NO328195B1 - Nye 1,2,4-tiadiazolderivater som melanokortinreseptormodulatorer - Google Patents
Nye 1,2,4-tiadiazolderivater som melanokortinreseptormodulatorer Download PDFInfo
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- NO328195B1 NO328195B1 NO20042372A NO20042372A NO328195B1 NO 328195 B1 NO328195 B1 NO 328195B1 NO 20042372 A NO20042372 A NO 20042372A NO 20042372 A NO20042372 A NO 20042372A NO 328195 B1 NO328195 B1 NO 328195B1
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US33792701P | 2001-11-08 | 2001-11-08 | |
PCT/US2002/035340 WO2003040117A1 (en) | 2001-11-08 | 2002-11-04 | Novel 1,2,4-thiadiazole derivatives as melanocortin receptor modulators |
Publications (2)
Publication Number | Publication Date |
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NO20042372L NO20042372L (no) | 2004-06-07 |
NO328195B1 true NO328195B1 (no) | 2010-01-04 |
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Application Number | Title | Priority Date | Filing Date |
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NO20042372A NO328195B1 (no) | 2001-11-08 | 2004-06-07 | Nye 1,2,4-tiadiazolderivater som melanokortinreseptormodulatorer |
Country Status (26)
Country | Link |
---|---|
US (2) | US7049331B2 (pt) |
EP (1) | EP1446394B1 (pt) |
JP (1) | JP4436676B2 (pt) |
CN (1) | CN1312139C (pt) |
AR (1) | AR037331A1 (pt) |
AT (1) | ATE344254T1 (pt) |
AU (1) | AU2009201842B2 (pt) |
BR (1) | BR0214024A (pt) |
CA (1) | CA2466140C (pt) |
CY (1) | CY1105907T1 (pt) |
DE (1) | DE60215848T2 (pt) |
DK (1) | DK1446394T3 (pt) |
ES (1) | ES2275918T3 (pt) |
IL (1) | IL161829A (pt) |
MX (1) | MXPA04004458A (pt) |
MY (1) | MY134993A (pt) |
NO (1) | NO328195B1 (pt) |
NZ (1) | NZ532883A (pt) |
PT (1) | PT1446394E (pt) |
RS (1) | RS51530B (pt) |
RU (1) | RU2317292C2 (pt) |
SG (1) | SG176310A1 (pt) |
SI (1) | SI1446394T1 (pt) |
TW (1) | TWI328586B (pt) |
WO (1) | WO2003040117A1 (pt) |
ZA (1) | ZA200404484B (pt) |
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JP2005504043A (ja) | 2001-08-10 | 2005-02-10 | パラチン テクノロジーズ インク. | 生物学的に活性な金属ペプチド類のペプチド模倣体類 |
US7732451B2 (en) | 2001-08-10 | 2010-06-08 | Palatin Technologies, Inc. | Naphthalene-containing melanocortin receptor-specific small molecule |
US7319107B2 (en) * | 2001-11-08 | 2008-01-15 | Johnson & Johnson Consumer Companies, Inc. | 1,2,4-thiadiazolium derivatives as melanocortin receptor modulators |
US7049331B2 (en) * | 2001-11-08 | 2006-05-23 | Ortho-Mcneil Pharmaceutical, Inc. | 1,2,4-thiadiazole derivatives as melanocortin receptor modulators |
US7968548B2 (en) * | 2003-05-01 | 2011-06-28 | Palatin Technologies, Inc. | Melanocortin receptor-specific piperazine compounds with diamine groups |
US7727990B2 (en) | 2003-05-01 | 2010-06-01 | Palatin Technologies, Inc. | Melanocortin receptor-specific piperazine and keto-piperazine compounds |
US7727991B2 (en) | 2003-05-01 | 2010-06-01 | Palatin Technologies, Inc. | Substituted melanocortin receptor-specific single acyl piperazine compounds |
WO2005054849A2 (en) * | 2003-12-06 | 2005-06-16 | Bayer Healthcare Ag | Diagnostics and therapeutics for diseases associated with g protein-coupled receptor mc5 (mc5r) |
EP1734963A4 (en) | 2004-04-02 | 2008-06-18 | Merck & Co Inc | METHOD FOR TREATING PEOPLE WITH METABOLIC AND ANTHROPOMETRIC DISORDER |
US7709484B1 (en) | 2004-04-19 | 2010-05-04 | Palatin Technologies, Inc. | Substituted melanocortin receptor-specific piperazine compounds |
CN1946703A (zh) | 2004-04-20 | 2007-04-11 | 特兰斯泰克制药公司 | 取代的噻唑和嘧啶衍生物作为黑素细胞皮质激素受体调节剂 |
