PE20150634A1 - Azaindolcarboxamidas y azaindoltiocarboxamidas como insecticidas y acaricidas - Google Patents

Azaindolcarboxamidas y azaindoltiocarboxamidas como insecticidas y acaricidas

Info

Publication number
PE20150634A1
PE20150634A1 PE2015000183A PE2015000183A PE20150634A1 PE 20150634 A1 PE20150634 A1 PE 20150634A1 PE 2015000183 A PE2015000183 A PE 2015000183A PE 2015000183 A PE2015000183 A PE 2015000183A PE 20150634 A1 PE20150634 A1 PE 20150634A1
Authority
PE
Peru
Prior art keywords
insecticides
ethyl
azaindoltiocarboxamides
azaindolcarboxamides
acaricides
Prior art date
Application number
PE2015000183A
Other languages
English (en)
Spanish (es)
Inventor
Markus Heil
Roland Andree
Eike Kevin Heilmann
Peter Jeschke
Matthias Riedrich
Kerstin Ilg
Ulrich Goergens
Arnd Voerste
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=46940225&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PE20150634(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of PE20150634A1 publication Critical patent/PE20150634A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N53/00—Biocides, pest repellants or attractants, or plant growth regulators containing cyclopropane carboxylic acids or derivatives thereof
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
PE2015000183A 2012-08-17 2013-08-13 Azaindolcarboxamidas y azaindoltiocarboxamidas como insecticidas y acaricidas PE20150634A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP12180826 2012-08-17

Publications (1)

Publication Number Publication Date
PE20150634A1 true PE20150634A1 (es) 2015-05-08

Family

ID=46940225

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2015000183A PE20150634A1 (es) 2012-08-17 2013-08-13 Azaindolcarboxamidas y azaindoltiocarboxamidas como insecticidas y acaricidas

Country Status (17)

Country Link
US (1) US9345247B2 (enExample)
EP (1) EP2885301A1 (enExample)
JP (1) JP2015530990A (enExample)
KR (1) KR20150044895A (enExample)
CN (1) CN104718206B (enExample)
AU (1) AU2013304133B2 (enExample)
BR (1) BR112015003098A2 (enExample)
CA (1) CA2881995A1 (enExample)
CL (1) CL2015000336A1 (enExample)
CO (1) CO7200270A2 (enExample)
IN (1) IN2015DN01061A (enExample)
MX (1) MX2015001897A (enExample)
PE (1) PE20150634A1 (enExample)
PH (1) PH12015500334A1 (enExample)
RU (1) RU2015109064A (enExample)
WO (1) WO2014026984A1 (enExample)
ZA (1) ZA201501211B (enExample)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2012178125A1 (en) 2011-06-22 2012-12-27 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of atr kinase
LT3418281T (lt) 2012-12-07 2021-01-11 Vertex Pharmaceuticals Inc. Pirazolo[1,5-a]pirimidinai, naudotini kaip atr kinazės inhibitoriai, skirti vėžinių ligų gydymui
EP2970289A1 (en) 2013-03-15 2016-01-20 Vertex Pharmaceuticals Inc. Compounds useful as inhibitors of atr kinase
WO2014143240A1 (en) 2013-03-15 2014-09-18 Vertex Pharmaceuticals Incorporated Fused pyrazolopyrimidine derivatives useful as inhibitors of atr kinase
EP2970288A1 (en) 2013-03-15 2016-01-20 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of atr kinase
HUE046727T2 (hu) 2013-12-06 2020-03-30 Vertex Pharma Az ATR-kináz inhibitoraként használható vegyület, 2-amino-6-fluoro-N-[5-fluoro-piridin-3-IL]-pirazolo-[1,5-A]-pirimidin-3-karboxamid, ennek elõállítása, különbözõ szilárd formái és ezek radioaktív nyomjelzett származékai
AR099336A1 (es) 2014-02-17 2016-07-13 Bayer Cropscience Ag Indol- y bencimidazolcarboxamidas como insecticidas y acaricidas
ES2777608T3 (es) 2014-06-05 2020-08-05 Vertex Pharma Derivados radiomarcados de un compuesto de 2-amino-6-fluoro-N-[5-fluoro-piridin-3-il]-pirazolo[1,5-a]pirimidin-3-carboxamida útiles como inhibidores de ATR cinasa, la preparación de dicho compuesto y diferentes formas sólidas del mismo
US11179394B2 (en) 2014-06-17 2021-11-23 Vertex Pharmaceuticals Incorporated Method for treating cancer using a combination of Chk1 and ATR inhibitors
CN104974075A (zh) * 2015-08-07 2015-10-14 新秀化学(烟台)有限公司 一种n, n-二(2,2,6,6-四甲基-4-哌啶基) -1,3-苯二甲酰胺的制备方法
US11464774B2 (en) 2015-09-30 2022-10-11 Vertex Pharmaceuticals Incorporated Method for treating cancer using a combination of DNA damaging agents and ATR inhibitors
TWI773657B (zh) 2015-12-18 2022-08-11 美商亞德利克斯公司 作爲非全身tgr5促效劑之經取代之4-苯基吡啶化合物
US12084472B2 (en) 2015-12-18 2024-09-10 Ardelyx, Inc. Substituted 4-phenyl pyridine compounds as non-systemic TGR5 agonists
CN107094790A (zh) * 2017-06-12 2017-08-29 刘鸿宇 一种具有协同杀虫作用的农药组合物
KR20220070491A (ko) * 2019-09-26 2022-05-31 더 글로벌 얼라이언스 포 티비 드러그 디벨롭먼트, 잉크. 미코박테리아 감염의 치료를 위한 아자인돌 카복사미드 화합물

