NO912982D0 - Fremgangsmaate for fremstilling av 4-amino-delta4'6-steroider. - Google Patents

Fremgangsmaate for fremstilling av 4-amino-delta4'6-steroider.

Info

Publication number
NO912982D0
NO912982D0 NO912982A NO912982A NO912982D0 NO 912982 D0 NO912982 D0 NO 912982D0 NO 912982 A NO912982 A NO 912982A NO 912982 A NO912982 A NO 912982A NO 912982 D0 NO912982 D0 NO 912982D0
Authority
NO
Norway
Prior art keywords
steroids
amino
delta4
procedure
preparation
Prior art date
Application number
NO912982A
Other languages
English (en)
Other versions
NO180197C (no
NO180197B (no
NO912982L (no
Inventor
Philip Marvin Weintraub
Original Assignee
Merrell Dow Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US07/671,555 external-priority patent/US5143909A/en
Priority claimed from US07/720,899 external-priority patent/US5130424A/en
Application filed by Merrell Dow Pharma filed Critical Merrell Dow Pharma
Publication of NO912982D0 publication Critical patent/NO912982D0/no
Publication of NO912982L publication Critical patent/NO912982L/no
Publication of NO180197B publication Critical patent/NO180197B/no
Publication of NO180197C publication Critical patent/NO180197C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0005—Oxygen-containing hetero ring
    • C07J71/001—Oxiranes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
    • C07J41/0011—Unsubstituted amino radicals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Reproductive Health (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
NO912982A 1990-08-01 1991-07-31 Analogifremgangsmåte for fremstilling av terapeutisk aktive 4-amino-<Delta>4'6-steroider NO180197C (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US56141090A 1990-08-01 1990-08-01
US07/671,555 US5143909A (en) 1991-03-19 1991-03-19 Aminosteroids in a method for inhibiting c17-20 lyase
US07/720,899 US5130424A (en) 1990-08-01 1991-07-02 4-amino-delta-4,6-steroids and their use as 5 alpha-reductase inhibitors

Publications (4)

Publication Number Publication Date
NO912982D0 true NO912982D0 (no) 1991-07-31
NO912982L NO912982L (no) 1992-02-03
NO180197B NO180197B (no) 1996-11-25
NO180197C NO180197C (no) 1997-03-05

Family

ID=27415853

Family Applications (1)

Application Number Title Priority Date Filing Date
NO912982A NO180197C (no) 1990-08-01 1991-07-31 Analogifremgangsmåte for fremstilling av terapeutisk aktive 4-amino-<Delta>4'6-steroider

Country Status (17)

Country Link
EP (1) EP0469547B1 (no)
JP (1) JP3021818B2 (no)
CN (1) CN1031574C (no)
AT (1) ATE138073T1 (no)
AU (1) AU642757B2 (no)
CA (1) CA2048243C (no)
DE (1) DE69119502T2 (no)
DK (1) DK0469547T3 (no)
ES (1) ES2089063T3 (no)
FI (1) FI102378B1 (no)
GR (1) GR3020268T3 (no)
HU (1) HU210042B (no)
IE (1) IE75199B1 (no)
IL (1) IL98998A (no)
NO (1) NO180197C (no)
NZ (1) NZ239141A (no)
PT (1) PT98519B (no)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2118222T3 (es) * 1991-12-20 1998-09-16 Glaxo Wellcome Inc Inhibidores de 5-alfa-testosterona reductasa.
US5302589A (en) * 1992-08-07 1994-04-12 Glaxo, Inc. Heterocyclic inhibitors of 5-α-testosterone reductase
US5486511A (en) * 1993-05-25 1996-01-23 Merrell Dow Pharmaceuticals Inc. 4-amino-17β-(cyclopropyloxy)androst-4-en-3-one, 4-amino-17β-(cyclopropylamino)androst-4-en-3-one and related compounds as C17-20 lyase and 5α-reductase
TW369521B (en) * 1993-09-17 1999-09-11 Smithkline Beecham Corp Androstenone derivative
US5356935A (en) * 1993-12-13 1994-10-18 Eli Lilly And Company Reduced phenanthrenes
AU686793B2 (en) * 1994-05-02 1998-02-12 Merrell Pharmaceuticals Inc. Process for the preparation of 4-amino- 4-3-ketosteroids via 4-nitro-delta 4-3-ketosteroids
US5541322A (en) * 1994-10-14 1996-07-30 Glaxo Wellcome Inc. Synthesis of 6-azaandrostenones
AU6087700A (en) * 1999-07-15 2001-02-05 Procter & Gamble Company, The Nitrogen-containing steroid compounds and their use to regulate hair growth
JP6353939B1 (ja) * 2017-02-15 2018-07-04 横関油脂工業株式会社 油状組成物、その製法、油性基剤および皮膚外用剤

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1154008A (en) * 1979-05-02 1983-09-20 Thomas R. Blohm STEROID 5.alpha.-REDUCTASE INHIBITORS
GB8503940D0 (en) * 1985-02-15 1985-03-20 Erba Farmitalia 4-substituted androstendione derivatives

Also Published As

Publication number Publication date
JPH05320189A (ja) 1993-12-03
IE912706A1 (en) 1992-02-12
AU8135691A (en) 1992-02-06
CA2048243A1 (en) 1992-02-02
HUT59157A (en) 1992-04-28
NO180197C (no) 1997-03-05
DE69119502T2 (de) 1996-09-26
ES2089063T3 (es) 1996-10-01
GR3020268T3 (en) 1996-09-30
DK0469547T3 (da) 1996-06-10
EP0469547A2 (en) 1992-02-05
FI913658A (fi) 1992-02-02
NZ239141A (en) 1994-04-27
DE69119502D1 (de) 1996-06-20
FI102378B (fi) 1998-11-30
CA2048243C (en) 2003-04-08
EP0469547A3 (en) 1992-06-03
EP0469547B1 (en) 1996-05-15
JP3021818B2 (ja) 2000-03-15
AU642757B2 (en) 1993-10-28
FI913658A0 (fi) 1991-07-31
HU210042B (en) 1995-01-30
HU912559D0 (en) 1992-01-28
NO180197B (no) 1996-11-25
FI102378B1 (fi) 1998-11-30
CN1031574C (zh) 1996-04-17
IL98998A0 (en) 1992-07-15
PT98519A (pt) 1992-06-30
NO912982L (no) 1992-02-03
IE75199B1 (en) 1997-08-27
PT98519B (pt) 1999-01-29
CN1059150A (zh) 1992-03-04
IL98998A (en) 1996-01-19
ATE138073T1 (de) 1996-06-15

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Legal Events

Date Code Title Description
MM1K Lapsed by not paying the annual fees

Free format text: LAPSED IN JANUARY 2001