PE20110542A1 - Nuevos derivados de azabiclo[3.2.0]hept-3ilo, sus procedimientos de preparacion y las composiciones farmaceuticas que los contienen - Google Patents
Nuevos derivados de azabiclo[3.2.0]hept-3ilo, sus procedimientos de preparacion y las composiciones farmaceuticas que los contienenInfo
- Publication number
- PE20110542A1 PE20110542A1 PE2010001083A PE2010001083A PE20110542A1 PE 20110542 A1 PE20110542 A1 PE 20110542A1 PE 2010001083 A PE2010001083 A PE 2010001083A PE 2010001083 A PE2010001083 A PE 2010001083A PE 20110542 A1 PE20110542 A1 PE 20110542A1
- Authority
- PE
- Peru
- Prior art keywords
- hept
- 3ilo
- azabiclo
- propoxi
- pharmaceutical compositions
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/16—Central respiratory analeptics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Hospice & Palliative Care (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Psychology (AREA)
- Diabetes (AREA)
- Child & Adolescent Psychology (AREA)
- Dermatology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Anesthesiology (AREA)
- Pulmonology (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Indole Compounds (AREA)
Abstract
REFERIDA A UN COMPUESTO AZABICICLO DE FORMULA (I), DONDE ALK REPRESENTA UN GRUPO ALQUILENO C2-C4 Y W ES -NR'-CO-R O -CO-NR'-R; R' Y R SON H ALQUILO C1-C6 OPCIONALMENTE SUSTITUIDO CON HALOGENO, OH U ALCOXI C1-C6. SON COMPUESTOS PREFERIDOS: 4-{3-[(1R,5S)-3-AZABICICLO[3.2.0]HEPT-3-IL]PROPOXI}BENZAMIDA, 4-{3-[(1R,5S)-3-AZABICICLO[3.2.0]HEPT-3-IL]PROPOXI}-N,N-DIMETILBENZAMIDA, N-(4-{3-[(1R,5S)-3-AZABICICLO[3.2.0]HEPT-3-IL]PROPOXI}FENIL)-N-METILACETAMIDA, ENTRE OTROS. TAMBIEN ESTA REFERIDA A UN PROCEDIMIENTO DE PREPARACION Y A UNA COMPOSICION FARMACEUTICA. DICHOS COMPUESTOS TIENEN ACTIVIDAD SOBRE EL SISTEMA HISTAMINERGICO Y SON UTILES EN EL TRATAMIENTO DE TRANSTORNOS COGNITIVOS ASOCIADOS CON EL ENVEJECIMIENTO CEREBRAL O CON ENFERMEDADES NEURODEGENERATIVAS, TRANSTORNOS DEL HUMOR, ENTRE OTROS
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0905957A FR2953514B1 (fr) | 2009-12-09 | 2009-12-09 | Nouveaux derives azabicyclo[3.2.0]hept-3-yl, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PE20110542A1 true PE20110542A1 (es) | 2011-08-18 |
Family
ID=42133738
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PE2010001083A PE20110542A1 (es) | 2009-12-09 | 2010-11-25 | Nuevos derivados de azabiclo[3.2.0]hept-3ilo, sus procedimientos de preparacion y las composiciones farmaceuticas que los contienen |
Country Status (44)
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SI9300625B (sl) * | 1993-12-02 | 2002-02-28 | Basf Aktiengesellschaft | N-substituirani derivati azabicikloheptana, njihova priprava in uporaba |
| DE4341402A1 (de) * | 1993-12-04 | 1995-06-08 | Basf Ag | N-substituierte Azabicycloheptan-Derivate, ihre Herstellung und Verwendung |
| DE4427647A1 (de) * | 1994-08-04 | 1996-02-08 | Basf Ag | N-substituierte Azabicycloheptan-Derivate, ihre Herstellung und Verwendung |
| FR2866647B1 (fr) * | 2004-02-20 | 2006-10-27 | Servier Lab | Nouveaux derives azabicycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
-
2009
