NO328710B1 - (Pyrido/tieno)-[f]-oksazepin-5-on-derivater, farmasoytiske preparater omfattende slike samt anvendelse av slike for fremstilling av medikamenter for behandling av sykdom - Google Patents
(Pyrido/tieno)-[f]-oksazepin-5-on-derivater, farmasoytiske preparater omfattende slike samt anvendelse av slike for fremstilling av medikamenter for behandling av sykdom Download PDFInfo
- Publication number
- NO328710B1 NO328710B1 NO20035523A NO20035523A NO328710B1 NO 328710 B1 NO328710 B1 NO 328710B1 NO 20035523 A NO20035523 A NO 20035523A NO 20035523 A NO20035523 A NO 20035523A NO 328710 B1 NO328710 B1 NO 328710B1
- Authority
- NO
- Norway
- Prior art keywords
- alkyl
- pyrido
- formula
- oxazepin
- thieno
- Prior art date
Links
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- A—HUMAN NECESSITIES
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- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
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- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
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- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
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- Addiction (AREA)
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- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Gynecology & Obstetrics (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Dermatology (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
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| EP01202284 | 2001-06-14 | ||
| PCT/EP2002/006364 WO2002102808A2 (en) | 2001-06-14 | 2002-06-10 | (PYRIDO/THIENO)-[f]-OXAZEPIN-5-ONE DERIVATIVES AS POSITIVE MODULATORS OF THE AMPA RECEPTOR |
Publications (2)
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| NO20035523D0 NO20035523D0 (no) | 2003-12-11 |
| NO328710B1 true NO328710B1 (no) | 2010-05-03 |
Family
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| NO20035523A NO328710B1 (no) | 2001-06-14 | 2003-12-11 | (Pyrido/tieno)-[f]-oksazepin-5-on-derivater, farmasoytiske preparater omfattende slike samt anvendelse av slike for fremstilling av medikamenter for behandling av sykdom |
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| JP (1) | JP4435562B2 (zh) |
| KR (1) | KR100864267B1 (zh) |
| CN (2) | CN101029051B (zh) |
| AR (1) | AR034482A1 (zh) |
| AU (1) | AU2002320841B2 (zh) |
| BR (1) | BR0210307A (zh) |
| CA (1) | CA2449215C (zh) |
| CO (1) | CO5550448A2 (zh) |
| CZ (1) | CZ296217B6 (zh) |
| EC (1) | ECSP034890A (zh) |
| HR (1) | HRP20031013A2 (zh) |
| HU (1) | HUP0400196A3 (zh) |
| IL (2) | IL158928A0 (zh) |
| IS (1) | IS7042A (zh) |
| MX (1) | MXPA03011562A (zh) |
| NO (1) | NO328710B1 (zh) |
| NZ (1) | NZ529671A (zh) |
| PE (1) | PE20030271A1 (zh) |
| PL (1) | PL367185A1 (zh) |
| RU (1) | RU2286347C2 (zh) |
| SK (1) | SK287583B6 (zh) |
| WO (1) | WO2002102808A2 (zh) |
| ZA (1) | ZA200309096B (zh) |
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| TW200817385A (en) * | 2006-07-04 | 2008-04-16 | Organon Nv | Heterocyclic derivatives |
| FR2964969B1 (fr) * | 2010-09-16 | 2012-08-24 | Servier Lab | Nouveaux derives dihydrobenzoxathiazepines, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
Family Cites Families (11)
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| GB1238719A (zh) | 1968-11-01 | 1971-07-07 | ||
| CA2450801C (en) | 1992-07-24 | 2009-11-17 | The Regent Of The University Of California | Drugs that enhance synaptic responses mediated by ampa receptors |
| DE59607274D1 (de) | 1995-01-06 | 2001-08-16 | Hoffmann La Roche | Hydroxymethyl-imidazodiazepine und deren ester |
| US5650409A (en) * | 1995-06-02 | 1997-07-22 | Cortex Pharmaceuticals, Inc. | Benzoyl piperidines/pyrrolidines for enhancing synaptic response |
