NO20051289L - Lincomycinderivater som fremviser antibakteriell aktivitet. - Google Patents

Lincomycinderivater som fremviser antibakteriell aktivitet.

Info

Publication number
NO20051289L
NO20051289L NO20051289A NO20051289A NO20051289L NO 20051289 L NO20051289 L NO 20051289L NO 20051289 A NO20051289 A NO 20051289A NO 20051289 A NO20051289 A NO 20051289A NO 20051289 L NO20051289 L NO 20051289L
Authority
NO
Norway
Prior art keywords
antibacterial activity
exhibiting antibacterial
derivatives exhibiting
lincomycin derivatives
linkomycin
Prior art date
Application number
NO20051289A
Other languages
English (en)
Norwegian (no)
Inventor
Dinesh V Patel
Mikhail F Gordeev
Jason Lewis
Sampath K Anandan
Original Assignee
Vicuron Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vicuron Pharm Inc filed Critical Vicuron Pharm Inc
Publication of NO20051289L publication Critical patent/NO20051289L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
    • C07H15/16—Lincomycin; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Saccharide Compounds (AREA)
NO20051289A 2002-08-15 2005-03-14 Lincomycinderivater som fremviser antibakteriell aktivitet. NO20051289L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US40377002P 2002-08-15 2002-08-15
PCT/US2003/025820 WO2004016632A2 (en) 2002-08-15 2003-08-15 Lincomycin derivatives possessing antibacterial activity

Publications (1)

Publication Number Publication Date
NO20051289L true NO20051289L (no) 2005-05-09

Family

ID=31888275

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20051289A NO20051289L (no) 2002-08-15 2005-03-14 Lincomycinderivater som fremviser antibakteriell aktivitet.

Country Status (15)

Country Link
US (1) US7164011B2 (enExample)
EP (1) EP1529052A2 (enExample)
JP (1) JP2006504673A (enExample)
KR (1) KR20050056195A (enExample)
CN (1) CN1315859C (enExample)
AU (1) AU2003265475B2 (enExample)
BR (1) BR0313725A (enExample)
CA (1) CA2493799A1 (enExample)
EA (1) EA200500353A1 (enExample)
IL (1) IL166476A (enExample)
MX (1) MXPA05001689A (enExample)
NO (1) NO20051289L (enExample)
NZ (1) NZ538141A (enExample)
WO (1) WO2004016632A2 (enExample)
ZA (1) ZA200501012B (enExample)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7199105B2 (en) 2002-08-15 2007-04-03 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
WO2004016632A2 (en) 2002-08-15 2004-02-26 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
US7256177B2 (en) 2003-06-17 2007-08-14 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
CA2528596A1 (en) * 2003-06-17 2005-01-27 Vicuron Pharmaceuticals Inc. Lincomycin derivatives possessing antibacterial activity
US7199106B2 (en) 2003-06-17 2007-04-03 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antimicrobial activity
AU2004261550A1 (en) * 2003-06-17 2005-02-10 Vicuron Pharmaceuticals, Inc. Novel lincomycin derivatives possessing antimicrobial activity
US7361743B2 (en) 2004-02-11 2008-04-22 Pfizer Inc Lincomycin derivatives possessing antibacterial activity
JP5064237B2 (ja) * 2005-12-09 2012-10-31 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 リンコマイシン誘導体およびこれを有効成分とする抗菌剤
JP5356223B2 (ja) * 2007-05-31 2013-12-04 Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 リンコマイシン誘導体及びこれを有効成分とする抗菌剤
US7867980B2 (en) * 2007-05-31 2011-01-11 Meiji Seika Kaisha, Ltd. Lincosamide derivatives and antimicrobial agents comprising the same as active ingredient
CN101555223B (zh) * 2009-04-17 2011-06-01 北京化工大学 一种吡利霉素中间体及其制备方法
US9533973B2 (en) 2011-12-08 2017-01-03 The Board Of Regents Of The University Of Texas System Allosteric modulators of 5-hydroxytryptamine 2C receptor (5-HT2CR)
CN105566411B (zh) * 2014-11-07 2020-11-13 中国科学院上海有机化学研究所 林可霉素生物合成中间产物及其制法和用途