- 2009-12-09 FR FR0905957A patent/FR2953514B1/fr not_active Expired - Fee Related
-
2010
- 2010-11-19 MY MYPI2010005458 patent/MY150598A/en unknown
- 2010-11-21 IL IL209463A patent/IL209463A/en not_active IP Right Cessation
- 2010-11-22 UY UY0001033046A patent/UY33046A/es unknown
- 2010-11-22 JO JO2010408A patent/JO2880B1/en active
- 2010-11-23 SG SG2010085959A patent/SG172543A1/en unknown
- 2010-11-24 CR CR11811A patent/CR11811A/es not_active Application Discontinuation
- 2010-11-25 PE PE2010001083A patent/PE20110542A1/es not_active Application Discontinuation
- 2010-11-25 AU AU2010246426A patent/AU2010246426B2/en not_active Ceased
- 2010-11-26 CL CL2010001309A patent/CL2010001309A1/es unknown
- 2010-11-26 TW TW099141093A patent/TWI419875B/zh not_active IP Right Cessation
- 2010-11-29 CN CN2010105733405A patent/CN102127004B/zh not_active Expired - Fee Related
- 2010-11-29 CO CO10150441A patent/CO6280059A1/es active IP Right Grant
- 2010-11-30 MX MX2010013093A patent/MX2010013093A/es active IP Right Grant
- 2010-12-01 MA MA33380A patent/MA32444B1/fr unknown
- 2010-12-01 ZA ZA2010/08651A patent/ZA201008651B/en unknown
- 2010-12-01 AP AP2010005489A patent/AP2755A/xx active
- 2010-12-01 EC EC2010010649A patent/ECSP10010649A/es unknown
- 2010-12-02 CU CU2010000236A patent/CU23993B1/es not_active IP Right Cessation
- 2010-12-02 NI NI201000206A patent/NI201000206A/es unknown
- 2010-12-02 SV SV2010003746A patent/SV2010003746A/es unknown
- 2010-12-03 CA CA2724151A patent/CA2724151C/fr not_active Expired - Fee Related
- 2010-12-06 UA UAA201014568A patent/UA106721C2/uk unknown
- 2010-12-06 AR ARP100104487A patent/AR079268A1/es unknown
- 2010-12-07 KR KR1020100124116A patent/KR101292705B1/ko not_active IP Right Cessation
- 2010-12-07 SA SA110320007A patent/SA110320007B1/ar unknown
- 2010-12-07 GE GEAP201012026A patent/GEP20135801B/en unknown
- 2010-12-07 NZ NZ589763A patent/NZ589763A/en not_active IP Right Cessation
- 2010-12-07 US US12/928,237 patent/US8008337B2/en not_active Expired - Fee Related
- 2010-12-07 EA EA201001755A patent/EA018971B1/ru not_active IP Right Cessation
- 2010-12-08 DK DK10290642.7T patent/DK2332910T3/da active
- 2010-12-08 ME MEP-2013-42A patent/ME01504B/me unknown
- 2010-12-08 WO PCT/FR2010/000820 patent/WO2011070250A1/fr active Application Filing
- 2010-12-08 ES ES10290642T patent/ES2405206T3/es active Active
- 2010-12-08 BR BRPI1005270-4A patent/BRPI1005270A2/pt not_active IP Right Cessation
- 2010-12-08 RS RS20130092A patent/RS52698B/en unknown
- 2010-12-08 PT PT102906427T patent/PT2332910E/pt unknown
- 2010-12-08 PL PL10290642T patent/PL2332910T3/pl unknown
- 2010-12-08 EP EP10290642A patent/EP2332910B1/fr active Active
- 2010-12-08 HN HN2010002593A patent/HN2010002593A/es unknown
- 2010-12-08 SI SI201030183T patent/SI2332910T1/sl unknown
- 2010-12-09 JP JP2010274280A patent/JP5511645B2/ja not_active Expired - Fee Related
-
2013
- 2013-04-04 HR HRP20130307AT patent/HRP20130307T1/hr unknown
- 2013-04-29 CY CY20131100354T patent/CY1113971T1/el unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant, registration | ||
| FD | Application declared void or lapsed |