CO6491089A2 - Derivados de 5-fluoruro-2-oxopirimidina-1(2h)-carboxilato - Google Patents

Derivados de 5-fluoruro-2-oxopirimidina-1(2h)-carboxilato

Info

Publication number
CO6491089A2
CO6491089A2 CO12012413A CO12012413A CO6491089A2 CO 6491089 A2 CO6491089 A2 CO 6491089A2 CO 12012413 A CO12012413 A CO 12012413A CO 12012413 A CO12012413 A CO 12012413A CO 6491089 A2 CO6491089 A2 CO 6491089A2
Authority
CO
Colombia
Prior art keywords
plant
formula
derivatives
oxopirimidina
carboxylate
Prior art date
Application number
CO12012413A
Other languages
English (en)
Spanish (es)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W Jhon Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Original Assignee
Dow Agroscience Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535293&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO6491089(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agroscience Llc filed Critical Dow Agroscience Llc
Publication of CO6491089A2 publication Critical patent/CO6491089A2/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/541,3-Diazines; Hydrogenated 1,3-diazines
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/16Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof the nitrogen atom being part of a heterocyclic ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/20Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D239/22Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to ring carbon atoms

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
CO12012413A 2009-08-07 2012-01-27 Derivados de 5-fluoruro-2-oxopirimidina-1(2h)-carboxilato CO6491089A2 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23223209P 2009-08-07 2009-08-07

Publications (1)

Publication Number Publication Date
CO6491089A2 true CO6491089A2 (es) 2012-07-31

Family

ID=43535293

Family Applications (1)

Application Number Title Priority Date Filing Date
CO12012413A CO6491089A2 (es) 2009-08-07 2012-01-27 Derivados de 5-fluoruro-2-oxopirimidina-1(2h)-carboxilato

Country Status (28)

Country Link
US (1) US8318758B2 (OSRAM)
EP (1) EP2462133B1 (OSRAM)
JP (1) JP5818791B2 (OSRAM)
KR (1) KR101792286B1 (OSRAM)
CN (1) CN102548979B (OSRAM)
AU (1) AU2010279408B2 (OSRAM)
BR (1) BR112012002807B1 (OSRAM)
CA (1) CA2769251C (OSRAM)
CL (1) CL2012000314A1 (OSRAM)
CO (1) CO6491089A2 (OSRAM)
CR (1) CR20120033A (OSRAM)
DK (1) DK2462133T3 (OSRAM)
EA (1) EA022930B1 (OSRAM)
EC (1) ECSP12011651A (OSRAM)
ES (1) ES2506169T3 (OSRAM)
HN (1) HN2012000261A (OSRAM)
IL (1) IL217954A (OSRAM)
IN (1) IN2012DN00695A (OSRAM)
MX (1) MX2012001623A (OSRAM)
NI (1) NI201200019A (OSRAM)
NZ (1) NZ597638A (OSRAM)
PE (1) PE20120689A1 (OSRAM)
PL (1) PL2462133T3 (OSRAM)
PT (1) PT2462133E (OSRAM)
RS (1) RS53658B1 (OSRAM)
UA (1) UA106086C2 (OSRAM)
WO (1) WO2011017544A1 (OSRAM)
ZA (1) ZA201305992B (OSRAM)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2462134B1 (en) * 2009-08-07 2014-05-07 Dow AgroSciences LLC N1-sulfonyl-5-fluoropyrimidinone derivatives
DK2938194T3 (da) 2012-12-28 2020-01-02 Adama Makhteshim Ltd N-(substituerede)-5-fluor-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidin-1 (2h)-carboxylatderivater
JP6336480B2 (ja) * 2012-12-28 2018-06-06 アダマ・マクテシム・リミテッド 1−(置換ベンゾイル)−5−フルオロ−4−イミノ−3−メチル−3,4−ジヒドロピリミジン−2(1h)−オンの誘導体
US9321734B2 (en) 2012-12-28 2016-04-26 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxamide derivatives
RU2644014C2 (ru) 2012-12-31 2018-02-07 Адама Мактешим Лтд. Производные 3-алкил-5-фтор-4-замещенного-имино-3,4-дигидропиримидин-2(н)-она в качестве фунгицидов
EA029457B1 (ru) 2013-12-31 2018-03-30 Адама Мактешим Лтд. Синергетические фунгицидные смеси и композиции для борьбы с грибами
MX392211B (es) 2013-12-31 2025-03-21 Adama Makhteshim Ltd 5-flúor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparación.
WO2016040193A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof
JP6982748B2 (ja) 2015-11-06 2021-12-17 バイオスプライス セラピューティクス インコーポレイテッド 2−(1H−インダゾール−3−イル)−3H−イミダゾ[4,5−c]ピリジンおよびそれらの抗炎症的使用
KR102477407B1 (ko) 2016-06-01 2022-12-13 사뮤메드, 엘엘씨 N-(5-(3-(7-(3-플루오로페닐)-3h-이미다조[4,5-c]피리딘-2-일)-1h-인다졸-5-일)피리딘-3-일)-3-메틸부탄아미드를 제조하기 위한 공정
AU2018320492C1 (en) 2017-07-17 2023-07-13 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
AU2019374510A1 (en) 2018-11-05 2021-06-17 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
UY38890A (es) 2019-09-23 2021-04-30 Adama Makhteshim Ltd Procedimiento para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
BR9708314A (pt) * 1996-03-11 1999-08-03 Novartis Ag Pesticida
WO2004037159A2 (en) * 2002-10-23 2004-05-06 Obetherapy Biotechnology Compounds, compositions and methods for modulating fat metabolism
ES2566327T3 (es) * 2007-04-27 2016-04-12 Daiichi Sankyo Company, Limited Derivados de anillo aromático de 6 miembros que contiene nitrógeno y productos farmacéuticos que contienen los mismos
EP2647287A1 (en) * 2008-08-01 2013-10-09 Dow AgroSciences LLC Use of 5-fluorocytosine and its derivatives as fungicides

