NO20091846L - Makrocykliske peptider som hepatitt C virus- inhibitorer - Google Patents

Makrocykliske peptider som hepatitt C virus- inhibitorer

Info

Publication number
NO20091846L
NO20091846L NO20091846A NO20091846A NO20091846L NO 20091846 L NO20091846 L NO 20091846L NO 20091846 A NO20091846 A NO 20091846A NO 20091846 A NO20091846 A NO 20091846A NO 20091846 L NO20091846 L NO 20091846L
Authority
NO
Norway
Prior art keywords
hepatitis
macrocyclic peptides
virus inhibitors
compounds
disclosed
Prior art date
Application number
NO20091846A
Other languages
English (en)
Norwegian (no)
Inventor
Nicholas A Meanwell
Paul Michael Scola
Stanley D'andrea
Barbara Zhizhen Zheng
Alan Xiangdong Wang
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20091846L publication Critical patent/NO20091846L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0815—Tripeptides with the first amino acid being basic

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO20091846A 2006-11-16 2009-05-12 Makrocykliske peptider som hepatitt C virus- inhibitorer NO20091846L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US86612006P 2006-11-16 2006-11-16
US11/939,753 US8003604B2 (en) 2006-11-16 2007-11-14 Hepatitis C virus inhibitors
PCT/US2007/084777 WO2008064057A1 (en) 2006-11-16 2007-11-15 Macrocyclic peptides as hepatitis c virus inhibitors

Publications (1)

Publication Number Publication Date
NO20091846L true NO20091846L (no) 2009-06-08

Family

ID=39251294

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20091846A NO20091846L (no) 2006-11-16 2009-05-12 Makrocykliske peptider som hepatitt C virus- inhibitorer

Country Status (7)

Country Link
US (1) US8003604B2 (en:Method)
EP (1) EP2089020B1 (en:Method)
JP (1) JP5241728B2 (en:Method)
AT (1) ATE492559T1 (en:Method)
DE (1) DE602007011493D1 (en:Method)
NO (1) NO20091846L (en:Method)
WO (1) WO2008064057A1 (en:Method)

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JP6342922B2 (ja) 2013-03-07 2018-06-13 ブリストル−マイヤーズ スクイブ カンパニーＢｒｉｓｔｏｌ−Ｍｙｅｒｓ Ｓｑｕｉｂｂ Ｃｏｍｐａｎｙ Ｃ型肝炎ウイルス阻害剤
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RU2016145449A (ru) 2014-06-12 2018-07-17 Аллосайт Фармасьютикалз Аг Низкомолекулярные ингибиторы функционального антигена лейкоцитов- lfa-1

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Also Published As

Publication number Publication date
US20080159982A1 (en) 2008-07-03
EP2089020A1 (en) 2009-08-19
ATE492559T1 (de) 2011-01-15
JP2010510967A (ja) 2010-04-08
JP5241728B2 (ja) 2013-07-17
US8003604B2 (en) 2011-08-23
EP2089020B1 (en) 2010-12-22
WO2008064057A1 (en) 2008-05-29
DE602007011493D1 (de) 2011-02-03

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