NO940928D0 - Nye 2-tiosubstituerte karbapenemer - Google Patents
Nye 2-tiosubstituerte karbapenemerInfo
- Publication number
- NO940928D0 NO940928D0 NO940928A NO940928A NO940928D0 NO 940928 D0 NO940928 D0 NO 940928D0 NO 940928 A NO940928 A NO 940928A NO 940928 A NO940928 A NO 940928A NO 940928 D0 NO940928 D0 NO 940928D0
- Authority
- NO
- Norway
- Prior art keywords
- thio
- new
- substituted carbapenems
- carbapenems
- substituted
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
- C07D307/04—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D307/18—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/30—Hetero atoms other than halogen
- C07D333/34—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D477/00—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
- C07D477/10—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D477/12—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6
- C07D477/14—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 3
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic System
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
- C07F9/65611—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings containing the ring system (X = CH2, O, S, NH) optionally with an additional double bond and/or substituents, e.g. penicillins and analogs
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H11/00—Compounds containing saccharide radicals esterified by inorganic acids; Metal salts thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/582—Recycling of unreacted starting or intermediate materials
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US3368493A | 1993-03-16 | 1993-03-16 |
Publications (3)
Publication Number | Publication Date |
---|---|
NO940928D0 true NO940928D0 (no) | 1994-03-15 |
NO940928L NO940928L (no) | 1994-09-19 |
NO311939B1 NO311939B1 (no) | 2002-02-18 |
Family
ID=21871845
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO19940928A NO311939B1 (no) | 1993-03-16 | 1994-03-15 | Nye 2-tiosubstituerte karbapenemer, anvendelse derav og farmasöytisk blanding |
Country Status (19)
Country | Link |
---|---|
US (4) | US5602118A (no) |
EP (1) | EP0617036A3 (no) |
JP (1) | JPH06321948A (no) |
KR (1) | KR100353751B1 (no) |
CN (3) | CN1482122A (no) |
AU (1) | AU676877B2 (no) |
CA (1) | CA2118961A1 (no) |
CZ (1) | CZ290494B6 (no) |
FI (1) | FI106718B (no) |
HU (2) | HUT67741A (no) |
IL (1) | IL108939A0 (no) |
NO (1) | NO311939B1 (no) |
NZ (1) | NZ260102A (no) |
PL (1) | PL179558B1 (no) |
RU (1) | RU2130457C1 (no) |
SG (2) | SG91908A1 (no) |
SK (1) | SK31694A3 (no) |
TW (1) | TW474937B (no) |
ZA (1) | ZA941828B (no) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0951894B1 (en) * | 1998-04-23 | 2010-07-14 | DENTSPLY DETREY GmbH | Storage stable polymerizable compositions |
DK1101497T3 (da) * | 1998-08-04 | 2008-03-31 | Schering Plough Animal Health | Stabiliserende olieagtige præparationer af tobicillin (beta-lactam antibiotikum) |
US6162924A (en) | 1999-04-09 | 2000-12-19 | Eastman Chemical Company | Process for halohydrin preparation |
JP2003531138A (ja) * | 2000-03-21 | 2003-10-21 | アセロジエニクス・インコーポレイテツド | 生物学的疾患の治療のためのn−置換ジチオカルバメート |
US6649756B2 (en) | 2000-07-13 | 2003-11-18 | Wyeth, Five Giralda Farms | Process improvement in the preparation of (4r, 5s, 6s)-3-[[(2r,3r)-2-[[[(s)-2-amino-3-methyl-1-oxobutyl]amino]methyl]tetrahydro-3-furanyl]thio]-6-[(r)-1-hydroxyethyl]-4-methyl-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid |
US20020049315A1 (en) * | 2000-09-06 | 2002-04-25 | Williams John M. | Crystalline forms of carbapenem intermediates |