Also Published As

Publication number Publication date
ZA201305992B (en) 2014-10-29
NZ597638A (en) 2014-06-27
KR20120043069A (ko) 2012-05-03
PT2462133E (pt) 2014-12-26
PL2462133T3 (pl) 2015-03-31
CN102548979A (zh) 2012-07-04
AU2010279408A1 (en) 2012-02-09
CA2769251A1 (en) 2011-02-10
IN2012DN00695A (OSRAM) 2015-06-19
ECSP12011651A (es) 2012-03-30
IL217954A (en) 2016-02-29
CL2012000314A1 (es) 2012-10-05
MX2012001623A (es) 2012-04-11
EA022930B1 (ru) 2016-03-31
JP2013501726A (ja) 2013-01-17
HN2012000261A (es) 2015-01-05
BR112012002807A2 (pt) 2015-10-13
NI201200019A (es) 2012-05-22
IL217954A0 (en) 2012-03-29
EP2462133A4 (en) 2013-01-16
WO2011017544A1 (en) 2011-02-10
CN102548979B (zh) 2015-05-13
US8318758B2 (en) 2012-11-27
CA2769251C (en) 2018-05-15
EP2462133A1 (en) 2012-06-13
US20110034491A1 (en) 2011-02-10
EP2462133B1 (en) 2014-09-24
UA106086C2 (uk) 2014-07-25
KR101792286B1 (ko) 2017-10-31
BR112012002807B1 (pt) 2018-07-10
AU2010279408B2 (en) 2015-09-10
RS53658B1 (sr) 2015-04-30
CR20120033A (es) 2012-03-22
BR112012002807A8 (pt) 2017-07-11
JP5818791B2 (ja) 2015-11-18
PE20120689A1 (es) 2012-06-06
EA201270255A1 (ru) 2012-07-30
ES2506169T3 (es) 2014-10-13
DK2462133T3 (en) 2015-01-05
HK1172892A1 (en) 2013-05-03

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