NO20052995L - 1,5-diaryl-pyrrol-3-karboksamid-derivater, og deres anvendelse som kannabinoid reseptormodulatorer. - Google Patents

1,5-diaryl-pyrrol-3-karboksamid-derivater, og deres anvendelse som kannabinoid reseptormodulatorer.

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Publication number
NO20052995L
NO20052995L NO20052995A NO20052995A NO20052995L NO 20052995 L NO20052995 L NO 20052995L NO 20052995 A NO20052995 A NO 20052995A NO 20052995 A NO20052995 A NO 20052995A NO 20052995 L NO20052995 L NO 20052995L
Authority
NO
Norway
Prior art keywords
group
alkyl group
optionally substituted
alkyl
heterocyclic group
Prior art date
Application number
NO20052995A
Other languages
English (en)
Norwegian (no)
Other versions
NO20052995D0 (no
Inventor
Stig Jonas Bostrom
Anna Ingrid Kristina Berggren
Stig Thomas Elebring
Peter Greasley
Johan Michael Wilstermann
Leifeng Cheng
Mats Nagard
Emma Terricabras
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NO20052995D0 publication Critical patent/NO20052995D0/no
Publication of NO20052995L publication Critical patent/NO20052995L/no

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    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4021-aryl substituted, e.g. piretanide
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • A61K31/4523Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
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    • C07D207/02Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

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  • Hospice & Palliative Care (AREA)
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  • Pulmonology (AREA)
  • Reproductive Health (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO20052995A 2002-12-24 2005-06-17 1,5-diaryl-pyrrol-3-karboksamid-derivater, og deres anvendelse som kannabinoid reseptormodulatorer. NO20052995L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB0230088.7A GB0230088D0 (en) 2002-12-24 2002-12-24 Therapeutic agents
PCT/GB2003/005569 WO2004058249A1 (en) 2002-12-24 2003-12-18 1,5-diaryl-pyrrole-3-carboxamide derivatives and their use as cannabinoid receptor modulators

Publications (2)

Publication Number Publication Date
NO20052995D0 NO20052995D0 (no) 2005-06-17
NO20052995L true NO20052995L (no) 2005-07-22

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NO20052995A NO20052995L (no) 2002-12-24 2005-06-17 1,5-diaryl-pyrrol-3-karboksamid-derivater, og deres anvendelse som kannabinoid reseptormodulatorer.

Country Status (20)

Country Link
US (1) US20060122230A1 (pl)
EP (1) EP1578417A1 (pl)
JP (1) JP2006513201A (pl)
KR (1) KR20050086931A (pl)
CN (1) CN1753668A (pl)
AR (1) AR042658A1 (pl)
AU (1) AU2003290292A1 (pl)
BR (1) BR0317705A (pl)
CA (1) CA2511601A1 (pl)
CL (1) CL2003002720A1 (pl)
GB (1) GB0230088D0 (pl)
IS (1) IS7944A (pl)
MX (1) MXPA05006919A (pl)
NO (1) NO20052995L (pl)
PL (1) PL377296A1 (pl)
RU (1) RU2005117783A (pl)
TW (1) TW200503692A (pl)
UY (1) UY28144A1 (pl)
WO (1) WO2004058249A1 (pl)
ZA (1) ZA200504822B (pl)

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EP2683701B1 (de) 2011-03-08 2014-12-24 Sanofi Mit benzyl- oder heteromethylengruppen substituierte oxathiazinderivate, verfahren zu deren herstellung, ihre verwendung als medikament sowie sie enthaltendes arzneimittel und deren verwendung
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WO2004058249A1 (en) 2004-07-15
CA2511601A1 (en) 2004-07-15
CL2003002720A1 (es) 2005-01-07
NO20052995D0 (no) 2005-06-17
CN1753668A (zh) 2006-03-29
US20060122230A1 (en) 2006-06-08
ZA200504822B (en) 2006-03-29
JP2006513201A (ja) 2006-04-20
KR20050086931A (ko) 2005-08-30
MXPA05006919A (es) 2005-08-18
EP1578417A1 (en) 2005-09-28
AR042658A1 (es) 2005-06-29
GB0230088D0 (en) 2003-01-29
UY28144A1 (es) 2004-07-30
PL377296A1 (pl) 2006-01-23
TW200503692A (en) 2005-02-01
RU2005117783A (ru) 2006-02-10
BR0317705A (pt) 2005-11-22
AU2003290292A1 (en) 2004-07-22

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