NO864741D0 - Amorfe, ikke-krystallinske former av terapeutisk virksomme benzimidazolderivater. - Google Patents
Amorfe, ikke-krystallinske former av terapeutisk virksomme benzimidazolderivater.Info
- Publication number
- NO864741D0 NO864741D0 NO864741A NO864741A NO864741D0 NO 864741 D0 NO864741 D0 NO 864741D0 NO 864741 A NO864741 A NO 864741A NO 864741 A NO864741 A NO 864741A NO 864741 D0 NO864741 D0 NO 864741D0
- Authority
- NO
- Norway
- Prior art keywords
- crystallinic
- amorph
- forms
- therapeutically effective
- benzimidazold
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/26—Oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/28—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/30—Nitrogen atoms not forming part of a nitro radical
- C07D235/32—Benzimidazole-2-carbamic acids, unsubstituted or substituted; Esters thereof; Thio-analogues thereof
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Tropical Medicine & Parasitology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Inorganic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Priority Applications (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| NO874739A NO874739D0 (no) | 1985-11-27 | 1987-11-13 | Fremgangsmaate for fremstilling av amorfe benzimidazolderivater med forbedret opploeselighet og anthelmintisk aktivitet. |
| NO881788A NO881788D0 (no) | 1985-11-27 | 1988-04-22 | Fremgangsmaate for fremtilling av amorfe benzimidazolderivater med forbedret opploeselighet og anthelmintisk aktivitet |
| NO881787A NO881787D0 (no) | 1985-11-27 | 1988-04-22 | Fremgangsmaate for femstilling av amorfe benzimidazolderivater med fobedret opploeselighet og anthelmintisk aktivitet. |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US80279885A | 1985-11-27 | 1985-11-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO864741D0 true NO864741D0 (no) | 1986-11-26 |
Family
ID=25184726
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO864741A NO864741D0 (no) | 1985-11-27 | 1986-11-26 | Amorfe, ikke-krystallinske former av terapeutisk virksomme benzimidazolderivater. |
Country Status (11)
| Country | Link |
|---|---|
| EP (1) | EP0224249A1 (no) |
| JP (1) | JPS62155263A (no) |
| KR (1) | KR870004967A (no) |
| AU (1) | AU6569886A (no) |
| DK (1) | DK569786A (no) |
| FI (1) | FI864812A (no) |
| HU (1) | HUT43575A (no) |
| IL (1) | IL80767A0 (no) |
| NO (1) | NO864741D0 (no) |
| PT (1) | PT83812B (no) |
| ZA (1) | ZA868963B (no) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5419897A (en) * | 1993-04-09 | 1995-05-30 | Buckman Laboratories International, Inc. | Ionene polymers as anthelmintics in animals |
| US5861142A (en) * | 1996-03-25 | 1999-01-19 | Schick; Mary Pichler | Method for promoting hair, nail, and skin keratinization |
| US6350786B1 (en) * | 1998-09-22 | 2002-02-26 | Hoffmann-La Roche Inc. | Stable complexes of poorly soluble compounds in ionic polymers |
| ATE313952T1 (de) * | 1999-06-04 | 2006-01-15 | Nufarm Ltd | Stabile biozidale zusammensetzung |
| EP2596792A1 (en) * | 2002-10-16 | 2013-05-29 | Takeda Pharmaceutical Company Limited | Stable solid preparations |
| JP2006513159A (ja) | 2002-11-01 | 2006-04-20 | メルク エンド カムパニー インコーポレーテッド | アンドロゲン受容体モジュレーターとしてのカルボニルアミノ−ベンズイミダゾール誘導体 |
| US9095585B2 (en) | 2011-07-21 | 2015-08-04 | Bristol-Myers Squibb Company | Bioavailable compositions of amorphous piperidinyl compounds |
| EA202192753A1 (ru) | 2019-04-11 | 2022-01-11 | Бристол-Маерс Сквибб Компани | Повышенная эффективность аморфных твердых и солюбилизированных составов для достижения терапевтических концентраций в плазме |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS601101A (ja) * | 1983-06-15 | 1985-01-07 | Yuukou Yakuhin Kogyo Kk | 水性懸濁農薬製剤 |
| DE3347579A1 (de) * | 1983-12-30 | 1985-07-11 | Hoechst Ag, 6230 Frankfurt | Zubereitungen schwer wasserloeslicher anthelminthika und verfahren zu ihrer herstellung |
-
1986
- 1986-11-26 PT PT83812A patent/PT83812B/pt unknown
- 1986-11-26 AU AU65698/86A patent/AU6569886A/en not_active Abandoned
- 1986-11-26 JP JP61283014A patent/JPS62155263A/ja active Pending
- 1986-11-26 HU HU864893A patent/HUT43575A/hu unknown
- 1986-11-26 IL IL80767A patent/IL80767A0/xx unknown
- 1986-11-26 NO NO864741A patent/NO864741D0/no unknown
- 1986-11-26 DK DK569786A patent/DK569786A/da not_active Application Discontinuation
- 1986-11-26 FI FI864812A patent/FI864812A/fi not_active IP Right Cessation
- 1986-11-26 KR KR860009984A patent/KR870004967A/ko not_active Application Discontinuation
- 1986-11-26 ZA ZA868963A patent/ZA868963B/xx unknown
- 1986-11-26 EP EP86116396A patent/EP0224249A1/en not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| JPS62155263A (ja) | 1987-07-10 |
| HUT43575A (en) | 1987-11-30 |
| ZA868963B (en) | 1988-07-27 |
| AU6569886A (en) | 1987-06-04 |
| FI864812A (fi) | 1987-05-28 |
| PT83812A (en) | 1986-12-01 |
| PT83812B (en) | 1988-03-15 |
| EP0224249A1 (en) | 1987-06-03 |
| IL80767A0 (en) | 1987-02-27 |
| DK569786D0 (da) | 1986-11-26 |
| DK569786A (da) | 1987-05-28 |
| FI864812A0 (fi) | 1986-11-26 |
| KR870004967A (ko) | 1987-06-02 |
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