OA13338A - 3-cycloalkylaminopyrrolidine derivates as modulators of chemokine receptors. - Google Patents

3-cycloalkylaminopyrrolidine derivates as modulators of chemokine receptors. Download PDF

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Publication number
OA13338A
OA13338A OA1200600195A OA1200600195A OA13338A OA 13338 A OA13338 A OA 13338A OA 1200600195 A OA1200600195 A OA 1200600195A OA 1200600195 A OA1200600195 A OA 1200600195A OA 13338 A OA13338 A OA 13338A
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OA
OAPI
Prior art keywords
amino
trifluoromethyl
mono
pyrrolidin
pyridin
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OA1200600195A
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English (en)
Inventor
Amy Qi Han
Brian Metcalf
Darius J Robinson
Anlai Wang
Chu-Biao Xue
Yingxin Zhang
Chansheng Zheng
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Incyte Corp
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Publication of OA13338A publication Critical patent/OA13338A/en

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    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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OA1200600195A 2003-12-18 2004-12-16 3-cycloalkylaminopyrrolidine derivates as modulators of chemokine receptors. OA13338A (en)

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US53127003P 2003-12-18 2003-12-18

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JP (1) JP4740151B2 (fr)
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Families Citing this family (46)

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Publication number Priority date Publication date Assignee Title
ATE555087T1 (de) * 2002-11-27 2012-05-15 Incyte Corp 3-aminopyrrolidinderivate als modulatoren von chemokinrezeptoren
BRPI0509803A (pt) * 2004-04-13 2007-09-18 Incyte Corp derivados de piperazinilpiperidina como antagonistas de receptor de quimiocina
AU2005247361B2 (en) 2004-05-11 2011-03-17 Incyte Corporation 3-(4-heteroarylcyclohexylamino) cyclopentanecarboxamides as modulators of chemokine receptors
BRPI0512634A (pt) 2004-06-28 2008-03-25 Incyte Corp 3-aminociclopentanocarboxamidas como moduladores de receptores de quimiocinas
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