NO991204L - FremgangsmÕte ved fremstilling av azitromycindihydrat - Google Patents
FremgangsmÕte ved fremstilling av azitromycindihydratInfo
- Publication number
- NO991204L NO991204L NO991204A NO991204A NO991204L NO 991204 L NO991204 L NO 991204L NO 991204 A NO991204 A NO 991204A NO 991204 A NO991204 A NO 991204A NO 991204 L NO991204 L NO 991204L
- Authority
- NO
- Norway
- Prior art keywords
- preparation
- azithromycin dihydrate
- azithromycin
- dihydrate
- azytromycin
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 3
- VQEMDSRIOVZAOM-UHFFFAOYSA-N 4-(4-methylsulfonylphenyl)-1,3-thiazol-2-amine Chemical compound C1=CC(S(=O)(=O)C)=CC=C1C1=CSC(N)=N1 VQEMDSRIOVZAOM-UHFFFAOYSA-N 0.000 title abstract 2
- 229960004924 azithromycin dihydrate Drugs 0.000 title abstract 2
- 238000002360 preparation method Methods 0.000 title abstract 2
- 230000003115 biocidal effect Effects 0.000 abstract 1
- 238000002955 isolation Methods 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 150000004682 monohydrates Chemical group 0.000 abstract 1
- 239000000825 pharmaceutical preparation Substances 0.000 abstract 1
- 229940127557 pharmaceutical product Drugs 0.000 abstract 1
- 239000002904 solvent Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PT102130A PT102130A (pt) | 1998-03-13 | 1998-03-13 | Processo de preparacao de dihidrato de azitromicina |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO991204D0 NO991204D0 (no) | 1999-03-11 |
| NO991204L true NO991204L (no) | 1999-09-14 |
Family
ID=20085748
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO991204A NO991204L (no) | 1998-03-13 | 1999-03-11 | FremgangsmÕte ved fremstilling av azitromycindihydrat |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP0941999A3 (de) |
| JP (1) | JPH11322776A (de) |
| KR (1) | KR19990077826A (de) |
| CN (1) | CN1232037A (de) |
| AU (1) | AU1952599A (de) |
| CA (1) | CA2265412A1 (de) |
| HU (1) | HUP9900550A3 (de) |
| NO (1) | NO991204L (de) |
| PT (1) | PT102130A (de) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HRP20020231A2 (en) | 2002-03-18 | 2003-12-31 | Pliva D D | ISOSTRUCTURAL PSEUDOPOLYMORPHS OF 9-DEOXO-9a-AZA-9a-METHYL-9a-HOMOERYTHROMYCIN A |
| DE20023815U1 (de) * | 1999-06-29 | 2006-06-08 | Sandoz Ag | Azithromycin enthaltende Zusammensetzungen |
| ES2177373B1 (es) | 1999-11-26 | 2003-11-01 | Astur Pharma Sa | Preparacion de azitromicina en su forma no cristalina |
| ATE388159T1 (de) | 2000-01-04 | 2008-03-15 | Teva Pharma | Verfahren zur herstellung von azithromycin- dihydrat |
| ES2162764B1 (es) * | 2000-05-17 | 2003-04-01 | Ercros Ind Sa | Forma polimorfica del dihidrato de azitromicina, y su procedimiento deobtencion. |
| UA76967C2 (uk) * | 2000-11-27 | 2006-10-16 | Сандоз Аг | Азитроміцин у формі моногідрату, фармацевтична композиція та спосіб його одержання |
| CZ303343B6 (cs) * | 2000-11-27 | 2012-08-08 | Sandoz Ag | Zpusob prípravy azithromycinu ve forme monohydrátu |
| IN190080B (de) * | 2001-01-29 | 2003-06-07 | Alembic Ltd | |