US7232924B2 (en) * | 2001-06-11 | 2007-06-19 | Xenoport, Inc. | Methods for synthesis of acyloxyalkyl derivatives of GABA analogs |
US7186855B2 (en) * | 2001-06-11 | 2007-03-06 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
US8048917B2 (en) | 2005-04-06 | 2011-11-01 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
US6818787B2 (en) * | 2001-06-11 | 2004-11-16 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
US20050152887A1 (en) * | 2004-01-14 | 2005-07-14 | Doctor's Signature Sales And Marketing International Corp. [Dba Life Force International | Protonic formulation |
KR100621782B1 (ko) * | 2004-06-14 | 2006-09-19 | 한국과학기술연구원 | 1-베타메틸카바페넴 유도체 및 이의 제조방법 |
EP1941873A4 (en) * | 2005-09-22 | 2012-09-26 | Meiji Seika Kaisha | METALLO-BETA-Lactamase INHIBITORS |
US8119667B2 (en) * | 2005-12-29 | 2012-02-21 | Schering-Plough Animal Health Corporation | Carbonates of fenicol antibiotics |
US8093378B2 (en) * | 2006-04-28 | 2012-01-10 | Kaneka Corporation | Crystallization method for intermediates of carbapenem antibiotics |
EA200900068A1 (ru) * | 2006-07-28 | 2009-06-30 | Крка, Товарна Здравил, Д. Д., Ново Место | Способ получения формы i кандесартана цилексетила |
US20110046101A1 (en) * | 2008-03-17 | 2011-02-24 | Dmitrienko Gary I | Bate-lactamase inhibitors |
US20110118462A1 (en) * | 2009-11-18 | 2011-05-19 | Guangzhou Baiyunshan Pharmaceutical Co., Ltd. Guangzhou Baiyunshan Pharmaceutical Factory | N-heterocyclic substituent-containing antibiotic, preparation and use thereof |
JP6457523B2 (ja) | 2013-12-04 | 2019-01-23 | エヴォテック・インターナショナル・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングEvotec International GmbH | 医薬組成物のためのスルホキシイミン置換キナゾリン |
WO2017158616A1 (en) | 2016-03-16 | 2017-09-21 | Orchid Pharma Ltd. | Carbapenem compounds |
Family Cites Families (29)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2656362A (en) * | 1951-07-05 | 1953-10-20 | Allied Lab Inc | Preparation of 2-halogenated tetrahydrothiophene 1, 1-dioxides |
GB1441177A (en) * | 1973-12-13 | 1976-06-30 | Beheer Bv Pfw | Sulphur-containing flavouring agents |
CS176325B1 (no) * | 1975-01-31 | 1977-06-30 | ||
US4347368A (en) * | 1977-10-19 | 1982-08-31 | Merck & Co., Inc. | 3-Substituted-6-substituted-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid |
US4260627A (en) * | 1978-10-24 | 1981-04-07 | Merck & Co., Inc. | 1-, 6- And 2-substituted-1-carba-2-penem-3-carboxylic acids |
DK446179A (da) * | 1978-10-24 | 1980-05-29 | Merck & Co Inc | Fremgangsmaade til fremstilling af substituerede 1-carbadethiapen-2-em-3-carboxylsyrer |
US4232036A (en) * | 1978-10-24 | 1980-11-04 | Merck & Co., Inc. | 6-, 1- and 2-Substituted-1-carbadethiapen-2-em-3-carboxylic acids |
US4341706A (en) * | 1980-10-10 | 1982-07-27 | Merck & Co., Inc. | Process for the preparation of carbapenem antibiotics |
US4745188A (en) * | 1980-11-21 | 1988-05-17 | Merck & Co., Inc. | Process for preparing 3-substituted-6-substituted-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid |
EP0060612A1 (en) * | 1981-02-04 | 1982-09-22 | Beecham Group Plc | Process for the preparation of azabicyclo(3.2.0)-hept-2-ene derivatives |
NZ201471A (en) * | 1981-08-10 | 1985-09-13 | Merck & Co Inc | Antibacterial compositions containing penems and dipeptidase inhibitors |
US4552873A (en) * | 1981-08-19 | 1985-11-12 | Sankyo Company Limited | Carbapenem compounds, and compositions containing them |
CA1283906C (en) * | 1983-05-09 | 1991-05-07 | Makoto Sunagawa | .beta.-LACTAM COMPOUNDS AND PRODUCTION THEREOF |
JPS60202886A (ja) * | 1984-03-27 | 1985-10-14 | Sankyo Co Ltd | 1―置換カルバペネム―3―カルボン酸誘導体 |
US4696923A (en) * | 1984-04-23 | 1987-09-29 | Merck & Co., Inc. | 6-[1-hydroxyethyl]-2-SR8 -1-methyl-1-carbadethiapen-2-em-3-carboxylic acids |
