NO315687B1 - Anvendelse av nebivolol for fremstilling av et anti-aterogent middel - Google Patents
Anvendelse av nebivolol for fremstilling av et anti-aterogent middel Download PDFInfo
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- NO315687B1 NO315687B1 NO19972980A NO972980A NO315687B1 NO 315687 B1 NO315687 B1 NO 315687B1 NO 19972980 A NO19972980 A NO 19972980A NO 972980 A NO972980 A NO 972980A NO 315687 B1 NO315687 B1 NO 315687B1
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- Prior art keywords
- nebivolol
- compound
- vascular
- formula
- acid
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
- A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline
- A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P39/00—General protective or antinoxious agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Epidemiology (AREA)
- Neurosurgery (AREA)
- Urology & Nephrology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Psychiatry (AREA)
- Toxicology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicinal Preparation (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP94203775 | 1994-12-28 | ||
| PCT/EP1995/005174 WO1996019987A1 (en) | 1994-12-28 | 1995-12-21 | Use of nebivolol as an anti-atherogenic |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO972980D0 NO972980D0 (no) | 1997-06-26 |
| NO972980L NO972980L (no) | 1997-06-26 |
| NO315687B1 true NO315687B1 (no) | 2003-10-13 |
Family
ID=8217503
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO19972980A NO315687B1 (no) | 1994-12-28 | 1997-06-26 | Anvendelse av nebivolol for fremstilling av et anti-aterogent middel |
Country Status (20)
| Country | Link |
|---|---|
| US (2) | US5874461A (hu) |
| EP (1) | EP0801564B1 (hu) |
| JP (1) | JPH10511655A (hu) |
| KR (1) | KR100264348B1 (hu) |
| CN (1) | CN1167418C (hu) |
| AT (1) | ATE214924T1 (hu) |
| AU (1) | AU700364B2 (hu) |
| CA (1) | CA2207333C (hu) |
| CZ (1) | CZ287513B6 (hu) |
| DE (1) | DE69526120T2 (hu) |
| DK (1) | DK0801564T3 (hu) |
| ES (1) | ES2176354T3 (hu) |
| FI (1) | FI118884B (hu) |
| HU (1) | HU226208B1 (hu) |
| NO (1) | NO315687B1 (hu) |
| NZ (1) | NZ298074A (hu) |
| PT (1) | PT801564E (hu) |
| SI (1) | SI0801564T1 (hu) |
| SK (1) | SK282144B6 (hu) |
| WO (1) | WO1996019987A1 (hu) |
Families Citing this family (33)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2207333C (en) * | 1994-12-28 | 2006-10-17 | Janssen Pharmaceutica, Naamloze Vennootschap | Use of nebivolol as an anti-atherogenic |
| DE19716120A1 (de) * | 1997-04-17 | 1998-10-22 | Europ Lab Molekularbiolog | Verwendung von cholesterinsenkenden Mitteln |
| US6541669B1 (en) | 1998-06-08 | 2003-04-01 | Theravance, Inc. | β2-adrenergic receptor agonists |
| US6713651B1 (en) | 1999-06-07 | 2004-03-30 | Theravance, Inc. | β2-adrenergic receptor agonists |
| JP2000207219A (ja) * | 1999-01-18 | 2000-07-28 | Fujitsu Ten Ltd | 車載端末とセンタ―との間の通信システム、及び、通信システムに使用する車載端末 |
| US6683115B2 (en) | 1999-06-02 | 2004-01-27 | Theravance, Inc. | β2-adrenergic receptor agonists |
| US6593497B1 (en) | 1999-06-02 | 2003-07-15 | Theravance, Inc. | β2-adrenergic receptor agonists |
| UA73965C2 (en) | 1999-12-08 | 2005-10-17 | Theravance Inc | b2 ADRENERGIC RECEPTOR ANTAGONISTS |
| WO2002087508A2 (en) * | 2001-05-02 | 2002-11-07 | Nitromed, Inc. | Nitrosated and nitrosylated nebivolol and its metabolites, compositions and methods of use |
| EP1558922B1 (en) * | 2002-10-30 | 2013-02-27 | Ampere Life Sciences, Inc. | Identifying therapeutic compounds based on their physical-chemical properties |
| ITTO20030140U1 (it) * | 2003-09-16 | 2005-03-17 | Interfila Srl | Matita cosmetica |
| CA2583087C (en) | 2003-09-19 | 2012-07-10 | Galileo Pharmaceuticals, Inc. | Chroman derivatives |
| US7838552B2 (en) | 2004-06-04 | 2010-11-23 | Forest Laboratories Holdings Limited | Compositions comprising nebivolol |
| US7803838B2 (en) | 2004-06-04 | 2010-09-28 | Forest Laboratories Holdings Limited | Compositions comprising nebivolol |
| ATE512961T1 (de) | 2004-07-30 | 2011-07-15 | Torrent Pharmaceuticals Ltd | Amorphes nebivolol hydrochlorid und seine herstellung |
