OA13039A - 3-(1-[3-(1,3-benzothiazol-6-yl)propylcarbamoyl]cycloalkyl)propanoic acid derivatives as NEP inhibitors. - Google Patents

3-(1-[3-(1,3-benzothiazol-6-yl)propylcarbamoyl]cycloalkyl)propanoic acid derivatives as NEP inhibitors. Download PDF

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Publication number
OA13039A
OA13039A OA1200500261A OA1200500261A OA13039A OA 13039 A OA13039 A OA 13039A OA 1200500261 A OA1200500261 A OA 1200500261A OA 1200500261 A OA1200500261 A OA 1200500261A OA 13039 A OA13039 A OA 13039A
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OA
OAPI
Prior art keywords
disorder
methyl
compound
compounds
sexual
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Application number
OA1200500261A
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English (en)
Inventor
David Hepworth
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0305916A external-priority patent/GB0305916D0/en
Priority claimed from GB0329143A external-priority patent/GB0329143D0/en
Application filed by Pfizer filed Critical Pfizer
Publication of OA13039A publication Critical patent/OA13039A/en

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P9/12—Antihypertensives

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  • Pain & Pain Management (AREA)
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  • Heart & Thoracic Surgery (AREA)
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OA1200500261A 2003-03-14 2004-03-09 3-(1-[3-(1,3-benzothiazol-6-yl)propylcarbamoyl]cycloalkyl)propanoic acid derivatives as NEP inhibitors. OA13039A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB0305916A GB0305916D0 (en) 2003-03-14 2003-03-14 New N-phenpropylcyclopentyl-substituted glutaramide derivatives as NEP inhibitors
GB0329143A GB0329143D0 (en) 2003-12-16 2003-12-16 Novel pharmaceuticals

Publications (1)

Publication Number Publication Date
OA13039A true OA13039A (en) 2006-11-10

Family

ID=32992599

Family Applications (1)

Application Number Title Priority Date Filing Date
OA1200500261A OA13039A (en) 2003-03-14 2004-03-09 3-(1-[3-(1,3-benzothiazol-6-yl)propylcarbamoyl]cycloalkyl)propanoic acid derivatives as NEP inhibitors.

Country Status (25)

Country Link
US (1) US20040180941A1 (pt)
EP (1) EP1606272A1 (pt)
JP (1) JP3923512B2 (pt)
KR (1) KR20050110003A (pt)
AP (1) AP2005003393A0 (pt)
AR (1) AR043551A1 (pt)
AU (1) AU2004220269A1 (pt)
BR (1) BRPI0408377A (pt)
CA (1) CA2519072A1 (pt)
CL (1) CL2004000512A1 (pt)
EA (1) EA200501204A1 (pt)
EC (1) ECSP056017A (pt)
HR (1) HRP20050797A2 (pt)
IS (1) IS8003A (pt)
MA (1) MA27720A1 (pt)
MX (1) MXPA05009788A (pt)
NL (1) NL1025709C2 (pt)
NO (1) NO20054169L (pt)
OA (1) OA13039A (pt)
PA (1) PA8597401A1 (pt)
PE (1) PE20050310A1 (pt)
TN (1) TNSN05227A1 (pt)
TW (1) TW200504038A (pt)
UY (1) UY28226A1 (pt)
WO (1) WO2004080985A1 (pt)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2575706A1 (en) * 2004-08-02 2006-02-23 Bebaas, Inc. Vitamin b12 compositions
WO2006027680A1 (en) * 2004-09-10 2006-03-16 Pfizer Limited 3-(1-carbamoylcyclohexyl) propionic acid derivatives as inhibitors of neutral endopeptidase enzyme
ES2425567T3 (es) 2004-12-24 2013-10-16 Spinifex Pharmaceuticals Pty Ltd Método de tratamiento o profilaxis
KR20080047375A (ko) 2005-07-29 2008-05-28 콘서트 파마슈티컬즈, 인크. 약제 화합물
US20130131007A1 (en) 2005-09-07 2013-05-23 Bebaas, Inc. Vitamin b12 compositions
US20070178141A1 (en) * 2005-09-07 2007-08-02 Bebaas, Inc. Vitamin B12 compositions
CN102885818B (zh) 2006-03-20 2016-05-04 诺华股份有限公司 治疗或预防炎性痛的方法
WO2008021666A2 (en) * 2006-08-18 2008-02-21 Morton Grove Pharmaceuticals, Inc. Stable liquid levetiracetam compositions and methods
KR101177866B1 (ko) 2011-03-24 2012-08-28 주식회사 케이엠더블유 케이블 접속 장치
JP2021527267A (ja) * 2018-06-14 2021-10-11 アストラゼネカ・ユーケイ・リミテッドＡｓｔｒａＺｅｎｅｃａ ＵＫ Ｌｉｍｉｔｅｄ Ｃｇｍｐ特異的ホスホジエステラーゼ５阻害剤の薬学的組成物により勃起不全を治療するための方法
CN112955967A (zh) * 2018-06-14 2021-06-11 阿斯利康(英国)有限公司 用cgmp特异性磷酸二酯酶5抑制剂医药组合物治疗勃起功能障碍的方法
IL292775A (en) * 2019-11-08 2022-07-01 Vella Bioscience Inc preparations containing cannabidiol (cbd) that act peripherally and their use to improve female sexual function or to treat female sexual disorders

