NO864740D0 - Amorfe, ikke-krystallinske former av terapeutisk virksomme benzimidazolderivater. - Google Patents

Amorfe, ikke-krystallinske former av terapeutisk virksomme benzimidazolderivater.

Info

Publication number
NO864740D0
NO864740D0 NO864740A NO864740A NO864740D0 NO 864740 D0 NO864740 D0 NO 864740D0 NO 864740 A NO864740 A NO 864740A NO 864740 A NO864740 A NO 864740A NO 864740 D0 NO864740 D0 NO 864740D0
Authority
NO
Norway
Prior art keywords
crystallinic
amorph
forms
therapeutically effective
benzimidazold
Prior art date
Application number
NO864740A
Other languages
English (en)
Norwegian (no)
Inventor
Richard Allen Runkel
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex Inc filed Critical Syntex Inc
Publication of NO864740D0 publication Critical patent/NO864740D0/no
Priority to NO880083A priority Critical patent/NO880083D0/no
Priority to NO881862A priority patent/NO881862D0/no
Priority to NO881861A priority patent/NO881861D0/no

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/32Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/30Nitrogen atoms not forming part of a nitro radical
    • C07D235/32Benzimidazole-2-carbamic acids, unsubstituted or substituted; Esters thereof; Thio-analogues thereof

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Inorganic Chemistry (AREA)
  • Dermatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO864740A 1985-11-27 1986-11-26 Amorfe, ikke-krystallinske former av terapeutisk virksomme benzimidazolderivater. NO864740D0 (no)

Priority Applications (3)

Application Number Priority Date Filing Date Title
NO880083A NO880083D0 (no) 1985-11-27 1988-01-11 Fremgangsmaate for fremstilling av amorfe benzimidazolderivater med forbedret opploeselighet og anthelmintisk aktivitet.
NO881862A NO881862D0 (no) 1985-11-27 1988-04-28 Fremgangsmaate for fremstilling av amorfe benzimidazolderivater med forbedret opploeselighet og anthelmintisk aktivitet.
NO881861A NO881861D0 (no) 1985-11-27 1988-04-28 Fremgangsmaate for fremstilling av amorfe benzimidazolderivater med forbedret opploeselighet og anthelmintisk aktivitet.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US80250885A 1985-11-27 1985-11-27

Publications (1)

Publication Number Publication Date
NO864740D0 true NO864740D0 (no) 1986-11-26

Family

ID=25183897

Family Applications (1)

Application Number Title Priority Date Filing Date
NO864740A NO864740D0 (no) 1985-11-27 1986-11-26 Amorfe, ikke-krystallinske former av terapeutisk virksomme benzimidazolderivater.

Country Status (14)

Country Link
EP (1) EP0224257A1 (fi)
JP (1) JPS62155264A (fi)
CN (1) CN86108096A (fi)
AU (1) AU6569986A (fi)
BR (1) BR8605798A (fi)
DD (1) DD252540A5 (fi)
DK (1) DK569686A (fi)
FI (1) FI864813A (fi)
HU (1) HU198025B (fi)
IL (1) IL80768A0 (fi)
IN (1) IN164294B (fi)
NO (1) NO864740D0 (fi)
PT (1) PT83811B (fi)
ZA (1) ZA868962B (fi)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102452987A (zh) * 2010-10-28 2012-05-16 桂林南药股份有限公司 一种不定形晶型阿苯达唑的制备方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS601101A (ja) * 1983-06-15 1985-01-07 Yuukou Yakuhin Kogyo Kk 水性懸濁農薬製剤
DE3347579A1 (de) * 1983-12-30 1985-07-11 Hoechst Ag, 6230 Frankfurt Zubereitungen schwer wasserloeslicher anthelminthika und verfahren zu ihrer herstellung

Also Published As

Publication number Publication date
HUT42076A (en) 1987-06-29
ZA868962B (en) 1988-07-27
DK569686A (da) 1987-05-28
FI864813A (fi) 1987-05-28
AU6569986A (en) 1987-06-04
FI864813A0 (fi) 1986-11-26
DD252540A5 (de) 1987-12-23
HU198025B (en) 1989-07-28
IL80768A0 (en) 1987-02-27
IN164294B (fi) 1989-02-11
DK569686D0 (da) 1986-11-26
CN86108096A (zh) 1987-07-08
PT83811B (en) 1988-03-15
JPS62155264A (ja) 1987-07-10
BR8605798A (pt) 1987-08-25
PT83811A (en) 1986-12-01
EP0224257A1 (en) 1987-06-03

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