US8394765B2 (en) | 2004-11-01 | 2013-03-12 | Amylin Pharmaceuticals Llc | Methods of treating obesity with two different anti-obesity agents |
ATE427759T1 (de) | 2004-11-01 | 2009-04-15 | Amylin Pharmaceuticals Inc | Behandlung von fettsucht und verbundenen erkrankungen |
US20070021433A1 (en) | 2005-06-03 | 2007-01-25 | Jian-Qiang Fan | Pharmacological chaperones for treating obesity |
BRPI0614649A2 (pt) | 2005-08-11 | 2011-04-12 | Amylin Pharmaceuticals Inc | polipeptìdeos hìbridos com propriedades selecionáveis |
EP2330124B1 (en) | 2005-08-11 | 2015-02-25 | Amylin Pharmaceuticals, LLC | Hybrid polypeptides with selectable properties |
US7834017B2 (en) | 2006-08-11 | 2010-11-16 | Palatin Technologies, Inc. | Diamine-containing, tetra-substituted piperazine compounds having identical 1- and 4-substituents |
US7704533B2 (en) * | 2006-12-13 | 2010-04-27 | J&J Consumer Companies, Inc. | Compositions and methods of inducing hair growth utilizing Continus coggygria |
JP5383498B2 (ja) * | 2006-12-14 | 2014-01-08 | ニューロノバ エービー | メラノコルチン4レセプターの活性を低下させる薬剤を使用した、神経系の疾患または損傷の処置 |
EP2278962B1 (en) | 2008-02-21 | 2014-02-12 | Janssen Pharmaceutica N.V. | Methods for the treatment of dermatological disorders |
US8377925B2 (en) | 2008-02-29 | 2013-02-19 | Mimetica Pty Ltd | Methods of modulating the activity of the MC5 receptor and treatment of conditions related to this receptor |
US8008291B2 (en) * | 2008-02-29 | 2011-08-30 | Mimetica Pty Ltd | 3-aminoalkyl-1,4-diazepan-2-one melanocortin-5 receptor antagonists |
US8343958B2 (en) | 2008-02-29 | 2013-01-01 | Mimetica Pty Ltd | 3-aminoalkyl-1,4-diazepan-2-one melanocortin-5-receptor antagonists |
US8563742B2 (en) | 2008-08-29 | 2013-10-22 | High Point Pharmaceuticals, Llc | Substituted aminothiazole derivatives, pharmaceutical compositions, and methods of use |
JP5514831B2 (ja) | 2008-11-17 | 2014-06-04 | メルク・シャープ・アンド・ドーム・コーポレーション | 糖尿病の治療のための置換二環式アミン |
US20100273838A1 (en) * | 2009-04-24 | 2010-10-28 | Chengji Cui | Stable topical compositions for 1,2,4-thiadiazole derivatives |
CA2768577A1 (en) | 2009-07-23 | 2011-01-27 | Schering Corporation | Benzo-fused oxazepine compounds as stearoyl-coenzyme a delta-9 desaturase inhibitors |
WO2011011506A1 (en) | 2009-07-23 | 2011-01-27 | Schering Corporation | Spirocyclic oxazepine compounds as stearoyl-coenzyme a delta-9 desaturase inhibitors |
ES2360783B1 (es) * | 2009-10-02 | 2012-07-04 | Consejo Superior De Investigaciones Científicas (Csic) | 1,2,4-tiadiazoles-5-imino sustituidos utiles en el tratamiento de enfermedades neurodegenerativas |
US8470880B2 (en) | 2009-12-15 | 2013-06-25 | Mcneil-Ppc, Inc. | Methods of reducing hair loss and/or facilitating hair growth and/or regrowth |
US8470833B2 (en) | 2009-12-15 | 2013-06-25 | Mcneil-Ppc, Inc. | Hair growth and/or regrowth compositions |
WO2011137024A1 (en) | 2010-04-26 | 2011-11-03 | Merck Sharp & Dohme Corp. | Novel spiropiperidine prolylcarboxypeptidase inhibitors |
EP2568812B1 (en) | 2010-05-11 | 2016-10-26 | Merck Sharp & Dohme Corp. | Novel prolylcarboxypeptidase inhibitors |
EP2579873A4 (en) | 2010-06-11 | 2013-11-27 | Merck Sharp & Dohme | NOVEL PROLYLCARBOXYPEPTIDASE HEMMER |
CA2825098C (en) | 2011-01-27 | 2020-03-10 | Universite De Montreal | Pyrazolopyridine and pyrazolopyrimidine derivatives as melanocortin-4 receptor modulators |
CN113679717A (zh) | 2012-08-22 | 2021-11-23 | 康奈尔大学 | 用于抑制肌成束蛋白的方法 |
US8962041B2 (en) | 2013-02-12 | 2015-02-24 | Johnson & Johnson Consumer Companies, Inc. | Methods and compositions for enhancing hair quality using blackberry extract |
