NO332186B1 - Metansulfonsyresalt av pyrazolpyrimidinforbindelse, krystall derav, fremgangsmate for fremstilling av det samme, farmasoytisk preparat samt anvendelse derav - Google Patents

Metansulfonsyresalt av pyrazolpyrimidinforbindelse, krystall derav, fremgangsmate for fremstilling av det samme, farmasoytisk preparat samt anvendelse derav Download PDF

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Publication number
NO332186B1
NO332186B1 NO20056093A NO20056093A NO332186B1 NO 332186 B1 NO332186 B1 NO 332186B1 NO 20056093 A NO20056093 A NO 20056093A NO 20056093 A NO20056093 A NO 20056093A NO 332186 B1 NO332186 B1 NO 332186B1
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NO
Norway
Prior art keywords
crystal
chloro
disorder
methoxyphenyl
methyl
Prior art date
Application number
NO20056093A
Other languages
English (en)
Norwegian (no)
Other versions
NO20056093L (no
Inventor
Tetsuji Saitoh
Tomoyuki Hasegawa
Toshiaki Matsui
Hiroshi Araki
Tetsuo Obitsu
Masaki Okamoto
Yuichi Gemba
Yutaka Mikami
Original Assignee
Ono Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ono Pharmaceutical Co filed Critical Ono Pharmaceutical Co
Publication of NO20056093L publication Critical patent/NO20056093L/no
Publication of NO332186B1 publication Critical patent/NO332186B1/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
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    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
  • Pulmonology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Addiction (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Hematology (AREA)
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  • Psychology (AREA)
  • Anesthesiology (AREA)
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NO20056093A 2003-06-25 2005-12-21 Metansulfonsyresalt av pyrazolpyrimidinforbindelse, krystall derav, fremgangsmate for fremstilling av det samme, farmasoytisk preparat samt anvendelse derav NO332186B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2003181908 2003-06-25
PCT/JP2004/009263 WO2004113344A1 (ja) 2003-06-25 2004-06-24 ピラゾロピリミジン化合物のメタンスルホン酸塩、その結晶およびその製造方法

Publications (2)

Publication Number Publication Date
NO20056093L NO20056093L (no) 2006-03-24
NO332186B1 true NO332186B1 (no) 2012-07-23

Family

ID=33535237

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20056093A NO332186B1 (no) 2003-06-25 2005-12-21 Metansulfonsyresalt av pyrazolpyrimidinforbindelse, krystall derav, fremgangsmate for fremstilling av det samme, farmasoytisk preparat samt anvendelse derav

Country Status (19)

Country Link
US (1) US7947697B1 (zh)
EP (1) EP1637531B1 (zh)
JP (1) JP4655276B2 (zh)
KR (1) KR101082227B1 (zh)
CN (1) CN100422186C (zh)
AT (1) ATE478873T1 (zh)
AU (1) AU2004249629B2 (zh)
BR (1) BRPI0411923A (zh)
CA (1) CA2529561C (zh)
DE (1) DE602004028820D1 (zh)
ES (1) ES2349393T3 (zh)
IL (1) IL172697A (zh)
MX (1) MXPA05013917A (zh)
NO (1) NO332186B1 (zh)
NZ (1) NZ544301A (zh)
RU (1) RU2345995C2 (zh)
TW (1) TWI356058B (zh)
WO (1) WO2004113344A1 (zh)
ZA (1) ZA200510450B (zh)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2005061508A1 (ja) * 2003-12-22 2005-07-07 Ono Pharmaceutical Co., Ltd. 三環式複素環化合物およびその化合物を有効成分とする医薬
WO2005087775A1 (ja) * 2004-03-15 2005-09-22 Ono Pharmaceutical Co., Ltd. 三環式複素環化合物およびその化合物を有効成分として含有する医薬組成物
CN112225732B (zh) * 2019-07-15 2024-01-09 四川科瑞德制药股份有限公司 一种盐酸哌罗匹隆水合物晶型及其制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1030768C (zh) * 1990-10-09 1996-01-24 大塚制药株式会社 嘧啶衍生物或其药用盐的制备方法
EP0503099A4 (en) 1990-10-09 1993-12-01 Otsuka Pharmaceutical Co., Ltd. Pyrimidine derivative, production thereof, and androgen inhibitor
JPH05112571A (ja) 1990-10-19 1993-05-07 Otsuka Pharmaceut Co Ltd ピリミジン誘導体
KR100260292B1 (ko) 1995-09-28 2000-07-01 오쓰카 요시미쓰 진통제
ES2196820T3 (es) 1998-06-09 2003-12-16 Neurogen Corp Derivados de pirido(2,3-b)indolizina y aza-analogos de la misma; ligandos especificos de crf 1.
WO2000027850A2 (en) 1998-11-12 2000-05-18 Neurocrine Biosciences, Inc. Crf receptor antagonists and methods relating thereto
US6531475B1 (en) 1998-11-12 2003-03-11 Neurocrine Biosciences, Inc. CRF receptor antagonists and methods relating thereto
PT1129091E (pt) 1998-11-12 2003-02-28 Neurocrine Biosciences Inc Antagonistas de receptor de crf e metodos relacionados
EP1354884B1 (en) 2000-12-28 2007-10-10 Ono Pharmaceutical Co., Ltd. Cyclopenta[d]pyrazolo[1,5-a]pyrimidine compound as crf receptor antagonist

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Publication number Publication date
EP1637531B1 (en) 2010-08-25
AU2004249629A1 (en) 2004-12-29
CA2529561A1 (en) 2004-12-29
ZA200510450B (en) 2006-12-27
AU2004249629B2 (en) 2009-07-30
EP1637531A1 (en) 2006-03-22
WO2004113344A1 (ja) 2004-12-29
RU2345995C2 (ru) 2009-02-10
NO20056093L (no) 2006-03-24
IL172697A (en) 2013-05-30
IL172697A0 (en) 2006-04-10
TW200504064A (en) 2005-02-01
US7947697B1 (en) 2011-05-24
JP4655276B2 (ja) 2011-03-23
CN1842530A (zh) 2006-10-04
NZ544301A (en) 2008-08-29
CN100422186C (zh) 2008-10-01
KR20060026060A (ko) 2006-03-22
DE602004028820D1 (de) 2010-10-07
EP1637531A4 (en) 2008-09-03
BRPI0411923A (pt) 2006-08-15
CA2529561C (en) 2012-05-29
JPWO2004113344A1 (ja) 2006-07-27
ATE478873T1 (de) 2010-09-15
MXPA05013917A (es) 2006-03-09
ES2349393T3 (es) 2010-12-30
KR101082227B1 (ko) 2011-11-09
RU2006101986A (ru) 2006-07-27
TWI356058B (en) 2012-01-11

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