NO20081551L - Heterocyklisk substituerte pyridinderivater og antisoppmidler inneholdende samme - Google Patents
Heterocyklisk substituerte pyridinderivater og antisoppmidler inneholdende sammeInfo
- Publication number
- NO20081551L NO20081551L NO20081551A NO20081551A NO20081551L NO 20081551 L NO20081551 L NO 20081551L NO 20081551 A NO20081551 A NO 20081551A NO 20081551 A NO20081551 A NO 20081551A NO 20081551 L NO20081551 L NO 20081551L
- Authority
- NO
- Norway
- Prior art keywords
- atom
- group
- same
- antifungal agents
- pyridine derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- Epidemiology (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Det er et formål med foreliggende oppfinnelse å tilveiebringe et fungicid som har utmerkede fungicide effekter og er overlegent når det gjelder dets fysiske egenskaper, sikkerhet og metabolsk stabilitet. Ifølge foreliggende oppfinnelse er det beskrevet en forbindelse representert ved følgende formel (I), eller et salt derav: hvor Rrepresenterer et hydrogenatom, et halogenatom, en aminogruppe, en C_-alkylgruppe, en C_-alkoksygruppe eller en C_-alkoksy-C_-alkylgruppe; Rrepresenterer et hydrogenatom, en C.-alkylgruppe, en aminogruppe eller en di-C_-alkylaminogruppe; én av X og Y er et nitrogenatom mens den andre er et nitrogenatom eller et oksygenatom; ring A representerer en 5- eller 6-leddet heteroarylring eller en benzenring som kan ha et halogenatom eller 1 eller 2 C_-alkylgrupper; Z representerer en enkeltbinding, en metylengruppe, en etylengruppe, et oksygenatom, et svovelatom, - CH0-, -OCH-, -NH-, -CHNH-, -NHCH-, -CHS- eller -SCH-; Rrepresenterer et hydrogenatom, et halogenatom, en C.-alkylgruppe, en C.-cykloalkylgruppe, en C_-arylgruppe, en 5- eller 6-leddet heteroarylgruppe eller en 5- eller 6-leddet, ikke-aromatisk heterocyklisk gruppe som kan ha 1 eller 2 substituenter; og Rrepresenterer et hydrogenatom eller et halogenatom.
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US73126705P | 2005-10-31 | 2005-10-31 | |
JP2005317680 | 2005-10-31 | ||
US75339105P | 2005-12-27 | 2005-12-27 | |
JP2005374395 | 2005-12-27 | ||
PCT/JP2006/321678 WO2007052615A1 (ja) | 2005-10-31 | 2006-10-30 | ヘテロ環置換ピリジン誘導体およびそれらを含有する抗真菌剤 |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20081551L true NO20081551L (no) | 2008-05-21 |
Family
ID=38005768
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20081551A NO20081551L (no) | 2005-10-31 | 2008-03-31 | Heterocyklisk substituerte pyridinderivater og antisoppmidler inneholdende samme |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP1944303B1 (no) |
KR (1) | KR101003569B1 (no) |
AU (1) | AU2006309762B2 (no) |
CA (1) | CA2626767C (no) |
IL (1) | IL190609A (no) |
NO (1) | NO20081551L (no) |
NZ (1) | NZ567191A (no) |
WO (1) | WO2007052615A1 (no) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7932272B2 (en) | 2003-09-30 | 2011-04-26 | Eisai R&D Management Co., Ltd. | Antifungal agent containing heterocyclic compound |
WO2006106711A1 (ja) | 2005-03-30 | 2006-10-12 | Eisai R & D Management Co., Ltd. | ピリジン誘導体を含有する抗真菌剤 |
TWI385169B (zh) | 2005-10-31 | 2013-02-11 | Eisai R&D Man Co Ltd | 經雜環取代之吡啶衍生物及含有彼之抗真菌劑 |
EP2065377B1 (en) | 2006-09-21 | 2011-11-23 | Eisai R&D Management Co., Ltd. | Pyridine derivative substituted by heteroaryl ring, and antifungal agent comprising the same |
CA2685194A1 (en) | 2007-04-27 | 2008-11-13 | Eisai R&D Management Co., Ltd. | Heterocycle-substituted pyridine derivatives salt or crystal thereof |