Family Cites Families (44)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2358890A1 (fr) 1976-05-24 1978-02-17 Science Union & Cie Nouvelles aryl trifluoroethylamines, leurs procedes d'obtention et les compositions pharmaceutiques en renfermant
WO1992000964A1 (fr) 1990-07-05 1992-01-23 Nippon Soda Co., Ltd. Derive d'amine
US20040077605A1 (en) 2001-06-20 2004-04-22 Salvati Mark E. Fused heterocyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
AU2002304109B2 (en) 2001-05-31 2005-07-21 Nihon Nohyaku Co., Ltd. Substituted anilide derivatives, intermediates thereof, agricultural and horticultural chemicals, and their usage
GB0213715D0 (en) 2002-06-14 2002-07-24 Syngenta Ltd Chemical compounds
TWI312272B (en) 2003-05-12 2009-07-21 Sumitomo Chemical Co Pyrimidine compound and pests controlling composition containing the same
EP1479680A1 (en) 2003-05-19 2004-11-24 Aventis Pharma Deutschland GmbH Azaindole derivatives as Factor Xa inhibitors
EP1636224B1 (en) 2003-05-21 2010-07-14 Prosidion Limited Pyrrolopyridine-2-carboxylic acid amide inhibitors of glycogen phoshorylase
UA79404C2 (en) 2003-10-02 2007-06-11 Basf Ag 2-cyanobenzenesulfonamide for controlling pests
WO2005063694A1 (en) 2003-12-26 2005-07-14 Sumitomo Chemical Company, Limited Nitrile compound and its use in pest control
DK2256112T3 (en) 2004-02-18 2016-03-21 Ishihara Sangyo Kaisha Anthranilamides, process for their production and insecticides containing the same
BRPI0508140B1 (pt) 2004-03-05 2015-03-17 Nissan Chemical Ind Ltd Composto benzamida substituída por isoxazolina da fórmula (1); da fórmula (2) substituído por 3,5-bis (aril substituído); da fórmula (4) substituída por alquinibenzeno ou um sal do mesmo; "pesticida, agroquímico, inseticida, parasiticida contendo como ingrediente ativo um ou mais composto benzamida substituída por isoxazolina e sal do mesmo"
KR101310073B1 (ko) 2004-10-20 2013-09-24 이하라케미칼 고교가부시키가이샤 3-트리아졸릴페닐설파이드 유도체 및 그것을유효성분으로서 함유하는 살충·살진드기·살선충제
DE102005008021A1 (de) 2005-02-22 2006-08-24 Bayer Cropscience Ag Spiroketal-substituierte cyclische Ketoenole
AU2006226300A1 (en) 2005-03-24 2006-09-28 Basf Aktiengesellschaft 2-cyanobenzenesulfonamide compounds for seed treatment
EP1932844B1 (en) 2005-10-06 2015-09-02 Nippon Soda Co., Ltd. Cross-linked cyclic amine compounds and agents for pest control
PT2404919E (pt) 2005-11-08 2013-10-22 Vertex Pharma Composto heterocíclico útil como um modulador de transportadores de cassete de ligação a atp
US7622466B2 (en) 2005-11-18 2009-11-24 Hoffman-La Roche Inc. Azaindole-2-carboxamide derivatives
EP1954138A2 (en) 2005-11-21 2008-08-13 Basf Se Insecticidal methods using 3-amino-1,2-benzisothiazole derivatives
