NZ597638A - 5-fluoro-2-oxopyrimidine- 1(2h)-carboxylate derivatives - Google Patents

5-fluoro-2-oxopyrimidine- 1(2h)-carboxylate derivatives

Info

Publication number
NZ597638A
NZ597638A NZ597638A NZ59763810A NZ597638A NZ 597638 A NZ597638 A NZ 597638A NZ 597638 A NZ597638 A NZ 597638A NZ 59763810 A NZ59763810 A NZ 59763810A NZ 597638 A NZ597638 A NZ 597638A
Authority
NZ
New Zealand
Prior art keywords
fluoro
oxopyrimidine
amino
carboxylate
optionally substituted
Prior art date
Application number
NZ597638A
Other languages
English (en)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535293&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NZ597638(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of NZ597638A publication Critical patent/NZ597638A/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/16Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof the nitrogen atom being part of a heterocyclic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/20Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D239/22Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
NZ597638A 2009-08-07 2010-08-05 5-fluoro-2-oxopyrimidine- 1(2h)-carboxylate derivatives NZ597638A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23223209P 2009-08-07 2009-08-07
PCT/US2010/044585 WO2011017544A1 (en) 2009-08-07 2010-08-05 5-fluoro-2-oxopyrimidine- 1(2h)-carboxylate derivatives

Publications (1)

Publication Number Publication Date
NZ597638A true NZ597638A (en) 2014-06-27

Family

ID=43535293

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ597638A NZ597638A (en) 2009-08-07 2010-08-05 5-fluoro-2-oxopyrimidine- 1(2h)-carboxylate derivatives

Country Status (28)

Country Link
US (1) US8318758B2 (OSRAM)
EP (1) EP2462133B1 (OSRAM)
JP (1) JP5818791B2 (OSRAM)
KR (1) KR101792286B1 (OSRAM)
CN (1) CN102548979B (OSRAM)
AU (1) AU2010279408B2 (OSRAM)
BR (1) BR112012002807B1 (OSRAM)
CA (1) CA2769251C (OSRAM)
CL (1) CL2012000314A1 (OSRAM)
CO (1) CO6491089A2 (OSRAM)
CR (1) CR20120033A (OSRAM)
DK (1) DK2462133T3 (OSRAM)
EA (1) EA022930B1 (OSRAM)
EC (1) ECSP12011651A (OSRAM)
ES (1) ES2506169T3 (OSRAM)
HN (1) HN2012000261A (OSRAM)
IL (1) IL217954A (OSRAM)
IN (1) IN2012DN00695A (OSRAM)
MX (1) MX2012001623A (OSRAM)
NI (1) NI201200019A (OSRAM)
NZ (1) NZ597638A (OSRAM)
PE (1) PE20120689A1 (OSRAM)
PL (1) PL2462133T3 (OSRAM)
PT (1) PT2462133E (OSRAM)
RS (1) RS53658B1 (OSRAM)
UA (1) UA106086C2 (OSRAM)
WO (1) WO2011017544A1 (OSRAM)
ZA (1) ZA201305992B (OSRAM)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA106764C2 (uk) * 2009-08-07 2014-10-10 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні n1-сульфоніл-5-фторпіримідинону
US9622474B2 (en) * 2012-12-28 2017-04-18 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxylate derivatives
HK1214518A1 (zh) * 2012-12-28 2016-07-29 Adama Makhteshim Ltd. 1-(经取代之苯甲醯基)-5-氟-4-亚胺基-3-甲基-3,4-二氢嘧啶-2(1h)-酮衍生物
US9321734B2 (en) 2012-12-28 2016-04-26 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxamide derivatives
AU2013370494B2 (en) 2012-12-31 2017-08-17 Adama Makhteshim Ltd. 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1H)-one derivatives as fungicides
CN106068268A (zh) 2013-12-31 2016-11-02 阿达玛马克西姆股份有限公司 5‑氟‑4‑亚氨基‑3‑(烷基/取代烷基)‑1‑(芳基磺酰基)‑3,4‑二氢嘧啶‑2(1h)‑酮及其制备方法
EA030056B1 (ru) 2013-12-31 2018-06-29 Адама Мактешим Лтд. Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами
WO2016040193A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof
WO2017079759A1 (en) 2015-11-06 2017-05-11 Samumed, Llc 2-(1h-indazol-3-yl)-3h-imidazo[4,5-c]pyridines and their anti-inflammatory uses thereof
SG10201912248RA (en) 2016-06-01 2020-02-27 Samumed Llc Process for preparing n-(5-(3-(7-(3-fluorophenyl)-3h-imidazo[4,5-c]pyridin-2-yl)-1h-indazol-5-yl)pyridin-3-yl)-3-methylbutanamide
MA49639A (fr) 2017-07-17 2020-05-27 Adama Makhteshim Ltd Polymorphes de 5-fluoro-4-imino-3-méthyl-1-tosyl-3,4-dihydropyrimidin-2-one
CR20210270A (es) 2018-11-05 2021-07-20 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de los mismos
US12466796B2 (en) 2019-09-23 2025-11-11 Adama Makhteshim Ltd. Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1H)-one and derivatives of the compound

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
AU716248B2 (en) * 1996-03-11 2000-02-24 Novartis Ag Pyrimidin-4-one derivatives as pesticide
AU2003274652A1 (en) * 2002-10-23 2004-05-13 Obetherapy Biotechnology Compounds, compositions and methods for modulating fat metabolism
CN101730691A (zh) * 2007-04-27 2010-06-09 阿斯比奥制药株式会社 含氮芳香族六元环衍生物及含有它们的药物
UA107651C2 (en) 2008-08-01 2015-02-10 Dow Agrosciences Llc Use of 5-fluorocytosine as a fungicide

Also Published As

Publication number Publication date
IL217954A0 (en) 2012-03-29
CN102548979B (zh) 2015-05-13
RS53658B1 (sr) 2015-04-30
CL2012000314A1 (es) 2012-10-05
US20110034491A1 (en) 2011-02-10
KR101792286B1 (ko) 2017-10-31
BR112012002807B1 (pt) 2018-07-10
PT2462133E (pt) 2014-12-26
CR20120033A (es) 2012-03-22
EA022930B1 (ru) 2016-03-31
EA201270255A1 (ru) 2012-07-30
KR20120043069A (ko) 2012-05-03
JP2013501726A (ja) 2013-01-17
AU2010279408B2 (en) 2015-09-10
BR112012002807A8 (pt) 2017-07-11
ZA201305992B (en) 2014-10-29
CA2769251A1 (en) 2011-02-10
WO2011017544A1 (en) 2011-02-10
EP2462133A4 (en) 2013-01-16
US8318758B2 (en) 2012-11-27
CN102548979A (zh) 2012-07-04
UA106086C2 (uk) 2014-07-25
AU2010279408A1 (en) 2012-02-09
DK2462133T3 (en) 2015-01-05
JP5818791B2 (ja) 2015-11-18
MX2012001623A (es) 2012-04-11
ECSP12011651A (es) 2012-03-30
HK1172892A1 (en) 2013-05-03
EP2462133B1 (en) 2014-09-24
PE20120689A1 (es) 2012-06-06
IN2012DN00695A (OSRAM) 2015-06-19
IL217954A (en) 2016-02-29
HN2012000261A (es) 2015-01-05
EP2462133A1 (en) 2012-06-13
NI201200019A (es) 2012-05-22
CO6491089A2 (es) 2012-07-31
ES2506169T3 (es) 2014-10-13
BR112012002807A2 (pt) 2015-10-13
PL2462133T3 (pl) 2015-03-31
CA2769251C (en) 2018-05-15

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