NO329414B1 - Farmasoytiske sammensetninger inneholdende flibanserin polymorf A, titandioksid og/eller talk - Google Patents
Farmasoytiske sammensetninger inneholdende flibanserin polymorf A, titandioksid og/eller talk Download PDFInfo
- Publication number
- NO329414B1 NO329414B1 NO20044547A NO20044547A NO329414B1 NO 329414 B1 NO329414 B1 NO 329414B1 NO 20044547 A NO20044547 A NO 20044547A NO 20044547 A NO20044547 A NO 20044547A NO 329414 B1 NO329414 B1 NO 329414B1
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- Prior art keywords
- pharmaceutical preparation
- core
- preparation according
- film
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- PPRRDFIXUUSXRA-UHFFFAOYSA-N flibanserin Chemical compound FC(F)(F)C1=CC=CC(N2CCN(CCN3C(NC4=CC=CC=C43)=O)CC2)=C1 PPRRDFIXUUSXRA-UHFFFAOYSA-N 0.000 title claims abstract description 38
- 229960002053 flibanserin Drugs 0.000 title claims abstract description 37
- GWEVSGVZZGPLCZ-UHFFFAOYSA-N Titan oxide Chemical compound O=[Ti]=O GWEVSGVZZGPLCZ-UHFFFAOYSA-N 0.000 title claims description 24
- 239000000454 talc Substances 0.000 title claims description 14
- 229910052623 talc Inorganic materials 0.000 title claims description 14
- 239000004408 titanium dioxide Substances 0.000 title claims description 12
- 239000008194 pharmaceutical composition Substances 0.000 title 1
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- UFVKGYZPFZQRLF-UHFFFAOYSA-N hydroxypropyl methyl cellulose Chemical compound OC1C(O)C(OC)OC(CO)C1OC1C(O)C(O)C(OC2C(C(O)C(OC3C(C(O)C(O)C(CO)O3)O)C(CO)O2)O)C(CO)O1 UFVKGYZPFZQRLF-UHFFFAOYSA-N 0.000 claims description 23
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Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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Landscapes
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- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Epidemiology (AREA)
- Psychiatry (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Pain & Pain Management (AREA)
- Hospice & Palliative Care (AREA)
- Anesthesiology (AREA)
- Gynecology & Obstetrics (AREA)
- Psychology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP02011224 | 2002-05-22 | ||
| PCT/EP2003/005226 WO2003097058A1 (en) | 2002-05-22 | 2003-05-19 | New pharmaceutical compositions containing flibanserin polymorph a |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| NO20044547L NO20044547L (no) | 2004-12-17 |
| NO329414B1 true NO329414B1 (no) | 2010-10-18 |
Family
ID=29433081
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20044547A NO329414B1 (no) | 2002-05-22 | 2004-10-22 | Farmasoytiske sammensetninger inneholdende flibanserin polymorf A, titandioksid og/eller talk |
Country Status (25)
| Country | Link |
|---|---|
| EP (1) | EP1511489B1 (zh) |
| JP (1) | JP3919788B2 (zh) |
| KR (1) | KR101054237B1 (zh) |
| CN (3) | CN102240289A (zh) |
| AT (1) | ATE499939T1 (zh) |
| BR (1) | BRPI0311189B8 (zh) |
| CA (1) | CA2483597C (zh) |
| CY (1) | CY1111470T1 (zh) |
| DE (1) | DE60336225D1 (zh) |
| DK (1) | DK1511489T3 (zh) |
| EA (1) | EA007185B1 (zh) |
| EC (1) | ECSP045493A (zh) |
| ES (1) | ES2361994T3 (zh) |
