaceutica NV | Monoacylglycerol-lipasemodulatoren |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SE0400970D0 (sv) * | 2004-04-14 | 2004-04-14 | Astrazeneca Ab | Nicotinic acetylcholine receptor ligands |
TW200639163A (en) * | 2005-02-04 | 2006-11-16 | Genentech Inc | RAF inhibitor compounds and methods |
US7576082B2 (en) * | 2005-06-24 | 2009-08-18 | Hoffman-La Roche Inc. | Oxindole derivatives |
EP2073806B1 (de) * | 2006-10-12 | 2012-02-15 | Xenon Pharmaceuticals Inc. | Verwendung von spiro-oxindol-verbindungen als therapeutika |
KR20100032886A (ko) * | 2007-06-08 | 2010-03-26 | 아보트 러보러터리즈 | 키나제 억제제로서의 5-헤테로아릴 치환된 인다졸 |
US8648069B2 (en) * | 2007-06-08 | 2014-02-11 | Abbvie Inc. | 5-substituted indazoles as kinase inhibitors |
-
2014
- 2014-03-04 JO JOP/2014/0067A patent/JO3383B1/ar active
- 2014-03-05 TW TW103107546A patent/TWI622396B/zh active
- 2014-03-07 AP AP2015008734A patent/AP2015008734A0/xx unknown
- 2014-03-07 PL PL14712966T patent/PL2970221T3/pl unknown
- 2014-03-07 RS RS20170791A patent/RS56122B1/sr unknown
- 2014-03-07 UA UAA201508675A patent/UA116125C2/uk unknown
- 2014-03-07 HU HUE14712966A patent/HUE033482T2/en unknown
- 2014-03-07 LT LTEP14712966.2T patent/LT2970221T/lt unknown
- 2014-03-07 EP EP14712966.2A patent/EP2970221B1/de active Active
- 2014-03-07 CN CN201480011202.4A patent/CN105008351B/zh active Active
- 2014-03-07 ES ES14712966.2T patent/ES2639793T3/es active Active
- 2014-03-07 SG SG11201507541PA patent/SG11201507541PA/en unknown
- 2014-03-07 CA CA2900773A patent/CA2900773C/en active Active
- 2014-03-07 MY MYPI2015703062A patent/MY188145A/en unknown
- 2014-03-07 SI SI201430280T patent/SI2970221T1/sl unknown
- 2014-03-07 MX MX2015012583A patent/MX363438B/es unknown
- 2014-03-07 PE PE2015001925A patent/PE20151654A1/es active IP Right Grant
- 2014-03-07 NZ NZ710392A patent/NZ710392A/en unknown
- 2014-03-07 AU AU2014228374A patent/AU2014228374B2/en active Active
- 2014-03-07 KR KR1020157024644A patent/KR101718645B1/ko not_active Application Discontinuation
- 2014-03-07 WO PCT/US2014/021466 patent/WO2014143601A1/en active Application Filing
- 2014-03-07 BR BR112015020466-0A patent/BR112015020466B1/pt active IP Right Grant
- 2014-03-07 ME MEP-2017-173A patent/ME02805B/de unknown
- 2014-03-07 JP JP2016500764A patent/JP6064079B2/ja active Active
- 2014-03-07 EA EA201591509A patent/EA027012B1/ru not_active IP Right Cessation
- 2014-03-07 DK DK14712966.2T patent/DK2970221T3/en active
- 2014-03-07 PT PT147129662T patent/PT2970221T/pt unknown
- 2014-03-07 US US14/200,141 patent/US9156824B2/en active Active
-
2015
- 2015-08-12 TN TN2015000349A patent/TN2015000349A1/en unknown
- 2015-08-14 CR CR20150416A patent/CR20150416A/es unknown
- 2015-08-31 IL IL240962A patent/IL240962B/en active IP Right Grant
- 2015-09-09 CL CL2015002530A patent/CL2015002530A1/es unknown
- 2015-09-09 GT GT201500263A patent/GT201500263A/es unknown
- 2015-09-14 PH PH12015502091A patent/PH12015502091B1/en unknown
-
2016
- 2016-01-21 HK HK16100636.2A patent/HK1212696A1/zh unknown
-
2017
- 2017-07-27 HR HRP20171151TT patent/HRP20171151T1/hr unknown
- 2017-08-10 CY CY20171100861T patent/CY1119199T1/el unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG | Grant, registration |