TW200841879A (en) | 2007-04-27 | 2008-11-01 | Eisai R&D Man Co Ltd | Pyridine derivatives substituted by heterocyclic ring and phosphonoamino group, and anti-fungal agent containing same |
JPWO2009081970A1 (ja) * | 2007-12-26 | 2011-05-06 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | ヘテロ環置換ピリジン誘導体の製造方法 |
US8513287B2 (en) | 2007-12-27 | 2013-08-20 | Eisai R&D Management Co., Ltd. | Heterocyclic ring and phosphonoxymethyl group substituted pyridine derivatives and antifungal agent containing same |
WO2010032874A1 (ja) | 2008-09-19 | 2010-03-25 | 住友化学株式会社 | 農業用組成物 |
US8188119B2 (en) * | 2008-10-24 | 2012-05-29 | Eisai R&D Management Co., Ltd | Pyridine derivatives substituted with heterocyclic ring and γ-glutamylamino group, and antifungal agents containing same |
WO2011051198A2 (de) | 2009-10-30 | 2011-05-05 | Bayer Cropscience Ag | Pyridin-derivate als pflanzenschutzmittel |
JPWO2012060448A1 (ja) | 2010-11-05 | 2014-05-12 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | 抗真菌剤としての併用医薬組成物 |
WO2013031694A1 (ja) * | 2011-08-26 | 2013-03-07 | 富山化学工業株式会社 | アミン化合物またはその塩 |
AU2018379077B2 (en) | 2017-12-07 | 2023-04-27 | Basilea Pharmaceutica International Ag, Allschwil | Heterocycle substituted pyridine derivative antifungal agents |
AU2019294474A1 (en) * | 2018-06-25 | 2021-02-11 | Basilea Pharmaceutica International Ag, Allschwil | Pyridine derivatives substituted by heterocyclic ring and amino group |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5973575A (ja) * | 1982-10-05 | 1984-04-25 | Shionogi & Co Ltd | プロピニルアミノイソオキサゾ−ル誘導体 |
AU6947201A (en) | 2000-07-07 | 2002-01-21 | Eisai Co Ltd | Fungal cell wall synthesis gene |
HUP0400823A3 (en) * | 2001-04-05 | 2010-06-28 | Torrent Pharmaceuticals Ltd | Heterocyclic compounds for treating aging-related and diabetic vascular complications, their preparation and pharmaceutical compositions containing them |
DE10149370A1 (de) | 2001-10-06 | 2003-04-10 | Merck Patent Gmbh | Pyrazolderivate |
KR100437972B1 (ko) * | 2001-10-27 | 2004-07-02 | 한국과학기술연구원 | 피롤리디논 유도체, 이의 제조 방법 및 이를 포함하는제약 조성물 |
WO2004033432A1 (ja) * | 2002-10-09 | 2004-04-22 | Ssp Co., Ltd. | 抗真菌活性を有する新規ピラゾール化合物 |
DE10315572A1 (de) | 2003-04-05 | 2004-10-14 | Merck Patent Gmbh | Substituierte Pyrazole |
US7932272B2 (en) | 2003-09-30 | 2011-04-26 | Eisai R&D Management Co., Ltd. | Antifungal agent containing heterocyclic compound |
-
2006
- 2006-10-30 CA CA2626767A patent/CA2626767C/en active Active
- 2006-10-30 EP EP06812187.0A patent/EP1944303B1/en active Active
- 2006-10-30 AU AU2006309762A patent/AU2006309762B2/en active Active
- 2006-10-30 NZ NZ567191A patent/NZ567191A/en not_active IP Right Cessation
- 2006-10-30 WO PCT/JP2006/321678 patent/WO2007052615A1/ja active Application Filing
- 2006-10-30 KR KR1020087010403A patent/KR101003569B1/ko active IP Right Grant
-
2008
- 2008-03-31 NO NO20081551A patent/NO20081551L/no unknown
- 2008-04-03 IL IL190609A patent/IL190609A/en active IP Right Grant
Also Published As
Publication number | Publication date |
---|---|
AU2006309762A1 (en) | 2007-05-10 |
AU2006309762B2 (en) | 2010-02-25 |
EP1944303A1 (en) | 2008-07-16 |
EP1944303B1 (en) | 2013-08-21 |
IL190609A (en) | 2012-06-28 |
NZ567191A (en) | 2010-06-25 |
CA2626767C (en) | 2012-01-17 |
CA2626767A1 (en) | 2007-05-10 |
WO2007052615A1 (ja) | 2007-05-10 |
KR101003569B1 (ko) | 2010-12-22 |
KR20080066740A (ko) | 2008-07-16 |
EP1944303A4 (en) | 2010-11-03 |
IL190609A0 (en) | 2008-11-03 |
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