| HR (1) | HRP20041092B1 (zh) |
| IL (1) | IL164440A0 (zh) |
| ME (1) | MEP55308A (zh) |
| MX (1) | MXPA04011487A (zh) |
| NO (1) | NO329414B1 (zh) |
| NZ (1) | NZ537253A (zh) |
| PL (1) | PL211062B1 (zh) |
| RS (1) | RS51718B (zh) |
| SI (1) | SI1511489T1 (zh) |
| UA (1) | UA80135C2 (zh) |
| WO (1) | WO2003097058A1 (zh) |
| ZA (1) | ZA200408151B (zh) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US10675280B2 (en) | 2001-10-20 | 2020-06-09 | Sprout Pharmaceuticals, Inc. | Treating sexual desire disorders with flibanserin |
| UA78974C2 (en) | 2001-10-20 | 2007-05-10 | Boehringer Ingelheim Pharma | Use of flibanserin for treating disorders of sexual desire |
| US20050239798A1 (en) * | 2004-04-22 | 2005-10-27 | Boehringer Ingelheim Pharmaceuticals, Inc. | Method for the treatment of premenstrual and other female sexual disorders |
| WO2006096439A2 (en) * | 2005-03-04 | 2006-09-14 | Boehringer Ingelheim International Gmbh | Pharmaceutical compositions for the treatment and/or prevention of schizophrenia and related diseases |
| JP2008540672A (ja) * | 2005-05-19 | 2008-11-20 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | 病状に起因する性的機能不全の治療方法 |
| WO2006125042A1 (en) * | 2005-05-19 | 2006-11-23 | Boehringer Ingelheim International Gmbh | Method for the treatment of drug-induced sexual dysfunction |
| EP1912650B8 (en) | 2005-08-03 | 2017-10-18 | Sprout Pharmaceuticals, Inc. | Use of flibanserin in the treatment of obesity |
| CA2626134C (en) | 2005-10-29 | 2013-12-24 | Boehringer Ingelheim International Gmbh | Benzimidazolone derivatives for the treatment of premenstrual and other female sexual disorders |
| US20070105869A1 (en) * | 2005-11-08 | 2007-05-10 | Stephane Pollentier | Use of flibanserin for the treatment of pre-menopausal sexual desire disorders |
| EP2037927B1 (en) | 2006-06-30 | 2010-01-27 | Boehringer Ingelheim International GmbH | Flibanserin for the treatment of urinary incontinence and related diseases |
| CL2007002214A1 (es) | 2006-08-14 | 2008-03-07 | Boehringer Ingelheim Int | Composicion farmaceutica en la forma de comprimido, donde al menos la longitud del comprimido en el estado anterior de la aplicacion es al menos 7/12 del diametro pilorico del paciente y despues de ingerirlo en estado alimentado, la longitud del comp |
| AU2007286288A1 (en) | 2006-08-14 | 2008-02-21 | Boehringer Ingelheim International Gmbh | Formulations of flibanserin and method for manufacturing the same |
| EA200900270A1 (ru) | 2006-08-25 | 2009-08-28 | Бёрингер Ингельхайм Интернациональ Гмбх | Системы регулируемого высвобождения и способ их приготовления |
| ATE524446T1 (de) | 2006-12-20 | 2011-09-15 | Boehringer Ingelheim Int | Sulfatierte benzimidazolon-derivate mit gemischter serotonin-rezeptor-affinität |
| EP1955699A1 (en) * | 2007-02-08 | 2008-08-13 | Boehringer Ingelheim Pharma GmbH & Co. KG | Use of flibanserin for the treatment of insomnia |
| PE20091188A1 (es) | 2007-09-12 | 2009-08-31 | Boehringer Ingelheim Int | Compuesto 1-[2-(4-(3-trifluorometil-fenil)piperazin-1-il)etil]-2,3-dihidro-1h-benzimidazol-2-ona (flibanserina), sus sales de adicion y composiciones farmaceuticas que los contienen |