TW200803740A (en) 2005-12-16 2008-01-16 Du Pont 5-aryl isoxazolines for controlling invertebrate pests
EP1997820A4 (en) 2006-03-09 2009-03-04 Univ East China Science & Tech METHOD OF MANUFACTURE AND USE OF COMPOUNDS HAVING HIGH BIOZIDER EFFECT
DE102006015467A1 (de) 2006-03-31 2007-10-04 Bayer Cropscience Ag Substituierte Enaminocarbonylverbindungen
DE102006015470A1 (de) 2006-03-31 2007-10-04 Bayer Cropscience Ag Substituierte Enaminocarbonylverbindungen
DE102006015468A1 (de) 2006-03-31 2007-10-04 Bayer Cropscience Ag Substituierte Enaminocarbonylverbindungen
TWI381811B (zh) 2006-06-23 2013-01-11 Dow Agrosciences Llc 用以防治可抵抗一般殺蟲劑之昆蟲的方法
DE102006033572A1 (de) 2006-07-20 2008-01-24 Bayer Cropscience Ag N'-Cyano-N-halogenalkyl-imidamid Derivate
ATE539080T1 (de) 2006-11-30 2012-01-15 Meiji Seika Pharma Co Ltd Schädlingsbekämpfungsmittel
DE102006057036A1 (de) 2006-12-04 2008-06-05 Bayer Cropscience Ag Biphenylsubstituierte spirocyclische Ketoenole
WO2008104503A1 (en) 2007-03-01 2008-09-04 Basf Se Pesticidal active mixtures comprising aminothiazoline compounds
CN101842098A (zh) 2007-08-10 2010-09-22 基因实验室技术有限公司 用于治疗病毒感染的含氮的二环化学实体
GB0720126D0 (en) 2007-10-15 2007-11-28 Syngenta Participations Ag Chemical compounds
WO2010005692A2 (en) 2008-06-16 2010-01-14 E. I. Du Pont De Nemours And Company Insecticidal cyclic carbonyl amidines
JP5268461B2 (ja) 2008-07-14 2013-08-21 Meiji Seikaファルマ株式会社 Pf1364物質、その製造方法、生産菌株、及び、それを有効成分とする農園芸用殺虫剤
CA2730844A1 (en) 2008-07-17 2010-01-21 Thomas Bretschneider Heterocyclic compounds used as pesticides
MX2011006319A (es) 2008-12-18 2011-06-24 Bayer Cropscience Ag Amidas del acido antranilico sustituidas con tetrazol como plaguicidas.
UA106363C2 (ru) 2008-12-26 2014-08-26 ДАУ АГРОСАЙЕНСИЗ, ЭлЭлСи Стабильные инсектицидные композиции на основе сульфоксимина
AR075494A1 (es) 2008-12-26 2011-04-06 Dow Agrosciences Llc Composiciones insecticidas estables y metodos para producirlas
JP2011042643A (ja) * 2009-07-24 2011-03-03 Bayer Cropscience Ag 殺虫性カルボキサミド類
WO2011050245A1 (en) 2009-10-23 2011-04-28 Yangbo Feng Bicyclic heteroaryls as kinase inhibitors
KR20120098645A (ko) 2009-10-23 2012-09-05 스미또모 가가꾸 가부시끼가이샤 유해 생물 방제 조성물
UY32940A (es) * 2009-10-27 2011-05-31 Bayer Cropscience Ag Amidas sustituidas con halogenoalquilo como insecticidas y acaricidas
CN101935291B (zh) 2010-09-13 2013-05-01 中化蓝天集团有限公司 一种含氰基的邻苯二甲酰胺类化合物、制备方法和作为农用化学品杀虫剂的用途
CN102057925B (zh) 2011-01-21 2013-04-10 陕西上格之路生物科学有限公司 一种含噻虫酰胺和生物源类杀虫剂的杀虫组合物
AR085509A1 (es) 2011-03-09 2013-10-09 Bayer Cropscience Ag Indol- y bencimidazolcarboxamidas como insecticidas y acaricidas