US4820817A (en) * | 1984-09-10 | 1989-04-11 | Merck & Co., Inc. | Process for preparing 3-substituted-6-substituted-7-oxo-1-azabicycl(3.2.0)-hept-2-ene-2-carboxylic acid |
EP0182213B1 (en) * | 1984-11-08 | 1990-09-26 | Sumitomo Pharmaceuticals Company, Limited | Carbapenem compounds and production thereof |
JPH075463B2 (ja) * | 1985-03-09 | 1995-01-25 | サントリー株式会社 | 抗菌剤 |
US4665169A (en) * | 1985-09-11 | 1987-05-12 | Bristol-Myers Company | Carbapenem antibiotics |
EP0368259B1 (en) * | 1988-11-08 | 1994-07-20 | Daiichi Pharmaceutical Co., Ltd. | Carbapenem derivatives |
HUT63167A (en) * | 1989-03-28 | 1993-07-28 | Pfizer | Process for producing antibacterial 2-carbapenem derivatives and pharmaceutical compositions comprising same as active ingredient |
US5321020A (en) * | 1989-03-28 | 1994-06-14 | Pfizer Inc. | Antibacterial 2-carbapenem derivatives |
CA2022382A1 (en) * | 1989-08-02 | 1991-02-03 | Susumu Nakagawa | Piperidylthiocarbapenem derivatives |
EP0942000B1 (en) * | 1989-10-24 | 2004-06-23 | Isis Pharmaceuticals, Inc. | 2'-Modified oligonucleotides |
WO1991009860A1 (en) * | 1989-12-28 | 1991-07-11 | Banyu Pharmaceutical Co., Ltd. | New carbapenem derivative |
CA2037767A1 (en) * | 1990-03-23 | 1991-09-24 | Mark D. Wittman | Conversion of amines to hydroxylamines |
US5116833A (en) * | 1990-10-19 | 1992-05-26 | Bristol-Myers Squibb Company | Antibiotic c-3 dithioacetal-substituted carbapenem compounds, compositions, and methods of use thereof |
JPH04368386A (ja) * | 1991-06-18 | 1992-12-21 | Sankyo Co Ltd | 1−メチルカルバペネム−3−カルボン酸の製造法 |
GB9202298D0 (en) * | 1992-02-04 | 1992-03-18 | Ici Plc | Antibiotic compounds |
-
1994
- 1994-01-26 US US08/182,781 patent/US5602118A/en not_active Expired - Lifetime
- 1994-02-17 SG SG200101813A patent/SG91908A1/en unknown
- 1994-02-17 EP EP94102400A patent/EP0617036A3/en not_active Withdrawn
- 1994-02-17 SG SG1996003099A patent/SG77541A1/en unknown
- 1994-03-11 HU HU9400724A patent/HUT67741A/hu unknown
- 1994-03-11 IL IL10893994A patent/IL108939A0/xx unknown
- 1994-03-14 CA CA002118961A patent/CA2118961A1/en not_active Abandoned
- 1994-03-15 FI FI941215A patent/FI106718B/fi not_active IP Right Cessation
- 1994-03-15 KR KR1019940005156A patent/KR100353751B1/ko not_active IP Right Cessation
- 1994-03-15 AU AU57831/94A patent/AU676877B2/en not_active Ceased
- 1994-03-15 PL PL94302626A patent/PL179558B1/pl unknown
- 1994-03-15 JP JP6069945A patent/JPH06321948A/ja active Pending
- 1994-03-15 RU RU94008616/04A patent/RU2130457C1/ru not_active IP Right Cessation
- 1994-03-15 ZA ZA941828A patent/ZA941828B/xx unknown
- 1994-03-15 CZ CZ1994586A patent/CZ290494B6/cs not_active IP Right Cessation
- 1994-03-15 NZ NZ260102A patent/NZ260102A/en unknown
- 1994-03-15 NO NO19940928A patent/NO311939B1/no not_active IP Right Cessation
- 1994-03-16 SK SK316-94A patent/SK31694A3/sk unknown
- 1994-03-16 CN CNA031457169A patent/CN1482122A/zh active Pending
- 1994-03-16 CN CN94102266A patent/CN1041633C/zh not_active Expired - Fee Related
- 1994-03-28 TW TW083102728A patent/TW474937B/zh not_active IP Right Cessation
-
1995
- 1995-05-19 US US08/445,388 patent/US5750735A/en not_active Expired - Lifetime
- 1995-05-23 US US08/448,295 patent/US5744465A/en not_active Expired - Lifetime
- 1995-05-23 US US08/448,052 patent/US5623081A/en not_active Expired - Lifetime
- 1995-06-30 HU HU95P/P00616P patent/HU211883A9/hu unknown
-
1998
- 1998-06-10 CN CNB981147682A patent/CN1136208C/zh not_active Expired - Fee Related
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM1K | Lapsed by not paying the annual fees |