| EP2090297A1 (en) * | 2008-02-13 | 2009-08-19 | Boehringer Ingelheim International GmbH | Formulations of flibanserin |
| DE102008047910A1 (de) | 2008-09-19 | 2010-03-25 | Molkerei Meggle Wasserburg Gmbh & Co. Kg | Tablettierhilfsstoff auf Laktose- und Cellulosebasis |
| US20120010216A1 (en) * | 2010-07-06 | 2012-01-12 | Brown Arthur M | Pharmaceutical compositions containing vanoxerine |
| CN104926734B (zh) * | 2015-07-07 | 2017-04-05 | 苏州立新制药有限公司 | 氟班色林的制备方法 |
| WO2017128932A1 (zh) * | 2016-01-31 | 2017-08-03 | 孟晓明 | 氟班色林的新晶型及其制备方法及其用途 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1251144B (it) * | 1991-07-30 | 1995-05-04 | Boehringer Ingelheim Italia | Derivati del benzimidazolone |
| UA76767C2 (uk) * | 2001-08-02 | 2006-09-15 | Бідакем С.П.А. | Стабільна поліморфна модифікація флібансерину, спосіб її промислового одержання та її застосування для одержання лікарських засобів |
| DE10138273A1 (de) * | 2001-08-10 | 2003-02-27 | Boehringer Ingelheim Pharma | Arzneimittel mit neuroprotektiver Wirkung |
-
2003
- 2003-05-19 UA UA20041210555A patent/UA80135C2/uk unknown
- 2003-05-19 MX MXPA04011487A patent/MXPA04011487A/es active IP Right Grant
- 2003-05-19 EP EP03730069A patent/EP1511489B1/en not_active Expired - Lifetime
- 2003-05-19 WO PCT/EP2003/005226 patent/WO2003097058A1/en active Application Filing
- 2003-05-19 CN CN201110122058XA patent/CN102240289A/zh active Pending
- 2003-05-19 DE DE60336225T patent/DE60336225D1/de not_active Expired - Lifetime
- 2003-05-19 KR KR1020047018741A patent/KR101054237B1/ko active IP Right Grant
- 2003-05-19 RS YU98704A patent/RS51718B/en unknown
- 2003-05-19 ES ES03730069T patent/ES2361994T3/es not_active Expired - Lifetime
- 2003-05-19 NZ NZ537253A patent/NZ537253A/en not_active IP Right Cessation
- 2003-05-19 SI SI200331994T patent/SI1511489T1/sl unknown
- 2003-05-19 JP JP2004505057A patent/JP3919788B2/ja not_active Expired - Fee Related
- 2003-05-19 DK DK03730069.6T patent/DK1511489T3/da active
- 2003-05-19 CN CNA2007100014771A patent/CN101002780A/zh active Pending
- 2003-05-19 BR BRPI0311189A patent/BRPI0311189B8/pt not_active IP Right Cessation
- 2003-05-19 AT AT03730069T patent/ATE499939T1/de active
- 2003-05-19 ME MEP-553/08A patent/MEP55308A/xx unknown
- 2003-05-19 EA EA200401515A patent/EA007185B1/ru not_active IP Right Cessation
- 2003-05-19 CA CA2483597A patent/CA2483597C/en not_active Expired - Fee Related
- 2003-05-19 CN CNA038117029A patent/CN1655789A/zh active Pending
- 2003-05-19 PL PL372457A patent/PL211062B1/pl unknown
-
2004
- 2004-10-05 IL IL16444004A patent/IL164440A0/xx unknown
- 2004-10-08 ZA ZA200408151A patent/ZA200408151B/en unknown
- 2004-10-22 NO NO20044547A patent/NO329414B1/no not_active IP Right Cessation
- 2004-11-19 HR HRP20041092AA patent/HRP20041092B1/hr not_active IP Right Cessation
- 2004-12-13 EC EC2004005493A patent/ECSP045493A/es unknown
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2011
- 2011-05-17 CY CY20111100475T patent/CY1111470T1/el unknown
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| MM1K | Lapsed by not paying the annual fees |