Also Published As

Publication number Publication date
CN104718206A (zh) 2015-06-17
AU2013304133B2 (en) 2017-02-23
WO2014026984A1 (de) 2014-02-20
CN104718206B (zh) 2017-03-08
KR20150044895A (ko) 2015-04-27
CO7200270A2 (es) 2015-02-27
ZA201501211B (en) 2016-10-26
US20150216175A1 (en) 2015-08-06
BR112015003098A2 (pt) 2017-08-22
CA2881995A1 (en) 2014-02-20
EP2885301A1 (de) 2015-06-24
IN2015DN01061A (enExample) 2015-06-26
RU2015109064A (ru) 2016-10-10
PH12015500334A1 (en) 2015-04-20
JP2015530990A (ja) 2015-10-29
US9345247B2 (en) 2016-05-24
CL2015000336A1 (es) 2015-06-26
MX2015001897A (es) 2015-05-11
AU2013304133A1 (en) 2015-02-26

Similar Documents

Publication Publication Date Title
DOP2014000156A (es) Nuevos derivados de indolizina, su procedimiento de preparación y las composiciones farmacéuticas que los contienen
CR20150370A (es) Compuestos antivirales
CO7200270A2 (es) Azaindolcarboxamidas y azaindoltiocarboxamidas como insecticidas y acaricidas
MX365744B (es) Derivados de sulfuro de trifluoroetilo o sustituidos con n-arilamidina como acaricidas e insecticidas.
EA201492165A1 (ru) Синтез пирроло[2,3-b]пиридинов
CR20140499A (es) Picolinamidas macrocíclicas como fungicidas
UY33978A (es) Piridinonas bicíclicas nuevas.
CO6950507A2 (es) Compuestos de 1,2,5-oxadiazoly su uso como herbicidas ii
PH12015500716A1 (en) N-prop-2-ynyl carboxamide derivatives and their use as trpa1 antagonists
PH12013501859A1 (en) Indolecarboxamides and benzimidazolecarboxamides as insecticides and acaricides
EP2731429A4 (en) COMPOUNDS, METHOD OF MANUFACTURING THEREFOR AND USE METHOD THEREFOR
UY34275A (es) derivados de dihidrofurano, a procesos e intermedios para preparar estos derivados, a composiciones insecticidas, acaricidas, nematicidas y molusquicidas
CR20130041A (es) ISOXAZOLO[5,4-b]PIRIDINAS HERBICIDAS
EP2757092A4 (en) SUBSTITUTED CYANANILIN COMPOUNDS, METHOD OF MANUFACTURING THEREOF AND USE THEREOF
UY34707A (es) Compuestos herbicidas, procesos para su preparación, composiciones herbicidas, su uso para controlar malezas y métodos para controlar malezas
MX2016006012A (es) Formulaciones novedosas.
EP2546226A4 (en) 1-METHOXYL-2,6,10-TRIMETHYL-1,3,5,9-UNDEC-TETRAEN AND METHOD FOR THE PRODUCTION AND USE THEREOF
CO7180217A2 (es) Métodos para preparar 3-sustituido.6-trifluorometil piridinas y métodos para la utilización de 6-triclorometil piridinas halogenadas
UY33167A (es) DERIVADOS DE 5-OXO-5,8-DIHIDRO-PIRIDO[2,3d]PIRIMIDINA, SU PREPARACION y SU APLICACIÓN EN TERAPÉUTICA
UY33975A (es) Formulaciones de otamixaban con estabilidad mejorada
PL402290A1 (pl) Nowe sulfonamidowe pochodne izoksazolo[5,4-b]pirydyny o aktywności przeciwbakteryjnej, sposób ich wytwarzania oraz nowe zastosowanie 3-aminoizoksazolo[5,4-b]pirydyny
CU20150015A7 (es) Tris-(hetero)aril-pirazoles y su uso
EP2835372A4 (en) THIOPHENE [2, 3-D] PYRIMIDINE DERIVATIVE AND METHOD OF PREPARATION AND USE
UY35665A (es) ?compuestos de carboxamida, proceso de preparación y su uso como nematicidas?.
CR20150160A (es) Derivados de macrólidos, su preparación y su uso terapéutico

Legal Events

Date Code Title Description
FD Application declared void or lapsed