| SG175477A1 (en) * | 2005-01-31 | 2011-11-28 | Mylan Lab Inc | Hydroxylated nebivolol metabolites |
| DK2564843T3 (en) | 2005-06-01 | 2019-03-11 | Bioelectron Tech Corp | Redox-active therapeutics for the treatment of mitochondrial diseases and other conditions as well as modulation of energy biomarkers |
| JP5374162B2 (ja) | 2006-02-22 | 2013-12-25 | エジソン ファーマシューティカルズ， インコーポレイテッド | ミトコンドリア病および他の症状の処置のためのレドックス活性化治療の側鎖変異体およびエネルギーバイオマーカーの調節 |
| PL3456707T3 (pl) | 2007-11-06 | 2020-09-21 | Ptc Therapeutics, Inc. | Pochodne 4-(p-chinonylo)-2-hydroksybutanamidu do leczenia chorób mitochondrialnych |
| WO2009091777A1 (en) * | 2008-01-15 | 2009-07-23 | Forest Laboratories Holdings Limited | Nebivolol in the treatment of sexual dysfunction |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA1337432C (en) * | 1988-03-23 | 1995-10-24 | Raymond M. Xhonneux | Method of lowering the blood pressure |
| TW355683B (en) * | 1994-02-17 | 1999-04-11 | Janssen Pharmaceutica Nv | Composition containing micronized nebivolol |
| CA2207333C (en) * | 1994-12-28 | 2006-10-17 | Janssen Pharmaceutica, Naamloze Vennootschap | Use of nebivolol as an anti-atherogenic |
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1995
- 1995-12-21 CA CA002207333A patent/CA2207333C/en not_active Expired - Fee Related
- 1995-12-21 SI SI9530591T patent/SI0801564T1/xx unknown
- 1995-12-21 PT PT95942209T patent/PT801564E/pt unknown
- 1995-12-21 DK DK95942209T patent/DK0801564T3/da active
- 1995-12-21 HU HU9800675A patent/HU226208B1/hu unknown
- 1995-12-21 KR KR1019970703648A patent/KR100264348B1/ko not_active IP Right Cessation
- 1995-12-21 AU AU43477/96A patent/AU700364B2/en not_active Expired
- 1995-12-21 SK SK856-97A patent/SK282144B6/sk not_active IP Right Cessation
- 1995-12-21 DE DE69526120T patent/DE69526120T2/de not_active Expired - Lifetime
- 1995-12-21 US US08/860,238 patent/US5874461A/en not_active Expired - Lifetime
- 1995-12-21 CZ CZ19971919A patent/CZ287513B6/cs not_active IP Right Cessation
- 1995-12-21 ES ES95942209T patent/ES2176354T3/es not_active Expired - Lifetime
- 1995-12-21 EP EP95942209A patent/EP0801564B1/en not_active Expired - Lifetime
- 1995-12-21 JP JP8520223A patent/JPH10511655A/ja active Pending
- 1995-12-21 NZ NZ298074A patent/NZ298074A/xx not_active IP Right Cessation
- 1995-12-21 CN CNB951971492A patent/CN1167418C/zh not_active Expired - Lifetime
- 1995-12-21 WO PCT/EP1995/005174 patent/WO1996019987A1/en active IP Right Grant
- 1995-12-21 AT AT95942209T patent/ATE214924T1/de active
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1997
- 1997-06-26 NO NO19972980A patent/NO315687B1/no not_active IP Right Cessation
- 1997-06-27 FI FI972793A patent/FI118884B/fi not_active IP Right Cessation
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1998
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Also Published As
| Publication number | Publication date |
|---|---|
| WO1996019987A1 (en) | 1996-07-04 |
| KR100264348B1 (ko) | 2000-08-16 |
| PT801564E (pt) | 2002-09-30 |
| CZ191997A3 (cs) | 1999-01-13 |
| FI118884B (fi) | 2008-04-30 |
| CN1167418C (zh) | 2004-09-22 |
| DE69526120T2 (de) | 2002-11-28 |
| SI0801564T1 (en) | 2002-08-31 |
| AU4347796A (en) | 1996-07-19 |
| CN1171739A (zh) | 1998-01-28 |
| US5874461A (en) | 1999-02-23 |
| MX9704669A (es) | 1997-09-30 |
| JPH10511655A (ja) | 1998-11-10 |
| EP0801564B1 (en) | 2002-03-27 |
| NO972980D0 (no) | 1997-06-26 |
| AU700364B2 (en) | 1999-01-07 |
| SK85697A3 (en) | 2000-04-10 |
| CZ287513B6 (en) | 2000-12-13 |
| NZ298074A (en) | 2001-01-26 |
| NO972980L (no) | 1997-06-26 |
| ATE214924T1 (de) | 2002-04-15 |
| CA2207333C (en) | 2006-10-17 |
| FI972793A (fi) | 1997-06-27 |
| DK0801564T3 (da) | 2002-07-15 |
| FI972793A0 (fi) | 1997-06-27 |
| HUT77927A (hu) | 1998-11-30 |
| DE69526120D1 (de) | 2002-05-02 |
| HU226208B1 (en) | 2008-06-30 |
| US6075046A (en) | 2000-06-13 |
| SK282144B6 (sk) | 2001-11-06 |
| EP0801564A1 (en) | 1997-10-22 |
| ES2176354T3 (es) | 2002-12-01 |
| CA2207333A1 (en) | 1996-07-04 |
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| MK1K | Patent expired |