EP3107902B1 (en) | 2014-02-20 | 2021-04-07 | Cornell University Cornell Center For Technology, Enterprise & Commercialization ("CCTEC") | Compounds and methods for inhibiting fascin |
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JPS6011481A (ja) | 1983-06-30 | 1985-01-21 | Nippon Soda Co Ltd | 1,2,4−チアジアゾ−ル系誘導体及び農園芸用殺菌剤 |
JPH02173165A (ja) | 1988-12-27 | 1990-07-04 | Nippon Soda Co Ltd | 防汚剤 |
AU3768799A (en) | 1998-04-28 | 1999-11-16 | Trega Biosciences, Inc. | Isoquinoline compound melanocortin receptor ligands and methods of using same |
WO1999055675A1 (de) | 1998-04-29 | 1999-11-04 | Axiva Gmbh | Verfahren zur katalytischen herstellung von substituierten bipyridylderivaten |
CA2334551A1 (en) | 1998-06-11 | 1999-12-16 | Merck & Co., Inc. | Spiropiperidine derivatives as melanocortin receptor agonists |
US6294534B1 (en) * | 1998-06-11 | 2001-09-25 | Merck & Co., Inc. | Spiropiperidine derivatives as melanocortin receptor agonists |
AU1324300A (en) | 1998-10-26 | 2000-05-15 | Vertex Pharmaceuticals Incorporated | Pentacyclic compounds useful as inhibitors of hepatitis c virus ns3 helicase |
WO2001055107A2 (en) | 2000-01-28 | 2001-08-02 | Melacure Therapeutics Ab | Aromatic amines and amides acting on the melanocortin receptors |
US7049331B2 (en) * | 2001-11-08 | 2006-05-23 | Ortho-Mcneil Pharmaceutical, Inc. | 1,2,4-thiadiazole derivatives as melanocortin receptor modulators |
US7319107B2 (en) * | 2001-11-08 | 2008-01-15 | Johnson & Johnson Consumer Companies, Inc. | 1,2,4-thiadiazolium derivatives as melanocortin receptor modulators |
-
2002
- 2002-11-04 US US10/287,095 patent/US7049331B2/en not_active Expired - Fee Related
- 2002-11-04 MX MXPA04004458A patent/MXPA04004458A/es active IP Right Grant
- 2002-11-04 BR BR0214024-1A patent/BR0214024A/pt active Search and Examination
- 2002-11-04 RU RU2004114214/04A patent/RU2317292C2/ru not_active IP Right Cessation
- 2002-11-04 ES ES02776448T patent/ES2275918T3/es not_active Expired - Lifetime
- 2002-11-04 DK DK02776448T patent/DK1446394T3/da active
- 2002-11-04 NZ NZ532883A patent/NZ532883A/en not_active IP Right Cessation
- 2002-11-04 EP EP02776448A patent/EP1446394B1/en not_active Expired - Lifetime
- 2002-11-04 SI SI200230459T patent/SI1446394T1/sl unknown
- 2002-11-04 SG SG2006034359A patent/SG176310A1/en unknown
- 2002-11-04 CA CA2466140A patent/CA2466140C/en not_active Expired - Fee Related
- 2002-11-04 JP JP2003542163A patent/JP4436676B2/ja not_active Expired - Fee Related
- 2002-11-04 CN CNB028268547A patent/CN1312139C/zh not_active Expired - Fee Related
- 2002-11-04 DE DE60215848T patent/DE60215848T2/de not_active Expired - Lifetime
- 2002-11-04 AT AT02776448T patent/ATE344254T1/de active
- 2002-11-04 RS YUP-397/04A patent/RS51530B/en unknown
- 2002-11-04 WO PCT/US2002/035340 patent/WO2003040117A1/en active IP Right Grant
- 2002-11-04 PT PT02776448T patent/PT1446394E/pt unknown
- 2002-11-07 AR ARP020104272A patent/AR037331A1/es not_active Application Discontinuation
- 2002-11-08 MY MYPI20024179A patent/MY134993A/en unknown
- 2002-11-08 TW TW091133320A patent/TWI328586B/zh not_active IP Right Cessation
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2004
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- 2004-06-07 NO NO20042372A patent/NO328195B1/no not_active IP Right Cessation
- 2004-06-07 ZA ZA2004/04484A patent/ZA200404484B/en unknown
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2006
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