NZ265304A - 3[(1-substituted-piperidin-4-yl)thio]-1-substituted-1h-indole derivatives - Google Patents

3[(1-substituted-piperidin-4-yl)thio]-1-substituted-1h-indole derivatives

Info

Publication number
NZ265304A
NZ265304A NZ265304A NZ26530494A NZ265304A NZ 265304 A NZ265304 A NZ 265304A NZ 265304 A NZ265304 A NZ 265304A NZ 26530494 A NZ26530494 A NZ 26530494A NZ 265304 A NZ265304 A NZ 265304A
Authority
NZ
New Zealand
Prior art keywords
formula
group
radical
thio
indole
Prior art date
Application number
NZ265304A
Other languages
English (en)
Inventor
Nicole Bru-Magniez
Dominique Potin
Jean-Marie Teulon
Original Assignee
Union Pharma Scient Appl
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Union Pharma Scient Appl filed Critical Union Pharma Scient Appl
Publication of NZ265304A publication Critical patent/NZ265304A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Rheumatology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
NZ265304A 1993-05-18 1994-04-13 3[(1-substituted-piperidin-4-yl)thio]-1-substituted-1h-indole derivatives NZ265304A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9305966A FR2705346B1 (fr) 1993-05-18 1993-05-18 Nouveaux dérivés de pipéridinyl thio indole, leurs procédés de préparation, compositions pharmaceutiques les contenant, utiles notamment comme antalgiques .

Publications (1)

Publication Number Publication Date
NZ265304A true NZ265304A (en) 1997-02-24

Family

ID=9447241

Family Applications (1)

Application Number Title Priority Date Filing Date
NZ265304A NZ265304A (en) 1993-05-18 1994-04-13 3[(1-substituted-piperidin-4-yl)thio]-1-substituted-1h-indole derivatives

Country Status (15)

Country Link
US (1) US5317025A (Sortimente)
EP (1) EP0699195A1 (Sortimente)
JP (1) JPH09500611A (Sortimente)
CN (1) CN1124026A (Sortimente)
AU (1) AU6571594A (Sortimente)
CA (1) CA2161021A1 (Sortimente)
CZ (1) CZ304195A3 (Sortimente)
EE (1) EE9400296A (Sortimente)
FI (1) FI954931A7 (Sortimente)
FR (1) FR2705346B1 (Sortimente)
HU (1) HUT74866A (Sortimente)
MD (1) MD522G2 (Sortimente)
NZ (1) NZ265304A (Sortimente)
TW (1) TW257756B (Sortimente)
WO (1) WO1994026736A1 (Sortimente)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK139593D0 (da) * 1993-12-16 1993-12-16 Lundbeck & Co As H Compounds
CA2195850A1 (en) * 1994-08-03 1996-02-15 Guillaume Lebaut Substituted indoles
US5521196A (en) * 1994-10-05 1996-05-28 Eli Lilly And Company 5-HT1F agonists for the treatment of migraine
TR199700993T1 (xx) * 1995-03-20 1998-03-21 Eli Lilly And Company 5-ikameli-3-(1,2,3,6-tetrahidropridin-4-il)- ve 3-(piperidin-4-il)-1H-indoller: yeni 5-HT1F agonistler.
TWI328009B (en) 2003-05-21 2010-08-01 Glaxo Group Ltd Quinoline derivatives as phosphodiesterase inhibitors
EP1838311A1 (en) * 2004-12-24 2007-10-03 Prosidion Limited G-protein coupled receptor (gpr116) agonists and use thereof for treating obesity and diabetes
BRPI0613505A2 (pt) * 2005-06-30 2011-01-11 Prosidion Ltd agonistas de gpcr
CL2008000018A1 (es) * 2007-01-04 2008-08-01 Prosidion Ltd Compuestos derivados de heterociclos de nitrogeno y oxigeno, agonistas de gpcr; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento de la obesidad, diabetes, sindrome metabolico, hiperlipidemia, toleranci
PE20081849A1 (es) * 2007-01-04 2009-01-26 Prosidion Ltd Derivados de piperidin-4-il-propoxi-benzamida como agonistas de gpcr
CN102917707A (zh) * 2010-05-06 2013-02-06 默沙东公司 可用作faah调节剂的氮杂吲哚衍生物
KR20180034466A (ko) 2015-07-02 2018-04-04 호리즌 오펀 엘엘씨 Ado-저항성 시스테아민 유사체 및 그의 용도
CN104945305A (zh) * 2015-07-03 2015-09-30 北京石油化工学院 一种实现吲哚类化合物选择性芳巯基化的方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB925429A (en) * 1960-04-01 1963-05-08 Irwin Neisler & Co Indole derivatives
US3264311A (en) * 1963-05-02 1966-08-02 Upjohn Co Esters of 3-(aminosulfinyl) indole-2-carboxylic acids

Also Published As

Publication number Publication date
HU9503281D0 (en) 1996-01-29
FI954931A0 (fi) 1995-10-17
CA2161021A1 (en) 1994-11-24
FI954931L (fi) 1995-11-20
HUT74866A (en) 1997-02-28
AU6571594A (en) 1994-12-12
US5317025A (en) 1994-05-31
MD522F1 (en) 1996-04-30
WO1994026736A1 (fr) 1994-11-24
TW257756B (Sortimente) 1995-09-21
MD522G2 (ro) 1997-01-31
FI954931A7 (fi) 1995-11-20
FR2705346A1 (fr) 1994-11-25
EP0699195A1 (fr) 1996-03-06
JPH09500611A (ja) 1997-01-21
CZ304195A3 (en) 1996-03-13
EE9400296A (et) 1996-04-15
CN1124026A (zh) 1996-06-05
FR2705346B1 (fr) 1995-08-11

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