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US2851463A (en) 1956-04-09 1958-09-09 Upjohn Co Desalicetin and salts, and hydrocarbon carboxylic acid esters
US2928844A (en) 1958-02-24 1960-03-15 Upjohn Co Celesticetin, its salts and method of preparation
US3086912A (en) 1961-07-03 1963-04-23 Upjohn Co Antibiotic lincolnensin and method of production
US3268556A (en) 1964-04-13 1966-08-23 Upjohn Co Novel lincomycin derivatives
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NL140527B (nl) 1965-02-08 1973-12-17 Upjohn Co Werkwijze ter bereiding van aan lincomycine verwante verbindingen.
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US3475407A (en) 1967-12-22 1969-10-28 Upjohn Co Process for preparing 7(r)- and 7(s)-halolincomycins
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US3544551A (en) 1968-04-30 1970-12-01 Upjohn Co 7-mercapto-7-deoxylincomycins and process for preparing the same
US3555007A (en) 1968-07-22 1971-01-12 Upjohn Co 7-deoxy-7-halo lincomycin d derivatives
US3549615A (en) * 1968-10-17 1970-12-22 Upjohn Co Lincomycin derivatives and process for producing the same
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DE2118636A1 (de) 1970-04-20 1971-11-04 The Upjohn Co., Kalamazoo, Mich. (V.StA.) 3-Nucleotide von Lincomycin und deren Analogen, Verfahren zu ihrer Herstellung und ihre Verwendung in therapeutischen Präparaten
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US3915954A (en) 1971-11-15 1975-10-28 Upjohn Co Derivatives of lincomycin and its analogs and process
BE793630A (fr) 1972-01-03 1973-07-03 Upjohn Co Nouvel antibiotique de la classe des celesticetines et son procede de preparation
US3853843A (en) 1972-12-13 1974-12-10 Upjohn Co Derivatives of thiolincosaminide compounds
US3849396A (en) 1973-01-08 1974-11-19 Upjohn Co Lincomycin and clindamycin 1-o-ethers
US3870699A (en) 1973-03-06 1975-03-11 Upjohn Co Lincomycin analogs
US3833475A (en) 1973-04-23 1974-09-03 Upjohn Co Process for preparing lincomycin
US4271266A (en) 1974-06-10 1981-06-02 The Upjohn Manufacturing Company Process for preparing lincomycin
US4031304A (en) 1976-01-30 1977-06-21 The Upjohn Company Process for preparing lincomycin derivatives
US4278789A (en) 1979-11-23 1981-07-14 The Upjohn Company Lincomycin compounds
US4309533A (en) 1980-05-19 1982-01-05 The Upjohn Company Lincomycin compounds
US4310660A (en) 1980-05-19 1982-01-12 The Upjohn Company Lincomycin compounds
US4293547A (en) 1980-08-25 1981-10-06 The Upjohn Company Method of treating malaria
US4317903A (en) 1981-01-26 1982-03-02 The Upjohn Company Process for the purification of lincomycin
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US4430495A (en) 1982-09-17 1984-02-07 The Upjohn Company Process for preparing lincomycin and clindamycin ribonucleotides
US4568741A (en) 1984-05-15 1986-02-04 The Upjohn Company Synthesis of 7-halo-7-deoxylincomycins
CN1004002B (zh) 1984-11-29 1989-04-26 厄普约翰公司 制备7-卤-7-去氧林可霉素及其类似化合物的改进方法
WO1989004672A1 (en) 1987-11-20 1989-06-01 The Upjohn Company Derivatives of lincosaminide antibiotics
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WO2004016632A2 (en) 2002-08-15 2004-02-26 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
US7199105B2 (en) 2002-08-15 2007-04-03 Vicuron Pharmaceuticals, Inc. Lincomycin derivatives possessing antibacterial activity
AU2004261550A1 (en) 2003-06-17 2005-02-10 Vicuron Pharmaceuticals, Inc. Novel lincomycin derivatives possessing antimicrobial activity
CA2528596A1 (en) 2003-06-17 2005-01-27 Vicuron Pharmaceuticals Inc. Lincomycin derivatives possessing antibacterial activity

Also Published As

Publication number Publication date
IL166476A (en) 2010-05-31
AU2003265475A1 (en) 2004-03-03
WO2004016632A3 (en) 2004-06-24
EA200500353A1 (ru) 2006-06-30
CN1315859C (zh) 2007-05-16
WO2004016632A2 (en) 2004-02-26
US20040116690A1 (en) 2004-06-17
CA2493799A1 (en) 2004-02-26
NZ538141A (en) 2007-06-29
EP1529052A2 (en) 2005-05-11
CN1681832A (zh) 2005-10-12
KR20050056195A (ko) 2005-06-14
US7164011B2 (en) 2007-01-16
ZA200501012B (en) 2006-10-25
IL166476A0 (en) 2006-01-15
BR0313725A (pt) 2006-06-13
WO2004016632A8 (en) 2004-09-30
WO2004016632B1 (en) 2004-08-19
AU2003265475B2 (en) 2009-08-27
MXPA05001689A (es) 2005-05-27
JP2006504673A (ja) 2006-02-09

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