PE20020589A1 - 5-espiropirimidin-2,4,6-triona como inhibidores de metaloproteinasas - Google Patents
5-espiropirimidin-2,4,6-triona como inhibidores de metaloproteinasasInfo
- Publication number
- PE20020589A1 PE20020589A1 PE2001001060A PE2001001060A PE20020589A1 PE 20020589 A1 PE20020589 A1 PE 20020589A1 PE 2001001060 A PE2001001060 A PE 2001001060A PE 2001001060 A PE2001001060 A PE 2001001060A PE 20020589 A1 PE20020589 A1 PE 20020589A1
- Authority
- PE
- Peru
- Prior art keywords
- heteroaryl
- aryl
- alkyl
- spiropyrimidin
- triona
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/10—Spiro-condensed systems
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- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/10—Spiro-condensed systems
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
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- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
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- Neurosurgery (AREA)
- Immunology (AREA)
- Physical Education & Sports Medicine (AREA)
- Reproductive Health (AREA)
- Endocrinology (AREA)
- Rheumatology (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Dermatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Pain & Pain Management (AREA)
- Pulmonology (AREA)
- Diabetes (AREA)
- Gynecology & Obstetrics (AREA)
- Tropical Medicine & Parasitology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Ophthalmology & Optometry (AREA)
- Cardiology (AREA)
- Pregnancy & Childbirth (AREA)
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Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US24338900P | 2000-10-26 | 2000-10-26 |
Publications (1)
Publication Number | Publication Date |
---|---|
PE20020589A1 true PE20020589A1 (es) | 2002-07-06 |
Family
ID=22918584
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PE2001001060A PE20020589A1 (es) | 2000-10-26 | 2001-10-25 | 5-espiropirimidin-2,4,6-triona como inhibidores de metaloproteinasas |
Country Status (32)
Country | Link |
---|---|
EP (1) | EP1332146A2 (ko) |
JP (1) | JP2004518635A (ko) |
KR (1) | KR20040004412A (ko) |
CN (1) | CN1501937A (ko) |
AP (1) | AP2001002318A0 (ko) |
AR (1) | AR035069A1 (ko) |
AU (1) | AU2002210813A1 (ko) |
BG (1) | BG107653A (ko) |
BR (1) | BR0114913A (ko) |
CA (1) | CA2425283A1 (ko) |
CZ (1) | CZ20031083A3 (ko) |
EA (1) | EA005762B1 (ko) |
EC (1) | ECSP034567A (ko) |
EE (1) | EE200300196A (ko) |
GT (1) | GT200100213A (ko) |
HN (1) | HN2001000244A (ko) |
HR (1) | HRP20030332A2 (ko) |
HU (1) | HUP0301577A3 (ko) |
IL (1) | IL154948A0 (ko) |
IS (1) | IS6762A (ko) |
MA (1) | MA26957A1 (ko) |
MX (1) | MXPA03003735A (ko) |
NO (1) | NO20031853L (ko) |
OA (1) | OA12529A (ko) |
PA (1) | PA8531401A1 (ko) |
PE (1) | PE20020589A1 (ko) |
PL (1) | PL366201A1 (ko) |
SK (1) | SK4972003A3 (ko) |
SV (1) | SV2003000705A (ko) |
TN (1) | TNSN01149A1 (ko) |
WO (1) | WO2002034753A2 (ko) |
ZA (1) | ZA200302190B (ko) |
Families Citing this family (36)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DOP2002000333A (es) | 2001-02-14 | 2002-09-30 | Warner Lambert Co | Derivados de acido isoftalico como inhibidores de metaloproteinasas de la matriz |
BR0207865A (pt) | 2001-02-14 | 2004-03-23 | Warner Lambert Co | Benzotiadiazinas inibidores de metaloproteinases de matriz |
DOP2002000332A (es) | 2001-02-14 | 2002-08-30 | Warner Lambert Co | Inhibidores de piridina de metaloproteinasas de la matriz |
PA8539501A1 (es) | 2001-02-14 | 2002-09-30 | Warner Lambert Co | Compuestos triazolo como inhibidores de mmp |
DOP2002000328A (es) | 2001-02-14 | 2003-08-30 | Warner Lambert Co | Pirimidinas inhibidoras de metaloproteinasas de matriz |
US6924276B2 (en) | 2001-09-10 | 2005-08-02 | Warner-Lambert Company | Diacid-substituted heteroaryl derivatives as matrix metalloproteinase inhibitors |
US6962922B2 (en) | 2001-10-12 | 2005-11-08 | Warner-Lambert Company Llc | Alkynylated quinazoline compounds |
BR0213233A (pt) | 2001-10-12 | 2005-01-04 | Warner Lambert Co | Alcinos inibidores de metaloproteinase de matriz |
US6894057B2 (en) | 2002-03-08 | 2005-05-17 | Warner-Lambert Company | Oxo-azabicyclic compounds |
WO2003091252A1 (en) * | 2002-04-25 | 2003-11-06 | Bristol-Myers Squibb Company | Spirobarbituric acid derivatives useful as inhibitors of matrix metalloproteases |
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JP2002504916A (ja) * | 1997-06-21 | 2002-02-12 | ロシュ ダイアグノスティクス ゲゼルシャフト ミット ベシュレンクテル ハフツング | 抗転移及び抗腫瘍活性を有するバルビツール酸誘導体 |
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