HUT43575A - Process for producing amorphous benzimidazol derivatives and pharmaceutical compositions containing them - Google Patents

Process for producing amorphous benzimidazol derivatives and pharmaceutical compositions containing them

Info

Publication number
HUT43575A
HUT43575A HU864893A HU489386A HUT43575A HU T43575 A HUT43575 A HU T43575A HU 864893 A HU864893 A HU 864893A HU 489386 A HU489386 A HU 489386A HU T43575 A HUT43575 A HU T43575A
Authority
HU
Hungary
Prior art keywords
pharmaceutical compositions
compositions containing
producing amorphous
benzimidazol derivatives
benzimidazol
Prior art date
Application number
HU864893A
Other languages
English (en)
Inventor
Richard A Runkel
Original Assignee
Syntex Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syntex Inc filed Critical Syntex Inc
Publication of HUT43575A publication Critical patent/HUT43575A/hu

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/26Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38Cellulose; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/28Sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/30Nitrogen atoms not forming part of a nitro radical
    • C07D235/32Benzimidazole-2-carbamic acids, unsubstituted or substituted; Esters thereof; Thio-analogues thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Inorganic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HU864893A 1985-11-27 1986-11-26 Process for producing amorphous benzimidazol derivatives and pharmaceutical compositions containing them HUT43575A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US80279885A 1985-11-27 1985-11-27

Publications (1)

Publication Number Publication Date
HUT43575A true HUT43575A (en) 1987-11-30

Family

ID=25184726

Family Applications (1)

Application Number Title Priority Date Filing Date
HU864893A HUT43575A (en) 1985-11-27 1986-11-26 Process for producing amorphous benzimidazol derivatives and pharmaceutical compositions containing them

Country Status (11)

Country Link
EP (1) EP0224249A1 (hu)
JP (1) JPS62155263A (hu)
KR (1) KR870004967A (hu)
AU (1) AU6569886A (hu)
DK (1) DK569786A (hu)
FI (1) FI864812A (hu)
HU (1) HUT43575A (hu)
IL (1) IL80767A0 (hu)
NO (1) NO864741D0 (hu)
PT (1) PT83812B (hu)
ZA (1) ZA868963B (hu)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5419897A (en) * 1993-04-09 1995-05-30 Buckman Laboratories International, Inc. Ionene polymers as anthelmintics in animals
US5861142A (en) * 1996-03-25 1999-01-19 Schick; Mary Pichler Method for promoting hair, nail, and skin keratinization
US6350786B1 (en) * 1998-09-22 2002-02-26 Hoffmann-La Roche Inc. Stable complexes of poorly soluble compounds in ionic polymers
AR035550A1 (es) * 1999-06-04 2004-06-16 Nufarm Ltd Composiciones estables biocidas
US8697094B2 (en) * 2002-10-16 2014-04-15 Takeda Pharmaceutical Company Limited Stable solid preparations
US7622592B2 (en) 2002-11-01 2009-11-24 Merck & Co., Inc. Carbonylamino-benzimidazole derivatives as androgen receptor modulators
AR087277A1 (es) 2011-07-21 2014-03-12 Bristol Myers Squibb Co Composiciones biodisponibles de compuestos amorfos de piperidinilo, composicion farmaceutica, metodos
BR112021020257A2 (pt) 2019-04-11 2021-12-07 Bristol Myers Squibb Co Desempenho intensificado de sólido amorfo e formulações solubilizadas para realizar concentrações de plasma terapêutico

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS601101A (ja) * 1983-06-15 1985-01-07 Yuukou Yakuhin Kogyo Kk 水性懸濁農薬製剤
DE3347579A1 (de) * 1983-12-30 1985-07-11 Hoechst Ag, 6230 Frankfurt Zubereitungen schwer wasserloeslicher anthelminthika und verfahren zu ihrer herstellung

Also Published As

Publication number Publication date
NO864741D0 (no) 1986-11-26
EP0224249A1 (en) 1987-06-03
PT83812B (en) 1988-03-15
AU6569886A (en) 1987-06-04
KR870004967A (ko) 1987-06-02
IL80767A0 (en) 1987-02-27
DK569786A (da) 1987-05-28
FI864812A (fi) 1987-05-28
PT83812A (en) 1986-12-01
ZA868963B (en) 1988-07-27
FI864812A0 (fi) 1986-11-26
JPS62155263A (ja) 1987-07-10
DK569786D0 (da) 1986-11-26

Similar Documents

Publication Publication Date Title
HUT41790A (en) Process for producing beta-amino-purine derivatives and pharmaceutical compositions containing them
HUT48267A (en) Process for producing fluoro-citidin derivatives and pharmaceutical compositions containing them
HUT49316A (en) Process for producing didehydro-d3-vitamine derivatives and pharmaceutical compositions containing them
HUT40453A (en) Process for producing 11-beta-phenyl-gonanes and pharmaceutical compositions containing them
HUT51272A (en) Process for producing thiadiazin derivatives and pharmaceutical composirions containing them
HUT41772A (en) Process for producing /4-substituted-piperazinyl- and -homopiperazinyl/-pyridazines and pharmaceutical compositions containing them
HUT43825A (en) Process for producing quinolon-carboxylic acid derivatives and pharmaceutical compositions containing them
HUT44512A (en) Process for producing bensyl derivatives and pharmaceutical compositions containing them
HUT48887A (en) Process for producing cyclopentenyl-purin derivatives and pharmaceutical compositions containing them
HUT52061A (en) Process for producing isoquinoline derivatives and pharmaceutical compositions containing them
HUT56098A (en) Process for producing azanaphtalenesultame derivatives and pharmaceutical compositions containing them
HUT51277A (en) Process for producing anellated tetrahydropyridin-acetic acid derivatives and pharmaceutical compositions containing them
HUT42478A (en) Process for producing gamma-carboline derivatives and pharmaceutical compositions containing them
HUT59908A (en) Process for producing benzazepine- and benzo-thiazepine derivatives and pharmaceutical compositions containing them
HUT49317A (en) Process for producing 16-dehydro-d3-vitamine derivatives and pharmaceutical compositions containing them
GR860849B (en) 4-demethyl -4- epipodophyllotoxin derivatives process for their preparation and their use as medicaments
HUT47079A (en) Process for producing n-amino-butyl-n-phenyl-aryl-amide derivatives and pharmaceutical compositions containing them
HUT41035A (en) Process for producing cepheme derivatives and pharmaceutical compositions containing them
HUT48870A (en) Process for producing aminoalkoxyphenyl derivatives and pharmaceutical compositions comprising same
HUT41392A (en) Process for producing new imidazolyl-alkyl-guanidine derivatives and pharmaceutical compositions containing them
HUT43820A (en) Process for producing n-(-2-((-2-hydroxy-phenyl-)(-phenyl-)-methylene-aminosquare )-ethyl-)-acetamide derivatives and pharmaceutical compositions containing them
HUT39746A (en) Process for producing cephalosporin derivatives and pharmaceutical compositions containing them
HUT48244A (en) Process for producing isoxazol-3-carbolin derivatives and pharmaceutical compositions containing them
HUT58739A (en) Process for producing 3-oxo-3-/benzopyrano- or -thiopyrano-pyrazol-3-yl/-propionitril derivatives and pharmaceutical compositions containing them
HUT48270A (en) Process for producing new purine derivatives and pharmaceutical compositions containing them

Legal Events

Date Code Title Description
DFD9 Temporary protection cancelled due to non-payment of fee