NO20090139L - Substituted phenyl acetic acids as DP-2 antagonists - Google Patents

Substituted phenyl acetic acids as DP-2 antagonists

Info

Publication number
NO20090139L
NO20090139L NO20090139A NO20090139A NO20090139L NO 20090139 L NO20090139 L NO 20090139L NO 20090139 A NO20090139 A NO 20090139A NO 20090139 A NO20090139 A NO 20090139A NO 20090139 L NO20090139 L NO 20090139L
Authority
NO
Norway
Prior art keywords
antagonists
substituted phenyl
acetic acids
phenyl acetic
conditions
Prior art date
Application number
NO20090139A
Other languages
English (en)
Norwegian (no)
Inventor
Eugene Thorsett
Fuqiang Ruan
Joshua Odingo
Andrew Lover
Kerry Fowler
Francine Farouz
Thomas Dudler
Amy Oliver
Mark Reed
Danwen Huang
Jin Bohan
Musong Kim
Nataly Hawthorn
Original Assignee
Icos Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Icos Corp filed Critical Icos Corp
Publication of NO20090139L publication Critical patent/NO20090139L/no

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    • C07D267/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D267/02—Seven-membered rings
    • C07D267/08—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D267/12—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D267/14—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
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    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
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    • C07D217/06—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines with the ring nitrogen atom acylated by carboxylic or carbonic acids, or with sulfur or nitrogen analogues thereof, e.g. carbamates
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    • C07D217/08—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines with a hetero atom directly attached to the ring nitrogen atom
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    • C07D223/02—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
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  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
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  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
  • Neurosurgery (AREA)
  • Hematology (AREA)
  • Biomedical Technology (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Pulmonology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
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  • Ophthalmology & Optometry (AREA)
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  • AIDS & HIV (AREA)
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NO20090139A 2006-06-09 2009-01-09 Substituted phenyl acetic acids as DP-2 antagonists NO20090139L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US81239906P 2006-06-09 2006-06-09
PCT/US2007/070805 WO2007146838A2 (fr) 2006-06-09 2007-06-08 Acides phénylacétiques substitués utilisés en tant qu'antagonistes de dp-2

Publications (1)

Publication Number Publication Date
NO20090139L true NO20090139L (no) 2009-03-05

Family

ID=38819983

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20090139A NO20090139L (no) 2006-06-09 2009-01-09 Substituted phenyl acetic acids as DP-2 antagonists

Country Status (10)

Country Link
EP (1) EP2044017A2 (fr)
JP (1) JP2009539881A (fr)
CN (1) CN101490001A (fr)
AU (1) AU2007257841A1 (fr)
BR (1) BRPI0712332A2 (fr)
CA (1) CA2654927A1 (fr)
EA (2) EA200802417A1 (fr)
MX (1) MX2008015638A (fr)
NO (1) NO20090139L (fr)
WO (1) WO2007146838A2 (fr)

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MX2010004309A (es) 2007-10-19 2010-05-03 Janssen Pharmaceutica Nv Moduladores de piperidinil y piperazinil de gamma-secretasa.
KR101618068B1 (ko) 2007-10-19 2016-05-04 얀센 파마슈티카 엔.브이. γ-세크레타아제의 탄소 결합된 조절제
MX2010004318A (es) 2007-10-19 2010-04-30 Janssen Pharmaceutica Nv Moduladores de la gamma-secretasa con enlaces de amina.
WO2011014588A2 (fr) * 2009-07-31 2011-02-03 Amira Pharmaceuticals, Inc. Préparations dermiques d'antagonistes du récepteur dp2
JP2013516475A (ja) * 2010-01-06 2013-05-13 アミラ ファーマシューティカルズ，インク． Ｄｐ２アンタゴニストおよびその使用
KR101920090B1 (ko) 2010-07-05 2018-11-19 이도르시아 파마슈티컬스 리미티드 1-페닐-치환된 헤테로시클릴 유도체 및 프로스타글란딘 ｄ２ 수용체 조절자로서 이의 용도
EP2457900A1 (fr) 2010-11-25 2012-05-30 Almirall, S.A. Nouveaux dérivés de pyrazole présentant un comportement antagoniste CRTH2
EP2487159A1 (fr) * 2011-02-11 2012-08-15 MSD Oss B.V. Inhibiteurs du RORgammaT
EP2688890B1 (fr) 2011-03-22 2017-08-30 Advinus Therapeutics Limited Composés tricycliques substitués; compositions et applications médicinales correspondantes
EP3409278B8 (fr) 2011-07-21 2020-11-04 Sumitomo Dainippon Pharma Oncology, Inc. Inhibiteurs de protéine kinase hétérocycliques
EP2573085A1 (fr) 2011-09-26 2013-03-27 AiCuris GmbH & Co. KG Monohydrate de mesylate acétamide N-[5-(aminosulfonyl)-4méthyl-1,3-thiazol-2-yl]-N-méthyl-2-[4-(2-pyridinyl)phényl] disposant d'une gamme de distribution de taille de particules spécifiques et portée de surface spécifique
EP2573086A1 (fr) * 2011-09-26 2013-03-27 AiCuris GmbH & Co. KG Monohydrate de mesylate acétamide N-[5-(Aminosulfonyl)-4-méthyl-1,3-thiazol-2-yl]-N-méthyl-2-[4-(2-pyridinyl)phényl]
JP6099149B2 (ja) * 2011-10-25 2017-03-22 塩野義製薬株式会社 Ｈｉｖ複製阻害剤
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WO2007146838A2 (fr) 2007-12-21
EA200802417A1 (ru) 2009-06-30
JP2009539881A (ja) 2009-11-19
WO2007146838A3 (fr) 2008-03-13
BRPI0712332A2 (pt) 2012-12-18
CA2654927A1 (fr) 2007-12-21
AU2007257841A1 (en) 2007-12-21
EA201200423A1 (ru) 2012-08-30

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