NO20081581L - Polymorfer av benzoatsalt av 2-[[6-[(3R)-3-amino-l-piperldinyl]-3,4-dihydro-3-metyl-2,4-diokso- 1(2H)-pyrlmidinylJmetyl)benzonitril, og fremgangsmater for anvendelse derav - Google Patents

Polymorfer av benzoatsalt av 2-[[6-[(3R)-3-amino-l-piperldinyl]-3,4-dihydro-3-metyl-2,4-diokso- 1(2H)-pyrlmidinylJmetyl)benzonitril, og fremgangsmater for anvendelse derav

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Publication number
NO20081581L
NO20081581L NO20081581A NO20081581A NO20081581L NO 20081581 L NO20081581 L NO 20081581L NO 20081581 A NO20081581 A NO 20081581A NO 20081581 A NO20081581 A NO 20081581A NO 20081581 L NO20081581 L NO 20081581L
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NO
Norway
Prior art keywords
methyl
polymorphs
methods
benzonitrile
dioxo
Prior art date
Application number
NO20081581A
Other languages
English (en)
Inventor
Mark Andres
Keith Lorimer
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Takeda Pharmaceutical
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
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Publication of NO20081581L publication Critical patent/NO20081581L/no

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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/513—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim having oxo groups directly attached to the heterocyclic ring, e.g. cytosine
    • A—HUMAN NECESSITIES
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    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

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Abstract

Det beskrives preparater omfattende Forbindelse I, der Forbindelse I er til stede i en eller flere polymorfe former.Det beskrives videre sett og produksjonsgjenstander med preparater omfattende en eller flere polymorfer av Forbindelse I samt metoder for å anvende preparatene for behandling av forskjellige sykdommer.
NO20081581A 2005-09-16 2008-03-31 Polymorfer av benzoatsalt av 2-[[6-[(3R)-3-amino-l-piperldinyl]-3,4-dihydro-3-metyl-2,4-diokso- 1(2H)-pyrlmidinylJmetyl)benzonitril, og fremgangsmater for anvendelse derav NO20081581L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US71813305P 2005-09-16 2005-09-16
PCT/US2006/035701 WO2007035372A2 (en) 2005-09-16 2006-09-13 Polymorphs of benzoate salt of 2-[[6-[(3r)-3-amino-1-piperidinyl]-3,4-dihydro-3-methyl-2,4-dioxo-1(2h)-pyrimidinyl]methyl]-benzonitrile and methods of use therefor

Publications (1)

Publication Number Publication Date
NO20081581L true NO20081581L (no) 2008-05-23

Family

ID=37758695

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20081581A NO20081581L (no) 2005-09-16 2008-03-31 Polymorfer av benzoatsalt av 2-[[6-[(3R)-3-amino-l-piperldinyl]-3,4-dihydro-3-metyl-2,4-diokso- 1(2H)-pyrlmidinylJmetyl)benzonitril, og fremgangsmater for anvendelse derav

Country Status (21)

Country Link
US (1) US20070066635A1 (no)
EP (1) EP1934198B1 (no)
JP (1) JP5124464B2 (no)
KR (1) KR20080056183A (no)
CN (1) CN101360735A (no)
AR (1) AR056518A1 (no)
AT (1) ATE518851T1 (no)
AU (1) AU2006292637A1 (no)
BR (1) BRPI0616215A2 (no)
CA (1) CA2622698A1 (no)
CR (1) CR9881A (no)
EA (1) EA015359B1 (no)
GE (1) GEP20115171B (no)
IL (1) IL190170A0 (no)
MA (1) MA29800B1 (no)
NO (1) NO20081581L (no)
NZ (1) NZ566798A (no)
PE (1) PE20070766A1 (no)
TW (1) TW200745079A (no)
WO (1) WO2007035372A2 (no)
ZA (1) ZA200802856B (no)

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AR056518A1 (es) 2007-10-10
EP1934198A2 (en) 2008-06-25
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MA29800B1 (fr) 2008-09-01
EA015359B1 (ru) 2011-06-30
ATE518851T1 (de) 2011-08-15
IL190170A0 (en) 2008-08-07
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TW200745079A (en) 2007-12-16
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US20070066635A1 (en) 2007-03-22
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