| KR100491183B1 (ko) * | 2001-03-21 | 2005-05-25 | 한미약품 주식회사 | 아지트로마이신의 제조방법 및 이 방법에 사용되는9-데옥소-9에이-아자-9에이-호모에리트로마이신 에이의결정성 수화물 |
| KR100431431B1 (ko) * | 2001-04-25 | 2004-05-14 | 한미약품 주식회사 | 아지트로마이신 수화물의 1,2-프로필렌글리콜 내포화합물,그의 제조방법 및 그의 약학적 조성물 |
| BR0209918A (pt) | 2001-05-22 | 2004-03-30 | Pfizer Prod Inc | Formas cristalinas da azitromicina |
| US6861413B2 (en) | 2001-05-22 | 2005-03-01 | Pfizer Inc. | Stable non-dihydrate azithromycin oral suspensions |
| EP1490382A4 (de) * | 2002-04-03 | 2007-09-12 | Hanmi Pharm Ind Co Ltd | Verfahren zur herstellung von azithromycin und dabei verwendetes kristallines 9-desoxo-9a-aza-9a-homoerythromycin-a-hydrat |
| GB2395482A (en) * | 2003-07-03 | 2004-05-26 | Jubilant Organosys Ltd | Process for preparing non-hygroscopic azithromycin dihydrate |
| US7164023B2 (en) * | 2003-09-04 | 2007-01-16 | Wockhardt Limited | Benzoquinolizine-2-carboxylic acid arginine salt tetrahydrate |
| RU2260012C1 (ru) * | 2004-01-29 | 2005-09-10 | Открытое акционерное общество "Акционерное курганское общество медицинских препаратов и изделий "Синтез" | Способ кристаллизации азитромицина дигидрата |
| US7468428B2 (en) | 2004-03-17 | 2008-12-23 | App Pharmaceuticals, Llc | Lyophilized azithromycin formulation |
| US7683162B2 (en) | 2004-08-30 | 2010-03-23 | Taro Pharmaceutical Industries Limited | Process of preparing a crystalline azithromycin monohydrate |
| CN101624412B (zh) | 2008-07-10 | 2012-07-04 | 刘力 | 大环内酯类衍生物及其制备和用途 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| RU2066324C1 (ru) * | 1987-07-09 | 1996-09-10 | Пфайзер Инк. | Кристаллический дигидрат азитромицина и способ его получения |
| ES2122905B1 (es) * | 1996-07-11 | 1999-11-16 | Astur Pharma Sa | Sintesis de 11,12-hidrogenoortoborato de 9-desoxo-9a-aza-11,12-desoxi-9a-metil-9a-homoeritromicina a. un procedimiento para la preparacion de 9-desoxo-9a-aza-9a-metil-9a-homoeritromicina a dihidrato (azitromicina dihidrato). |
-
1998
- 1998-03-13 PT PT102130A patent/PT102130A/pt not_active Application Discontinuation
-
1999
- 1999-03-08 HU HU9900550A patent/HUP9900550A3/hu unknown
- 1999-03-10 AU AU19525/99A patent/AU1952599A/en not_active Abandoned
- 1999-03-10 EP EP99301788A patent/EP0941999A3/de not_active Withdrawn
- 1999-03-11 JP JP11065443A patent/JPH11322776A/ja active Pending
- 1999-03-11 NO NO991204A patent/NO991204L/no unknown
- 1999-03-12 CA CA002265412A patent/CA2265412A1/en not_active Abandoned
- 1999-03-12 CN CN99105538A patent/CN1232037A/zh active Pending
- 1999-03-12 KR KR1019990008297A patent/KR19990077826A/ko not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| KR19990077826A (ko) | 1999-10-25 |
| PT102130A (pt) | 1999-09-30 |
| HUP9900550A2 (hu) | 1999-09-28 |
| HUP9900550A3 (en) | 2000-04-28 |
| NO991204D0 (no) | 1999-03-11 |
| EP0941999A3 (de) | 1999-10-13 |
| EP0941999A2 (de) | 1999-09-15 |
| HU9900550D0 (en) | 1999-04-28 |
| AU1952599A (en) | 1999-09-23 |
| CA2265412A1 (en) | 1999-09-13 |
| JPH11322776A (ja) | 1999-11-24 |
| CN1232037A (zh) | 1999-10-20 |
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