NO20034836L - Sammensmeltede pyrimidiner som antagonister av kortikotropinfrigivelsesfaktoren (CRF) - Google Patents

Sammensmeltede pyrimidiner som antagonister av kortikotropinfrigivelsesfaktoren (CRF)

Info

Publication number
NO20034836L
NO20034836L NO20034836A NO20034836A NO20034836L NO 20034836 L NO20034836 L NO 20034836L NO 20034836 A NO20034836 A NO 20034836A NO 20034836 A NO20034836 A NO 20034836A NO 20034836 L NO20034836 L NO 20034836L
Authority
NO
Norway
Prior art keywords
crf
pyrimidines
antagonists
concentrated
release factor
Prior art date
Application number
NO20034836A
Other languages
English (en)
Norwegian (no)
Other versions
NO20034836D0 (no
Inventor
Anna Maria Capelli
Benedetta Perini
Chiara Marchionni
Yves St-Denis
Fabrizio Micheli
Romano Di Fabio
Alessandra Pasquarello
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0110567A external-priority patent/GB0110567D0/en
Priority claimed from GB0110569A external-priority patent/GB0110569D0/en
Priority claimed from GB0110570A external-priority patent/GB0110570D0/en
Priority claimed from GB0117399A external-priority patent/GB0117399D0/en
Priority claimed from GB0117401A external-priority patent/GB0117401D0/en
Priority claimed from GB0117420A external-priority patent/GB0117420D0/en
Priority claimed from GB0203201A external-priority patent/GB0203201D0/en
Priority claimed from GB0206834A external-priority patent/GB0206834D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of NO20034836D0 publication Critical patent/NO20034836D0/no
Publication of NO20034836L publication Critical patent/NO20034836L/no

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
    • A61K51/04—Organic compounds
    • A61K51/041—Heterocyclic compounds
    • A61K51/044—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K51/0459—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
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    • A61K51/0463—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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    • C07D—HETEROCYCLIC COMPOUNDS
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NO20034836A 2001-04-30 2003-10-29 Sammensmeltede pyrimidiner som antagonister av kortikotropinfrigivelsesfaktoren (CRF) NO20034836L (no)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
GB0110567A GB0110567D0 (en) 2001-04-30 2001-04-30 Chemical compounds
GB0110569A GB0110569D0 (en) 2001-04-30 2001-04-30 Chemical compounds
GB0110570A GB0110570D0 (en) 2001-04-30 2001-04-30 Chemical compounds
GB0117399A GB0117399D0 (en) 2001-07-17 2001-07-17 Chemical compounds
GB0117401A GB0117401D0 (en) 2001-07-17 2001-07-17 Chemical compounds
GB0117420A GB0117420D0 (en) 2001-07-17 2001-07-17 Chemical compounds
GB0203201A GB0203201D0 (en) 2002-02-11 2002-02-11 Chemical compounds
GB0206834A GB0206834D0 (en) 2002-03-22 2002-03-22 Chemical compounds
PCT/GB2002/002029 WO2002088095A1 (en) 2001-04-30 2002-04-30 Fused pyrimidines as antagonists of the corticotropin releasing factor (crf)

Publications (2)

Publication Number Publication Date
NO20034836D0 NO20034836D0 (no) 2003-10-29
NO20034836L true NO20034836L (no) 2003-10-29

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NO20034836A NO20034836L (no) 2001-04-30 2003-10-29 Sammensmeltede pyrimidiner som antagonister av kortikotropinfrigivelsesfaktoren (CRF)

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Families Citing this family (61)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002100863A1 (en) * 2001-06-12 2002-12-19 Glaxo Group Limited Corticotropin releasing factor antagonists
GB0117396D0 (en) * 2001-07-17 2001-09-05 Glaxo Group Ltd Chemical compounds
EP1583531B1 (en) * 2003-01-16 2007-04-18 SB Pharmco Puerto Rico Inc Heteroaryl-substituted pyrrolo[2, 3- b]pyridine derivatives as crf receptor antagonists
US7772188B2 (en) 2003-01-28 2010-08-10 Ironwood Pharmaceuticals, Inc. Methods and compositions for the treatment of gastrointestinal disorders
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KR20040015206A (ko) 2004-02-18
CA2446514A1 (en) 2002-11-07
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PL366934A1 (en) 2005-02-07
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AU2002253357B2 (en) 2006-08-24
ATE386727T1 (de) 2008-03-15
WO2002088095A1 (en) 2002-11-07
DE60225127D1 (en) 2008-04-03
CN1649848A (zh) 2005-08-03
CZ20032946A3 (en) 2004-05-12
DE60225127T2 (de) 2009-02-19
BR0209267A (pt) 2004-06-15
US7279474B2 (en) 2007-10-09
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EP1383747B1 (en) 2008-02-20
US20040176400A1 (en) 2004-09-09

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