NO20070870L - Oksazolidinonforbindelser og sammensetninger og fremgangsmater relatert dertil - Google Patents

Oksazolidinonforbindelser og sammensetninger og fremgangsmater relatert dertil

Info

Publication number
NO20070870L
NO20070870L NO20070870A NO20070870A NO20070870L NO 20070870 L NO20070870 L NO 20070870L NO 20070870 A NO20070870 A NO 20070870A NO 20070870 A NO20070870 A NO 20070870A NO 20070870 L NO20070870 L NO 20070870L
Authority
NO
Norway
Prior art keywords
compositions
oxazolidinone compounds
compounds
formula
methods related
Prior art date
Application number
NO20070870A
Other languages
English (en)
Inventor
Albert Palomer
Antonio Guglietta
Montserrat Cano
Original Assignee
Ferrer Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ferrer Int filed Critical Ferrer Int
Publication of NO20070870L publication Critical patent/NO20070870L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/541—Non-condensed thiazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Oppfinnelsen tilveiebringer nye oksazolidinoner med formel (I), der Ri, R2, R3 og R4 er uavhengig valgt fra hydrogen, F og Cl; A er valgt fra visse eventuelt substituerte heterocykler; X er valgt fra O, S, NR'er og CR8Rg; Y er valgt fra O, S, SO, SO2, NO, NRi 1 og CRi iR]2; og n er valgt fra 0 til 1. Oppfinnelsen tilveiebringer også forskjellige prosesser for fremstillingen av slike forbindelser. Oksazolidinonforbindelser med formel (I) er aktive mot gram-positive og noen gram-negative humane og veterinære patogener med en svak monoaminoksidase (MAO) inhibitoraktivitet. De er anvendelige for behandling av bakterielle infeksjoner.
NO20070870A 2004-07-29 2007-02-15 Oksazolidinonforbindelser og sammensetninger og fremgangsmater relatert dertil NO20070870L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP04103657 2004-07-29
PCT/EP2005/053627 WO2006010756A1 (en) 2004-07-29 2005-07-26 Oxazolidinone compounds and compositions and methods related thereto

Publications (1)

Publication Number Publication Date
NO20070870L true NO20070870L (no) 2007-04-16

Family

ID=35355681

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20070870A NO20070870L (no) 2004-07-29 2007-02-15 Oksazolidinonforbindelser og sammensetninger og fremgangsmater relatert dertil

Country Status (17)

Country Link
US (1) US20090005369A1 (no)
EP (1) EP1786805A1 (no)
JP (1) JP2008508236A (no)
KR (1) KR20070048227A (no)
CN (1) CN101027296A (no)
AR (1) AR050426A1 (no)
AU (1) AU2005266318A1 (no)
BR (1) BRPI0512691A (no)
CA (1) CA2574668A1 (no)
MX (1) MX2007001065A (no)
NO (1) NO20070870L (no)
PA (1) PA8640401A1 (no)
PE (1) PE20060619A1 (no)
RU (1) RU2007107490A (no)
TW (1) TW200612923A (no)
UY (1) UY29012A1 (no)
WO (1) WO2006010756A1 (no)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102006033572A1 (de) * 2006-07-20 2008-01-24 Bayer Cropscience Ag N'-Cyano-N-halogenalkyl-imidamid Derivate
EP2072513A1 (en) * 2007-12-17 2009-06-24 Ferrer Internacional, S.A. A cyano piperidinyl-phenil-oxazolidinone and use thereof
US9173887B2 (en) 2010-12-22 2015-11-03 Abbvie Inc. Hepatitis C inhibitors and uses thereof
CN103483329B (zh) * 2013-09-07 2015-08-05 吉首大学 呋喃酮-芳基-噁唑烷酮型化合物及其制法和用途
CN103420996B (zh) * 2013-09-07 2015-06-24 吉首大学 苯并吡喃酮-胺甲基-噁唑烷酮类化合物及其制法和用途
CN103420995B (zh) * 2013-09-07 2015-07-01 吉首大学 噁唑烷酮-烷胺基-呋喃酮型化合物及其制法和用途

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1250538A (no) * 1969-03-18 1971-10-20
DE19962924A1 (de) * 1999-12-24 2001-07-05 Bayer Ag Substituierte Oxazolidinone und ihre Verwendung
DE10105989A1 (de) * 2001-02-09 2002-08-14 Bayer Ag Substituierte Oxazolidinone und ihre Verwendung
CA2463794A1 (en) 2001-11-29 2003-06-12 Merck & Co., Inc. Cyclopropyl hexane containing oxazolidinone antibiotics and derivatives thereof
TW200302095A (en) 2002-01-25 2003-08-01 Upjohn Co Oxazolidinone cotherapy
JP2005527575A (ja) * 2002-03-29 2005-09-15 ファルマシア・アンド・アップジョン・カンパニー・エルエルシー 糖尿病性足病変感染を治療するためのオキサゾリジノンの非経口、静脈内および経口投与
US20080214565A1 (en) * 2003-04-07 2008-09-04 Anita Mehta Oxazolidinone Derivatives as Antimicrobials

Also Published As

Publication number Publication date
WO2006010756A1 (en) 2006-02-02
RU2007107490A (ru) 2008-09-10
US20090005369A1 (en) 2009-01-01
MX2007001065A (es) 2007-04-10
KR20070048227A (ko) 2007-05-08
CN101027296A (zh) 2007-08-29
CA2574668A1 (en) 2006-02-02
JP2008508236A (ja) 2008-03-21
PE20060619A1 (es) 2006-07-11
UY29012A1 (es) 2005-10-31
TW200612923A (en) 2006-05-01
EP1786805A1 (en) 2007-05-23
AU2005266318A1 (en) 2006-02-02
AR050426A1 (es) 2006-10-25
PA8640401A1 (es) 2006-03-24
BRPI0512691A (pt) 2008-04-01

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Legal Events

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FC2A Withdrawal, rejection or dismissal of laid open patent application