NO982363L - Fosfonsyrederivater med metallopeptidasehemmende aktivitet - Google Patents

Fosfonsyrederivater med metallopeptidasehemmende aktivitet

Info

Publication number
NO982363L
NO982363L NO982363A NO982363A NO982363L NO 982363 L NO982363 L NO 982363L NO 982363 A NO982363 A NO 982363A NO 982363 A NO982363 A NO 982363A NO 982363 L NO982363 L NO 982363L
Authority
NO
Norway
Prior art keywords
aryl
heterocycle
inhibitory activity
acid derivatives
phosphonic acid
Prior art date
Application number
NO982363A
Other languages
English (en)
Norwegian (no)
Other versions
NO982363D0 (no
Inventor
Gabriele Norcini
Daniela Botta
Francesco Santangelo
Original Assignee
Zambon Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon Spa filed Critical Zambon Spa
Publication of NO982363D0 publication Critical patent/NO982363D0/no
Publication of NO982363L publication Critical patent/NO982363L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06008—Dipeptides with the first amino acid being neutral
    • C07K5/06017—Dipeptides with the first amino acid being neutral and aliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Detergent Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cosmetics (AREA)
NO982363A 1995-11-23 1998-05-25 Fosfonsyrederivater med metallopeptidasehemmende aktivitet NO982363L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT95MI002430A IT1276161B1 (it) 1995-11-23 1995-11-23 Derivati dell'acido fosfonico ad attivita' inibitrice delle metallopeptidasi
PCT/EP1996/004911 WO1997019102A1 (en) 1995-11-23 1996-11-11 Phosphonic acid derivatives with metallopeptidase inhibitory activity

Publications (2)

Publication Number Publication Date
NO982363D0 NO982363D0 (no) 1998-05-25
NO982363L true NO982363L (no) 1998-07-22

Family

ID=11372578

Family Applications (1)

Application Number Title Priority Date Filing Date
NO982363A NO982363L (no) 1995-11-23 1998-05-25 Fosfonsyrederivater med metallopeptidasehemmende aktivitet

Country Status (23)

Country Link
US (1) US6548480B1 (pt)
EP (1) EP0868428B1 (pt)
JP (1) JP2000501079A (pt)
KR (1) KR100458359B1 (pt)
CN (1) CN1127513C (pt)
AT (1) ATE234856T1 (pt)
AU (1) AU707570B2 (pt)
BR (1) BR9611465A (pt)
CA (1) CA2249343A1 (pt)
CZ (1) CZ291926B6 (pt)
DE (1) DE69626846T2 (pt)
DK (1) DK0868428T3 (pt)
EA (1) EA000743B1 (pt)
ES (1) ES2192619T3 (pt)
HU (1) HUP0000080A3 (pt)
IL (1) IL124021A (pt)
IT (1) IT1276161B1 (pt)
MX (1) MX9803760A (pt)
NO (1) NO982363L (pt)
PT (1) PT868428E (pt)
SI (1) SI0868428T1 (pt)
WO (1) WO1997019102A1 (pt)
ZA (1) ZA969774B (pt)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3973748B2 (ja) 1998-01-14 2007-09-12 花王株式会社 発毛抑制剤
JP4796296B2 (ja) * 2004-12-02 2011-10-19 インターナショナル・ビジネス・マシーンズ・コーポレーション Ｗｅｂページ・オーサリング装置、Ｗｅｂページ・オーサリング方法及びプログラム
KR101135332B1 (ko) * 2007-03-15 2012-04-17 닛코킨조쿠 가부시키가이샤 구리전해액 및 그것을 이용하여 얻어진 2층 플렉시블 기판

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4432972A (en) * 1981-08-03 1984-02-21 E. R. Squibb & Sons, Inc. Phosphonamidate compounds
ATE22692T1 (de) * 1981-08-03 1986-10-15 Squibb & Sons Inc Phosphonamidate verbindungen.
IT1274673B (it) * 1994-04-14 1997-07-24 Zambon Spa Derivati dell'acido fosfonico utili nel trattamento delle malattie car.iovascolari

Also Published As

Publication number Publication date
MX9803760A (es) 1998-09-30
EP0868428A1 (en) 1998-10-07
NO982363D0 (no) 1998-05-25
ITMI952430A1 (it) 1997-05-23
DE69626846T2 (de) 2003-12-24
AU707570B2 (en) 1999-07-15
AU7568996A (en) 1997-06-11
EA199800470A1 (ru) 1998-12-24
BR9611465A (pt) 1999-05-18
CN1127513C (zh) 2003-11-12
CZ158898A3 (cs) 1998-11-11
EA000743B1 (ru) 2000-02-28
CZ291926B6 (cs) 2003-06-18
ITMI952430A0 (pt) 1995-11-23
CA2249343A1 (en) 1997-05-29
KR19990071550A (ko) 1999-09-27
HUP0000080A2 (hu) 2001-04-28
ES2192619T3 (es) 2003-10-16
PT868428E (pt) 2003-06-30
EP0868428B1 (en) 2003-03-19
US6548480B1 (en) 2003-04-15
ZA969774B (en) 1997-06-17
HUP0000080A3 (en) 2001-05-28
IT1276161B1 (it) 1997-10-27
KR100458359B1 (ko) 2005-01-15
CN1202901A (zh) 1998-12-23
WO1997019102A1 (en) 1997-05-29
SI0868428T1 (en) 2003-06-30
DE69626846D1 (de) 2003-04-24
ATE234856T1 (de) 2003-04-15
JP2000501079A (ja) 2000-02-02
IL124021A (en) 2001-06-14
DK0868428T3 (da) 2003-07-21

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Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application