EE9400296A - Piperidinüültioindooli derivaadid, ravimvormid, aktiivne valuvaigisti, nende valmistamise meetodid - Google Patents

Piperidinüültioindooli derivaadid, ravimvormid, aktiivne valuvaigisti, nende valmistamise meetodid

Info

Publication number
EE9400296A
EE9400296A EE9400296A EE9400296A EE9400296A EE 9400296 A EE9400296 A EE 9400296A EE 9400296 A EE9400296 A EE 9400296A EE 9400296 A EE9400296 A EE 9400296A EE 9400296 A EE9400296 A EE 9400296A
Authority
EE
Estonia
Prior art keywords
piperidinylthioindole
derivatives
preparation
methods
dosage forms
Prior art date
Application number
EE9400296A
Other languages
English (en)
Inventor
Bru-Magniez Nicole
Potin Dominique
Teulon Jean-Marie
Original Assignee
Laboratoires Upsa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Laboratoires Upsa filed Critical Laboratoires Upsa
Publication of EE9400296A publication Critical patent/EE9400296A/et

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
EE9400296A 1993-05-18 1994-11-23 Piperidinüültioindooli derivaadid, ravimvormid, aktiivne valuvaigisti, nende valmistamise meetodid EE9400296A (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9305966A FR2705346B1 (fr) 1993-05-18 1993-05-18 Nouveaux dérivés de pipéridinyl thio indole, leurs procédés de préparation, compositions pharmaceutiques les contenant, utiles notamment comme antalgiques .
PCT/FR1994/000410 WO1994026736A1 (fr) 1993-05-18 1994-04-13 Derives de piperidinyl thio indole comme antalgiques

Publications (1)

Publication Number Publication Date
EE9400296A true EE9400296A (et) 1996-04-15

Family

ID=9447241

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9400296A EE9400296A (et) 1993-05-18 1994-11-23 Piperidinüültioindooli derivaadid, ravimvormid, aktiivne valuvaigisti, nende valmistamise meetodid

Country Status (15)

Country Link
US (1) US5317025A (et)
EP (1) EP0699195A1 (et)
JP (1) JPH09500611A (et)
CN (1) CN1124026A (et)
AU (1) AU6571594A (et)
CA (1) CA2161021A1 (et)
CZ (1) CZ304195A3 (et)
EE (1) EE9400296A (et)
FI (1) FI954931A (et)
FR (1) FR2705346B1 (et)
HU (1) HUT74866A (et)
MD (1) MD522G2 (et)
NZ (1) NZ265304A (et)
TW (1) TW257756B (et)
WO (1) WO1994026736A1 (et)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK139593D0 (da) * 1993-12-16 1993-12-16 Lundbeck & Co As H Compounds
AU3162695A (en) * 1994-08-03 1996-03-04 Asta Medica Aktiengesellschaft Indol, indazol, pyridopyrrol and pyridopyrazol derivatives with anti-asthmatic, anti-allergic, anti-inflammatory and immunomodulating effects
US5521196A (en) * 1994-10-05 1996-05-28 Eli Lilly And Company 5-HT1F agonists for the treatment of migraine
CA2215322A1 (en) * 1995-03-20 1996-09-26 Stephen Warren Kaldor 5-substituted-3-(1,2,3,6-tetrahydropyridin-4-yl)-and 3-(piperidin-4-yl)-1h-indoles: new 5-ht1f agonists
TWI328009B (en) 2003-05-21 2010-08-01 Glaxo Group Ltd Quinoline derivatives as phosphodiesterase inhibitors
MX2007007553A (es) * 2004-12-24 2007-08-15 Prosidion Ltd Agonistas del receptor acoplado a proteina g (gpr116) y uso de los mismos para tratar obesidad y diabetes.
KR20080027908A (ko) * 2005-06-30 2008-03-28 프로시디온 리미티드 Gpcr 효능제
CL2008000017A1 (es) * 2007-01-04 2008-08-01 Prosidion Ltd Compuestos derivados de heterociclos de nitrogeno y oxigeno, agonistas de gpcr; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento de la obesidad, diabetes, sindrome metabolico, hiperlipidemia, toleranci
CL2008000018A1 (es) * 2007-01-04 2008-08-01 Prosidion Ltd Compuestos derivados de heterociclos de nitrogeno y oxigeno, agonistas de gpcr; composicion farmaceutica que comprende a dicho compuesto; y uso del compuesto para el tratamiento de la obesidad, diabetes, sindrome metabolico, hiperlipidemia, toleranci
US20130059850A1 (en) * 2010-05-06 2013-03-07 Merck Sharp & Dohme Corp. Aza-indole derivatives useful as modulators of faah
RU2022103033A (ru) 2015-07-02 2022-04-01 ХОРАЙЗОН ОРФАН ЭлЭлСи Цистеаминдиоксигеназа-резистентные аналоги цистеамина и их применение
CN104945305A (zh) * 2015-07-03 2015-09-30 北京石油化工学院 一种实现吲哚类化合物选择性芳巯基化的方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB925429A (en) * 1960-04-01 1963-05-08 Irwin Neisler & Co Indole derivatives
US3264311A (en) * 1963-05-02 1966-08-02 Upjohn Co Esters of 3-(aminosulfinyl) indole-2-carboxylic acids

Also Published As

Publication number Publication date
EP0699195A1 (fr) 1996-03-06
MD522F1 (en) 1996-04-30
US5317025A (en) 1994-05-31
HUT74866A (en) 1997-02-28
WO1994026736A1 (fr) 1994-11-24
NZ265304A (en) 1997-02-24
CZ304195A3 (en) 1996-03-13
FR2705346B1 (fr) 1995-08-11
CN1124026A (zh) 1996-06-05
CA2161021A1 (en) 1994-11-24
TW257756B (et) 1995-09-21
FI954931A (fi) 1995-11-20
FR2705346A1 (fr) 1994-11-25
MD522G2 (ro) 1997-01-31
AU6571594A (en) 1994-12-12
JPH09500611A (ja) 1997-01-21
FI954931A0 (fi) 1995-10-17
HU9503281D0 (en) 1996-01-29

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