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US2503059A (en) * 1950-04-04 Nxchj
US2599000A (en) * 1950-09-02 1952-06-03 Smith Kline French Lab Nu, nu-disubstituted-beta-halo-alkylamines
US3238215A (en) * 1963-10-17 1966-03-01 Sterling Drug Inc 1-[(3-, 2-, and 1-indolyl)-lower-alkyl-, lower-alkenyl-, and lower-alkynyl]piperidines
IT1066857B (it) * 1965-12-15 1985-03-12 Acraf Derivati della s ipiazolo 4.3 a piridina e processi per la loro preparazione
US3511836A (en) * 1967-12-13 1970-05-12 Pfizer & Co C 2,4,6,7-tetra substituted quinazolines
NL175059C (nl) * 1974-02-23 Boehringer Mannheim Gmbh Bereiding van bloeddrukverlagende stoffen en van preparaten die ze bevatten.
US4026894A (en) * 1975-10-14 1977-05-31 Abbott Laboratories Antihypertensive agents
US4188390A (en) * 1977-11-05 1980-02-12 Pfizer Inc. Antihypertensive 4-amino-2-[4-(1,4-benzodioxan-2-carbonyl) piperazin-1-yl or homopiperazin-1-yl]quinazolines
FR2421888A1 (fr) * 1978-02-06 1979-11-02 Synthelabo Amides d'alkylene-diamines et leur application en therapeutique
IT1094076B (it) * 1978-04-18 1985-07-26 Acraf Cicloalchiltriazoli
JPS56110665A (en) * 1980-02-08 1981-09-01 Yamanouchi Pharmaceut Co Ltd Sulfamoyl-substituted phenetylamine derivative and its preparation
DE3528032A1 (de) * 1985-08-05 1987-02-05 Hoechst Ag Verfahren zur herstellung 2-substituierter benzthiazole
PT100905A (pt) * 1991-09-30 1994-02-28 Eisai Co Ltd Compostos heterociclicos azotados biciclicos contendo aneis de benzeno, ciclo-hexano ou piridina e de pirimidina, piridina ou imidazol substituidos e composicoes farmaceuticas que os contem
US5698560A (en) * 1995-03-01 1997-12-16 Kyowa Hakko Kogyo Co., Ltd. Imidazoquinazoline derivatives
GB9518953D0 (en) * 1995-09-15 1995-11-15 Pfizer Ltd Pharmaceutical formulations
US6037346A (en) * 1997-10-28 2000-03-14 Vivus, Inc. Local administration of phosphodiesterase inhibitors for the treatment of erectile dysfunction
OA12553A (en) * 2001-03-28 2006-06-07 Pfizer N-Phenpropylcyclopentyl-substituted glutaramide derivatives as NEP inhibitors for FSAD.

Also Published As

Publication number Publication date
BRPI0408377A (pt) 2006-03-21
JP3923512B2 (ja) 2007-06-06
IS8003A (is) 2005-08-29
EP1606272A1 (en) 2005-12-21
NO20054169L (no) 2005-12-07
ECSP056017A (es) 2006-01-27
MA27720A1 (fr) 2006-01-02
AP2005003393A0 (en) 2005-09-30
KR20050110003A (ko) 2005-11-22
PE20050310A1 (es) 2005-05-04
EA200501204A1 (ru) 2006-06-30
AU2004220269A1 (en) 2004-09-23
PA8597401A1 (es) 2005-05-24
CA2519072A1 (en) 2004-09-23
TNSN05227A1 (fr) 2007-06-11
JP2006526572A (ja) 2006-11-24
AR043551A1 (es) 2005-08-03
NL1025709A1 (nl) 2004-09-16
US20040180941A1 (en) 2004-09-16
UY28226A1 (es) 2004-11-08
CL2004000512A1 (es) 2005-01-21
TW200504038A (en) 2005-02-01
WO2004080985A1 (en) 2004-09-23
MXPA05009788A (es) 2005-10-26
HRP20050797A2 (en) 2006-02-28
NL1025709C2 (nl) 2005-03-14
NO20054169D0 (no) 2005-09-07

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