NO991776L - Aminotiofenkarboksylsyreamider og anvendelse derav som fosfodiesteraseinhibitorer - Google Patents

Aminotiofenkarboksylsyreamider og anvendelse derav som fosfodiesteraseinhibitorer

Info

Publication number
NO991776L
NO991776L NO991776A NO991776A NO991776L NO 991776 L NO991776 L NO 991776L NO 991776 A NO991776 A NO 991776A NO 991776 A NO991776 A NO 991776A NO 991776 L NO991776 L NO 991776L
Authority
NO
Norway
Prior art keywords
acid amides
phosphodiesterase inhibitors
aminothiophenecarboxylic
aminothiophenecarboxylic acid
phosphodiesterase
Prior art date
Application number
NO991776A
Other languages
English (en)
Norwegian (no)
Other versions
NO991776D0 (no
Inventor
Rochus Jonas
Pierre Schelling
Franz-Werner Kluxen
Maria Christadler
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of NO991776D0 publication Critical patent/NO991776D0/no
Publication of NO991776L publication Critical patent/NO991776L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/62Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/68Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
NO991776A 1996-10-15 1999-04-14 Aminotiofenkarboksylsyreamider og anvendelse derav som fosfodiesteraseinhibitorer NO991776L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19642451A DE19642451A1 (de) 1996-10-15 1996-10-15 Aminothiophencarbonsäureamide
PCT/EP1997/005531 WO1998016521A1 (de) 1996-10-15 1997-10-08 Aminothiophencarbonsäureamide und ihre verwendung als phosphodiesterase inhibitoren

Publications (2)

Publication Number Publication Date
NO991776D0 NO991776D0 (no) 1999-04-14
NO991776L true NO991776L (no) 1999-06-09

Family

ID=7808775

Family Applications (1)

Application Number Title Priority Date Filing Date
NO991776A NO991776L (no) 1996-10-15 1999-04-14 Aminotiofenkarboksylsyreamider og anvendelse derav som fosfodiesteraseinhibitorer

Country Status (25)

Country Link
US (1) US6143777A (cs)
EP (1) EP0934301B1 (cs)
JP (1) JP4243352B2 (cs)
KR (1) KR100479811B1 (cs)
CN (1) CN1110493C (cs)
AR (1) AR009985A1 (cs)
AT (1) ATE202347T1 (cs)
AU (1) AU725741B2 (cs)
BR (1) BR9712321A (cs)
CA (1) CA2268886C (cs)
CZ (1) CZ297253B6 (cs)
DE (2) DE19642451A1 (cs)
DK (1) DK0934301T3 (cs)
ES (1) ES2159851T3 (cs)
GR (1) GR3036341T3 (cs)
HU (1) HUP9904703A3 (cs)
NO (1) NO991776L (cs)
PL (1) PL192109B1 (cs)
PT (1) PT934301E (cs)
RU (1) RU2184731C2 (cs)
SI (1) SI0934301T1 (cs)
SK (1) SK283807B6 (cs)
TW (1) TW438791B (cs)
WO (1) WO1998016521A1 (cs)
ZA (1) ZA979199B (cs)

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EP2258359A3 (en) 2005-08-26 2011-04-06 Braincells, Inc. Neurogenesis by muscarinic receptor modulation with sabcomelin
CA2625153A1 (en) 2005-10-21 2007-04-26 Braincells, Inc. Modulation of neurogenesis by pde inhibition
JP2009513672A (ja) 2005-10-31 2009-04-02 ブレインセルス,インコーポレイティド 神経発生のgaba受容体媒介調節
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RU2501795C1 (ru) * 2012-10-01 2013-12-20 Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Пермский государственный национальный исследовательский университет" N-R-АМИДЫ (Z)-2[(3-ЭТОКСИКАРБОНИЛ)-4,5,6,7-ТЕТРАГИДРОБЕНЗО[b]ТИЕН-2-ИЛ)АМИНО]-4-ФЕНИЛ-4-ОКСОБУТ-2-ЕНОВЫХ КИСЛОТ, ОБЛАДАЮЩИЕ АНАЛЬГЕТИЧЕСКОЙ АКТИВНОСТЬЮ
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Also Published As

Publication number Publication date
DE59703869D1 (de) 2001-07-26
TW438791B (en) 2001-06-07
NO991776D0 (no) 1999-04-14
HUP9904703A2 (hu) 2001-05-28
BR9712321A (pt) 1999-08-31
CN1233246A (zh) 1999-10-27
KR100479811B1 (ko) 2005-03-30
KR20000049154A (ko) 2000-07-25
WO1998016521A1 (de) 1998-04-23
JP2001501957A (ja) 2001-02-13
CN1110493C (zh) 2003-06-04
DK0934301T3 (da) 2001-10-08
ATE202347T1 (de) 2001-07-15
SK283807B6 (sk) 2004-02-03
JP4243352B2 (ja) 2009-03-25
EP0934301A1 (de) 1999-08-11
CA2268886C (en) 2008-05-20
SI0934301T1 (en) 2001-12-31
US6143777A (en) 2000-11-07
PT934301E (pt) 2001-10-31
AU725741B2 (en) 2000-10-19
PL192109B1 (pl) 2006-08-31
PL332802A1 (en) 1999-10-11
CZ124099A3 (cs) 1999-07-14
HK1020724A1 (en) 2000-05-19
ZA979199B (en) 1998-05-11
HUP9904703A3 (en) 2001-06-28
GR3036341T3 (en) 2001-11-30
DE19642451A1 (de) 1998-04-16
EP0934301B1 (de) 2001-06-20
AU4945197A (en) 1998-05-11
RU2184731C2 (ru) 2002-07-10
SK43299A3 (en) 2000-04-10
AR009985A1 (es) 2000-05-17
CA2268886A1 (en) 1998-04-23
CZ297253B6 (cs) 2006-10-11
ES2159851T3 (es) 2001-10-16

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