NO932218D0 - Imidazopyridiner - Google Patents

Imidazopyridiner

Info

Publication number
NO932218D0
NO932218D0 NO932218A NO932218A NO932218D0 NO 932218 D0 NO932218 D0 NO 932218D0 NO 932218 A NO932218 A NO 932218A NO 932218 A NO932218 A NO 932218A NO 932218 D0 NO932218 D0 NO 932218D0
Authority
NO
Norway
Prior art keywords
imidazopyridines
Prior art date
Application number
NO932218A
Other languages
English (en)
Other versions
NO300924B1 (no
NO932218L (no
Inventor
Werner Mederski
Dieter Dorsch
Norbert Beier
Pierre Schelling
Ingeborg Lues
Klaus-Otto Minck
Mathias Osswald
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of NO932218D0 publication Critical patent/NO932218D0/no
Publication of NO932218L publication Critical patent/NO932218L/no
Publication of NO300924B1 publication Critical patent/NO300924B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO932218A 1992-06-17 1993-06-16 Imidazopyridinderivater, farmasöytiske preparater og anvendelse av slike forbindelser til fremstilling av et legemiddel NO300924B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4219818 1992-06-17
DE4305602A DE4305602A1 (de) 1992-06-17 1993-02-24 Imidazopyridine

Publications (3)

Publication Number Publication Date
NO932218D0 true NO932218D0 (no) 1993-06-16
NO932218L NO932218L (no) 1993-12-20
NO300924B1 NO300924B1 (no) 1997-08-18

Family

ID=25915778

Family Applications (1)

Application Number Title Priority Date Filing Date
NO932218A NO300924B1 (no) 1992-06-17 1993-06-16 Imidazopyridinderivater, farmasöytiske preparater og anvendelse av slike forbindelser til fremstilling av et legemiddel

Country Status (15)

Country Link
US (1) US5476857A (no)
EP (1) EP0574846A3 (no)
JP (1) JPH0656832A (no)
KR (1) KR940005623A (no)
CN (1) CN1038511C (no)
AU (1) AU669895B2 (no)
CA (1) CA2098473A1 (no)
CZ (1) CZ283081B6 (no)
DE (1) DE4305602A1 (no)
HU (1) HUT64761A (no)
MX (1) MX9303597A (no)
NO (1) NO300924B1 (no)
PL (1) PL173777B1 (no)
SK (1) SK57893A3 (no)
TW (1) TW254941B (no)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5798364A (en) * 1992-03-26 1998-08-25 Merck Patent Gesellschaft Mit Beschrankter Haftung Imidazopyridines
DE4141788A1 (de) * 1991-12-18 1993-06-24 Merck Patent Gmbh Imidazopyridine
DE4242459A1 (de) * 1992-12-16 1994-06-23 Merck Patent Gmbh Imidazopyridine
DE4318813A1 (de) * 1993-06-07 1994-12-08 Merck Patent Gmbh Imidazopyridine
DE4339868A1 (de) * 1993-11-23 1995-05-24 Merck Patent Gmbh Imidazopyridazine
DE4341453A1 (de) * 1993-12-06 1995-06-08 Merck Patent Gmbh Imidazopyridine
DE4432860A1 (de) * 1994-09-15 1996-03-21 Merck Patent Gmbh Imidazopyridine
US6060480A (en) * 1996-08-30 2000-05-09 Yoshitomi Pharmaceutical Industries, Ltd. Preventives/remedies for muscle tissue degenerations
US5975601A (en) * 1998-04-22 1999-11-02 O. Ames Co. One-piece hand-held gardening tool
DE19845153A1 (de) 1998-10-01 2000-04-06 Merck Patent Gmbh Imidazo[4,5]-pyridin-4-on-derivate
US20040242568A1 (en) 2003-03-25 2004-12-02 Syrrx, Inc. Dipeptidyl peptidase inhibitors
US7678909B1 (en) 2003-08-13 2010-03-16 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
US7169926B1 (en) 2003-08-13 2007-01-30 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
US7790736B2 (en) 2003-08-13 2010-09-07 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
US7790734B2 (en) 2003-09-08 2010-09-07 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
US7732446B1 (en) 2004-03-11 2010-06-08 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
CN102134229B (zh) 2004-03-15 2020-08-04 武田药品工业株式会社 二肽基肽酶抑制剂
WO2005118555A1 (en) 2004-06-04 2005-12-15 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
WO2006019965A2 (en) 2004-07-16 2006-02-23 Takeda San Diego, Inc. Dipeptidyl peptidase inhibitors
WO2006068978A2 (en) 2004-12-21 2006-06-29 Takeda Pharmaceutial Company Limited Dipeptidyl peptidase inhibitors
PL1942898T5 (pl) 2005-09-14 2014-10-31 Takeda Pharmaceuticals Co Inhibitory peptydazy dipeptydylowej do leczenia cukrzycy
CN102675221A (zh) 2005-09-16 2012-09-19 武田药品工业株式会社 用于制备嘧啶二酮衍生物的方法中的中间体
WO2007112347A1 (en) 2006-03-28 2007-10-04 Takeda Pharmaceutical Company Limited Dipeptidyl peptidase inhibitors
US8324383B2 (en) 2006-09-13 2012-12-04 Takeda Pharmaceutical Company Limited Methods of making polymorphs of benzoate salt of 2-[[6-[(3R)-3-amino-1-piperidinyl]-3,4-dihydro-3-methyl-2,4-dioxo-1(2H)-pyrimidinyl]methyl]-benzonitrile
TW200838536A (en) 2006-11-29 2008-10-01 Takeda Pharmaceutical Polymorphs of succinate salt of 2-[6-(3-amino-piperidin-1-yl)-3-methyl-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-ylmethy]-4-fluor-benzonitrile and methods of use therefor
US8093236B2 (en) 2007-03-13 2012-01-10 Takeda Pharmaceuticals Company Limited Weekly administration of dipeptidyl peptidase inhibitors
CA2711461A1 (en) * 2008-02-08 2009-08-13 Merck Sharp & Dohme Corp. Angiotensin ii receptor antagonists

