OA12081A - Hygromycin derivatives. - Google Patents

Hygromycin derivatives. Download PDF

Info

Publication number
OA12081A
OA12081A OA1200200129A OA1200200129A OA12081A OA 12081 A OA12081 A OA 12081A OA 1200200129 A OA1200200129 A OA 1200200129A OA 1200200129 A OA1200200129 A OA 1200200129A OA 12081 A OA12081 A OA 12081A
Authority
OA
OAPI
Prior art keywords
alkyl
groups
aryl
independently
methyl
Prior art date
Application number
OA1200200129A
Other languages
English (en)
Inventor
Matthew Merrill Hayward
Takushi Kaneko
Linde Robert Gerald Ii
Katherine Elizabeth Brighty
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of OA12081A publication Critical patent/OA12081A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/26—Acyclic or carbocyclic radicals, substituted by hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Genetics & Genomics (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
OA1200200129A 1999-10-29 2000-10-09 Hygromycin derivatives. OA12081A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US16258199P 1999-10-29 1999-10-29

Publications (1)

Publication Number Publication Date
OA12081A true OA12081A (en) 2006-05-04

Family

ID=22586256

Family Applications (1)

Application Number Title Priority Date Filing Date
OA1200200129A OA12081A (en) 1999-10-29 2000-10-09 Hygromycin derivatives.

Country Status (32)

Country Link
US (1) US6562792B1 (bg)
EP (1) EP1224197A1 (bg)
JP (1) JP2003512473A (bg)
KR (1) KR20020063885A (bg)
CN (1) CN1382150A (bg)
AP (1) AP2002002494A0 (bg)
AR (1) AR023282A1 (bg)
AU (1) AU7549400A (bg)
BG (1) BG106727A (bg)
BR (1) BR0015153A (bg)
CA (1) CA2389191A1 (bg)
CO (1) CO5261498A1 (bg)
CZ (1) CZ20021355A3 (bg)
EA (1) EA200200292A1 (bg)
EE (1) EE200200228A (bg)
GT (1) GT200000185A (bg)
HK (1) HK1049672A1 (bg)
HU (1) HUP0203525A3 (bg)
IL (1) IL148577A0 (bg)
IS (1) IS6311A (bg)
MA (1) MA26838A1 (bg)
MX (1) MXPA02004360A (bg)
NO (1) NO20021850L (bg)
OA (1) OA12081A (bg)
PA (1) PA8505801A1 (bg)
PE (1) PE20010763A1 (bg)
PL (1) PL357083A1 (bg)
SK (1) SK5472002A3 (bg)
SV (1) SV2002000211A (bg)
TN (1) TNSN00211A1 (bg)
TR (1) TR200201145T2 (bg)
WO (1) WO2001030795A1 (bg)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EE200200671A (et) 2000-06-02 2004-08-16 Pfizer Products Inc. Hügromütsiin A derivaadid bakteriaalsete ja algloomadest põhjustatud infektsioonide ravimiseks
US6653481B2 (en) * 2000-12-29 2003-11-25 Synthon Bv Process for making amlodipine
US7923439B2 (en) * 2008-10-15 2011-04-12 Tyco Healthcare Group Lp Hydroxamate compositions
US20210275559A1 (en) * 2018-08-20 2021-09-09 Kim Lewis Hygromycin a compounds and methods of treating spirochete diseases
TW202128675A (zh) 2019-12-06 2021-08-01 美商維泰克斯製藥公司 作為鈉通道調節劑之經取代四氫呋喃
PE20241335A1 (es) 2021-06-04 2024-07-03 Vertex Pharma N-(hidroxialquil (hetero)aril) tetrahidrofurano carboxamidas como moduladores de canales de sodio

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100418167B1 (ko) * 1998-12-02 2004-02-11 화이자 프로덕츠 인크. 항균제로서의 하이그로마이신 ａ 유도체

Also Published As

Publication number Publication date
WO2001030795A1 (en) 2001-05-03
PA8505801A1 (es) 2002-08-26
KR20020063885A (ko) 2002-08-05
HUP0203525A3 (en) 2003-08-28
AR023282A1 (es) 2002-09-04
IL148577A0 (en) 2002-09-12
CO5261498A1 (es) 2003-03-31
US6562792B1 (en) 2003-05-13
SK5472002A3 (en) 2003-02-04
GT200000185A (es) 2002-04-18
TR200201145T2 (tr) 2002-09-23
CN1382150A (zh) 2002-11-27
NO20021850D0 (no) 2002-04-19
CA2389191A1 (en) 2001-05-03
SV2002000211A (es) 2002-07-16
AP2002002494A0 (en) 2002-06-30
IS6311A (is) 2002-03-19
PL357083A1 (en) 2004-07-12
EA200200292A1 (ru) 2002-10-31
JP2003512473A (ja) 2003-04-02
MA26838A1 (fr) 2004-12-20
EP1224197A1 (en) 2002-07-24
AU7549400A (en) 2001-05-08
BG106727A (bg) 2003-01-31
PE20010763A1 (es) 2001-07-25
TNSN00211A1 (fr) 2005-11-10
EE200200228A (et) 2003-06-16
MXPA02004360A (es) 2002-11-07
HUP0203525A2 (hu) 2003-02-28
CZ20021355A3 (cs) 2002-11-13
NO20021850L (no) 2002-04-19
BR0015153A (pt) 2002-07-16
HK1049672A1 (zh) 2003-05-23

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