NO20054169L - 3-(1-[3-(1,3-benzotiazol-6-yl) propylkarbamoyl]sykloalkyl]propansyrederivater som NEP-inhibitorer. - Google Patents

3-(1-[3-(1,3-benzotiazol-6-yl) propylkarbamoyl]sykloalkyl]propansyrederivater som NEP-inhibitorer.

Info

Publication number
NO20054169L
NO20054169L NO20054169A NO20054169A NO20054169L NO 20054169 L NO20054169 L NO 20054169L NO 20054169 A NO20054169 A NO 20054169A NO 20054169 A NO20054169 A NO 20054169A NO 20054169 L NO20054169 L NO 20054169L
Authority
NO
Norway
Prior art keywords
propylcarbamoyl
benzothiazol
cycloalkyl
inhibitors
acid derivatives
Prior art date
Application number
NO20054169A
Other languages
English (en)
Other versions
NO20054169D0 (no
Inventor
David Hepworth
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0305916A external-priority patent/GB0305916D0/en
Priority claimed from GB0329143A external-priority patent/GB0329143D0/en
Application filed by Pfizer filed Critical Pfizer
Publication of NO20054169D0 publication Critical patent/NO20054169D0/no
Publication of NO20054169L publication Critical patent/NO20054169L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

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Abstract

Oppfinnelsen angår inhibitorer av nøytralt endopeptidase-enzym (NEP) med formel (I), anvendelser derav, fremgangsmåter for fremstilling derav, mellomprodukter anvendt ved fremstilling derav og preparater inneholdende nevnte inhibitorer. Disse inhibitorer er anvendelige på en rekke terapeutiske områder omfattende behandling av mannlig og kvinnelig seksuell dysfunksjon, spesielt kvinnelig seksuell dysfunksjon (FSD), spesielt hvor FSD er kvinnelig seksuell opphisselse-lidelse (FSAD).
NO20054169A 2003-03-14 2005-09-07 3-(1-[3-(1,3-benzotiazol-6-yl) propylkarbamoyl]sykloalkyl]propansyrederivater som NEP-inhibitorer. NO20054169L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0305916A GB0305916D0 (en) 2003-03-14 2003-03-14 New N-phenpropylcyclopentyl-substituted glutaramide derivatives as NEP inhibitors
GB0329143A GB0329143D0 (en) 2003-12-16 2003-12-16 Novel pharmaceuticals
PCT/IB2004/000822 WO2004080985A1 (en) 2003-03-14 2004-03-09 3-(1-[3-(1,3-benzothiazol-6-yl)propylcarbamoyl]cycloalkyl)propanoic acid derivatives as nep inhibitors

Publications (2)

Publication Number Publication Date
NO20054169D0 NO20054169D0 (no) 2005-09-07
NO20054169L true NO20054169L (no) 2005-12-07

Family

ID=32992599

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20054169A NO20054169L (no) 2003-03-14 2005-09-07 3-(1-[3-(1,3-benzotiazol-6-yl) propylkarbamoyl]sykloalkyl]propansyrederivater som NEP-inhibitorer.

Country Status (25)

Country Link
US (1) US20040180941A1 (no)
EP (1) EP1606272A1 (no)
JP (1) JP3923512B2 (no)
KR (1) KR20050110003A (no)
AP (1) AP2005003393A0 (no)
AR (1) AR043551A1 (no)
AU (1) AU2004220269A1 (no)
BR (1) BRPI0408377A (no)
CA (1) CA2519072A1 (no)
CL (1) CL2004000512A1 (no)
EA (1) EA200501204A1 (no)
EC (1) ECSP056017A (no)
HR (1) HRP20050797A2 (no)
IS (1) IS8003A (no)
MA (1) MA27720A1 (no)
MX (1) MXPA05009788A (no)
NL (1) NL1025709C2 (no)
NO (1) NO20054169L (no)
OA (1) OA13039A (no)
PA (1) PA8597401A1 (no)
PE (1) PE20050310A1 (no)
TN (1) TNSN05227A1 (no)
TW (1) TW200504038A (no)
UY (1) UY28226A1 (no)
WO (1) WO2004080985A1 (no)

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CA2575706A1 (en) * 2004-08-02 2006-02-23 Bebaas, Inc. Vitamin b12 compositions
WO2006027680A1 (en) * 2004-09-10 2006-03-16 Pfizer Limited 3-(1-carbamoylcyclohexyl) propionic acid derivatives as inhibitors of neutral endopeptidase enzyme
ES2425567T3 (es) 2004-12-24 2013-10-16 Spinifex Pharmaceuticals Pty Ltd Método de tratamiento o profilaxis
KR20080047375A (ko) 2005-07-29 2008-05-28 콘서트 파마슈티컬즈, 인크. 약제 화합물
US20130131007A1 (en) 2005-09-07 2013-05-23 Bebaas, Inc. Vitamin b12 compositions
US20070178141A1 (en) * 2005-09-07 2007-08-02 Bebaas, Inc. Vitamin B12 compositions
CN102885818B (zh) 2006-03-20 2016-05-04 诺华股份有限公司 治疗或预防炎性痛的方法
WO2008021666A2 (en) * 2006-08-18 2008-02-21 Morton Grove Pharmaceuticals, Inc. Stable liquid levetiracetam compositions and methods
KR101177866B1 (ko) 2011-03-24 2012-08-28 주식회사 케이엠더블유 케이블 접속 장치
JP2021527267A (ja) * 2018-06-14 2021-10-11 アストラゼネカ・ユーケイ・リミテッドＡｓｔｒａＺｅｎｅｃａ ＵＫ Ｌｉｍｉｔｅｄ Ｃｇｍｐ特異的ホスホジエステラーゼ５阻害剤の薬学的組成物により勃起不全を治療するための方法
CN112955967A (zh) * 2018-06-14 2021-06-11 阿斯利康(英国)有限公司 用cgmp特异性磷酸二酯酶5抑制剂医药组合物治疗勃起功能障碍的方法
IL292775A (en) * 2019-11-08 2022-07-01 Vella Bioscience Inc preparations containing cannabidiol (cbd) that act peripherally and their use to improve female sexual function or to treat female sexual disorders

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Also Published As

Publication number Publication date
BRPI0408377A (pt) 2006-03-21
JP3923512B2 (ja) 2007-06-06
IS8003A (is) 2005-08-29
EP1606272A1 (en) 2005-12-21
ECSP056017A (es) 2006-01-27
MA27720A1 (fr) 2006-01-02
AP2005003393A0 (en) 2005-09-30
KR20050110003A (ko) 2005-11-22
PE20050310A1 (es) 2005-05-04
EA200501204A1 (ru) 2006-06-30
AU2004220269A1 (en) 2004-09-23
OA13039A (en) 2006-11-10
PA8597401A1 (es) 2005-05-24
CA2519072A1 (en) 2004-09-23
TNSN05227A1 (fr) 2007-06-11
JP2006526572A (ja) 2006-11-24
AR043551A1 (es) 2005-08-03
NL1025709A1 (nl) 2004-09-16
US20040180941A1 (en) 2004-09-16
UY28226A1 (es) 2004-11-08
CL2004000512A1 (es) 2005-01-21
TW200504038A (en) 2005-02-01
WO2004080985A1 (en) 2004-09-23
MXPA05009788A (es) 2005-10-26
HRP20050797A2 (en) 2006-02-28
NL1025709C2 (nl) 2005-03-14
NO20054169D0 (no) 2005-09-07

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