| US5736543A (en) | 1996-04-03 | 1998-04-07 | The Regents Of The University Of California | Benzoxazines for enhancing synaptic response |
| DE69831446T2 (de) * | 1997-06-09 | 2006-06-14 | Pfizer Prod Inc | Chinazolin-4-on AMPA Antagonisten |
| US5985871A (en) | 1997-12-24 | 1999-11-16 | Cortex Pharmaceuticals, Inc. | Benzoxazine compounds for enhancing synaptic response |
| EE200000468A (et) * | 1998-02-18 | 2002-04-15 | Neurosearch A/S | Ühendid, nende kasutamine ja farmatseutiline kompositsioon |
| US6124278A (en) | 1998-04-03 | 2000-09-26 | The Regents Of The University Of California | Acylbenzoxazines for enhancing synaptic response |
| DE60035591D1 (de) | 1999-05-12 | 2007-08-30 | Us Health | Thiazepin-hemmer von hiv-1 integrase |
| TWI232863B (en) | 2001-06-11 | 2005-05-21 | Akzo Nobel Nv | Benzoxazepine derivatives |
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2002
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- 2002-06-10 US US10/480,569 patent/US7345036B2/en not_active Expired - Fee Related
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- 2002-06-10 JP JP2003506280A patent/JP4435562B2/ja not_active Expired - Fee Related
- 2002-06-10 MX MXPA03011562A patent/MXPA03011562A/es active IP Right Grant
- 2002-06-10 CN CN2006100598858A patent/CN101029051B/zh not_active Expired - Fee Related
- 2002-06-10 CN CNB028118154A patent/CN1255413C/zh not_active Expired - Fee Related
- 2002-06-10 EP EP02754652A patent/EP1446407A2/en not_active Withdrawn
- 2002-06-10 PL PL02367185A patent/PL367185A1/xx unknown
- 2002-06-10 AU AU2002320841A patent/AU2002320841B2/en not_active Ceased
- 2002-06-10 BR BR0210307-9A patent/BR0210307A/pt not_active Application Discontinuation
- 2002-06-10 HU HU0400196A patent/HUP0400196A3/hu unknown
- 2002-06-10 SK SK1526-2003A patent/SK287583B6/sk not_active IP Right Cessation
- 2002-06-10 WO PCT/EP2002/006364 patent/WO2002102808A2/en active IP Right Grant
- 2002-06-10 CA CA2449215A patent/CA2449215C/en not_active Expired - Fee Related
- 2002-06-10 KR KR1020037016248A patent/KR100864267B1/ko not_active IP Right Cessation
- 2002-06-10 CZ CZ20033392A patent/CZ296217B6/cs not_active IP Right Cessation
- 2002-06-10 RU RU2004100702/04A patent/RU2286347C2/ru not_active IP Right Cessation
- 2002-06-13 AR ARP020102223A patent/AR034482A1/es unknown
- 2002-06-13 PE PE2002000511A patent/PE20030271A1/es not_active Application Discontinuation
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2003
- 2003-11-17 IS IS7042A patent/IS7042A/is unknown
- 2003-11-18 IL IL158928A patent/IL158928A/en not_active IP Right Cessation
- 2003-11-21 ZA ZA200309096A patent/ZA200309096B/en unknown
- 2003-12-08 HR HR20031013A patent/HRP20031013A2/hr not_active Application Discontinuation
- 2003-12-11 EC EC2003004890A patent/ECSP034890A/es unknown
- 2003-12-11 NO NO20035523A patent/NO328710B1/no not_active IP Right Cessation
- 2003-12-16 CO CO03109961A patent/CO5550448A2/es not_active Application Discontinuation
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2008
- 2008-02-01 US US12/024,597 patent/US7566778B2/en not_active Expired - Fee Related
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2009
- 2009-02-20 US US12/389,968 patent/US8034804B2/en not_active Expired - Fee Related
Also Published As
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| Publication | Publication Date | Title |
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| US7504390B2 (en) | Benzoxazepine derivatives and their use as AMPA receptor stimulators | |
| AU2002314144A1 (en) | Benzoxazepine derivatives and their use as AMPA receptor stimulators | |
| US7566778B2 (en) | (Pyrido/thieno)-[f]-oxazepine-5-one derivatives | |
| AU2002320841A1 (en) | (Pyrido/thieno)-[f]-oxazepin-5-one derivatives as positive modulators of the AMPA receptor |
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