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5036048A (en) * 1986-03-07 1991-07-30 Schering Corporation Angiotensin II receptor blockers as antiglaucoma agents
US4880804A (en) * 1988-01-07 1989-11-14 E. I. Du Pont De Nemours And Company Angiotensin II receptor blocking benzimidazoles
IL94390A (en) * 1989-05-30 1996-03-31 Merck & Co Inc The 6-membered trans-nitrogen-containing heterocycles are compressed with imidazo and pharmaceutical preparations containing them
US5332744A (en) * 1989-05-30 1994-07-26 Merck & Co., Inc. Substituted imidazo-fused 6-membered heterocycles as angiotensin II antagonists
US5240928A (en) * 1989-07-03 1993-08-31 Merck & Co., Inc. Substituted quinazolinones as angiotensin II antagonists
IE70593B1 (en) * 1989-09-29 1996-12-11 Eisai Co Ltd Biphenylmethane derivative the use of it and pharmacological compositions containing same
US5240938A (en) * 1991-02-13 1993-08-31 Merck & Co., Inc. Angiotensin II antagonists incorporating a substituted pyridoimidazolyl ring
US5124335A (en) * 1991-01-30 1992-06-23 Merck & Co., Inc. Substituted pyrollo-fused 6 membered heterocycles as angiotensin ii antagonists
DE4110019C2 (de) * 1991-03-27 2000-04-13 Merck Patent Gmbh Imidazopyridine, Verfahren zu ihrer Herstellung und diese enthaltende pharmazeutische Zubereitungen
AU644540B2 (en) * 1991-09-10 1993-12-09 Tanabe Seiyaku Co., Ltd. Imidazopyridine derivatives and process for preparation thereof
DE4141788A1 (de) * 1991-12-18 1993-06-24 Merck Patent Gmbh Imidazopyridine
DE4211474A1 (de) * 1992-04-06 1993-10-07 Merck Patent Gmbh Imidazopyridine
DE4242459A1 (de) * 1992-12-16 1994-06-23 Merck Patent Gmbh Imidazopyridine

Also Published As

Publication number Publication date
DE4305602A1 (de) 1993-12-23
JPH0656832A (ja) 1994-03-01
CN1038511C (zh) 1998-05-27
NO300924B1 (no) 1997-08-18
CZ114593A3 (en) 1994-01-19
AU669895B2 (en) 1996-06-27
EP0574846A3 (en) 1994-07-06
CA2098473A1 (en) 1993-12-18
CN1082545A (zh) 1994-02-23
PL299368A1 (en) 1994-02-21
HUT64761A (en) 1994-02-28
EP0574846A2 (de) 1993-12-22
HU9301766D0 (en) 1993-09-28
CZ283081B6 (cs) 1997-12-17
KR940005623A (ko) 1994-03-22
PL173777B1 (pl) 1998-04-30
MX9303597A (es) 1994-01-31
US5476857A (en) 1995-12-19
AU4123893A (en) 1993-12-23
NO932218L (no) 1993-12-20
SK57893A3 (en) 1994-01-12
TW254941B (no) 1995-08-21

Similar Documents

Publication Publication Date Title
NO934622L (no) Imidazopyridiner
NO932218L (no) Imidazopyridiner
DK88892D0 (da) Forbindelse
NO924890D0 (no) Imidazopyridiner
AT399443B (de) Sportschuh
NO942095D0 (no) Imidazopyridiner
NO931302L (no) Imidazopyridiner
ATA236892A (de) Rotornut
NO933804D0 (no) Imidazopyridiner
FI933203A0 (fi) Kinolin- och naftyridinprolaekemedel
ATA80192A (de) Rohr-nippel-verbindung
DE59301550D1 (de) Flansch-Rohrverbindung
ATA227792A (de) Sportschuh
KR940000399U (ko) 납골단지
KR940000228U (ko) 재치대
DK113492D0 (da) Forbindelse
BR9201149A (pt) Mutlimovel
BR7200318U (pt) Cabide sanfonado
BR9201140A (pt) Tarara batedora
BR9200611A (pt) Hidrocofre
BR9200554A (pt) Lixoduto
BR9200298A (pt) Microsisten-telesupervisao
BR9200296A (pt) Varre-lava
BR9200295A (pt) Aurissima
BR9200231A (pt) Agrupador