NO20030772D0 - Fremgangsmåte til fremstilling av vannfritt azitromycin - Google Patents

Fremgangsmåte til fremstilling av vannfritt azitromycin

Info

Publication number
NO20030772D0
NO20030772D0 NO20030772A NO20030772A NO20030772D0 NO 20030772 D0 NO20030772 D0 NO 20030772D0 NO 20030772 A NO20030772 A NO 20030772A NO 20030772 A NO20030772 A NO 20030772A NO 20030772 D0 NO20030772 D0 NO 20030772D0
Authority
NO
Norway
Prior art keywords
preparation
anhydrous azithromycin
azithromycin
anhydrous
antibiotics
Prior art date
Application number
NO20030772A
Other languages
English (en)
Other versions
NO20030772L (no
Inventor
Shiva P Singh
Siddiqui Mohammed Jaw Mukarram
Manish Purohit
Anjum Reyaz Khan
Original Assignee
Anjum Reyaz Khan
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Anjum Reyaz Khan filed Critical Anjum Reyaz Khan
Publication of NO20030772D0 publication Critical patent/NO20030772D0/no
Publication of NO20030772L publication Critical patent/NO20030772L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicinal Preparation (AREA)
NO20030772A 2000-08-23 2003-02-18 Fremgangsmate til fremstilling av vannfritt azitromycin NO20030772L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US22734100P 2000-08-23 2000-08-23
PCT/IB2001/001523 WO2002015842A2 (en) 2000-08-23 2001-08-23 Process for preparation of anhydrous azithromycin

Publications (2)

Publication Number Publication Date
NO20030772D0 true NO20030772D0 (no) 2003-02-18
NO20030772L NO20030772L (no) 2003-04-22

Family

ID=22852706

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20030772A NO20030772L (no) 2000-08-23 2003-02-18 Fremgangsmate til fremstilling av vannfritt azitromycin

Country Status (10)

Country Link
US (2) US7414114B2 (no)
EP (1) EP1313749B1 (no)
JP (1) JP2004506664A (no)
AT (1) ATE306491T1 (no)
AU (1) AU2001280000A1 (no)
CA (1) CA2419873A1 (no)
DE (1) DE60114028T2 (no)
NO (1) NO20030772L (no)
WO (1) WO2002015842A2 (no)
ZA (1) ZA200301384B (no)

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JP2004530703A (ja) 2001-05-22 2004-10-07 ファイザー・プロダクツ・インク 結晶形アジスロマイシン
US6861413B2 (en) 2001-05-22 2005-03-01 Pfizer Inc. Stable non-dihydrate azithromycin oral suspensions
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HRP20020614A2 (en) 2002-07-22 2004-06-30 PLIVA-ISTRAŽIVAČKI INSTITUT d.o.o. Rhombic pseudopolymorph of 9-deoxo-9a-aza-9a-methyl-9a-homoerythromycin a
US7435805B2 (en) * 2003-05-30 2008-10-14 Glaxpsmithkline Istrazivacki O-alkyl macrolide and azalide derivatives and regioselective process for their preparation
US20060116336A1 (en) * 2004-03-17 2006-06-01 American Pharmaceutical Partners, Inc. Lyophilized azithromycin formulation
US7468428B2 (en) * 2004-03-17 2008-12-23 App Pharmaceuticals, Llc Lyophilized azithromycin formulation
US7683162B2 (en) 2004-08-30 2010-03-23 Taro Pharmaceutical Industries Limited Process of preparing a crystalline azithromycin monohydrate
WO2007080507A2 (en) * 2006-01-12 2007-07-19 Wockhardt Ltd Processes for the preparation of azithromycin
MX2011009548A (es) 2009-03-13 2011-12-14 Da Volterra Composiciones y metodos para la eliminacion de bacterias gram-negativas.
US8106111B2 (en) 2009-05-15 2012-01-31 Eastman Chemical Company Antimicrobial effect of cycloaliphatic diol antimicrobial agents in coating compositions
DK2661254T3 (da) 2011-01-05 2017-11-06 Hospira Inc Sprøjtetørring af vancomycin
US20130172271A1 (en) * 2012-01-04 2013-07-04 Cynthia Fragale Pharmaceutical Spray Drying
CN103897002A (zh) * 2012-12-31 2014-07-02 菏泽市方明制药有限公司 一种粗品硫氰酸红霉素制备红霉素a9-肟的方法
CN104043104B (zh) 2013-03-15 2018-07-10 浙江创新生物有限公司 含盐酸万古霉素的喷雾干粉及其工业化制备方法

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WO1992006991A1 (fr) * 1990-10-15 1992-04-30 Taisho Pharmaceutical Co., Ltd. Erythromycine modifiee en 2' ou derive de cette substance
US5202434A (en) 1991-04-05 1993-04-13 Merck & Co., Inc. 8a-aza-8a-homoerythromycin lactams
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US5215980A (en) 1992-01-17 1993-06-01 Merck & Co., Inc. 10-AZA-9-deoxo-11-deoxy-erythromycin A and derivatives thereof
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US5441939A (en) 1994-03-04 1995-08-15 Pfizer Inc. 3"-desmethoxy derivatives of erythromycin and azithromycin
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PT102006B (pt) 1997-05-19 2000-06-30 Hovione Sociedade Quimica S A Novo processo de preparacao de azitromicina
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CA2245398C (en) * 1998-08-21 2002-01-29 Apotex Inc. Azithromycin monohydrate isopropanol clathrate and methods for the manufacture thereof
AU2001214115A1 (en) * 2000-08-01 2002-02-13 Habil F. Khorakiwala Process for the preparation of anhydrous azithromycin
JP2004506664A (ja) * 2000-08-23 2004-03-04 ウォックハート・リミテッド 無水アジトロマイシンの製造法
JP2004530703A (ja) * 2001-05-22 2004-10-07 ファイザー・プロダクツ・インク 結晶形アジスロマイシン
US6855813B2 (en) * 2002-07-19 2005-02-15 Alembic Limited Process for the preparation of azithromycin monohydrate
US7235646B2 (en) * 2004-06-28 2007-06-26 Alembic Limited Process for the preparation of azithromycin monohydrate isopropanol clathrate
US7683162B2 (en) * 2004-08-30 2010-03-23 Taro Pharmaceutical Industries Limited Process of preparing a crystalline azithromycin monohydrate

Also Published As

Publication number Publication date
ATE306491T1 (de) 2005-10-15
WO2002015842A2 (en) 2002-02-28
CA2419873A1 (en) 2002-02-28
JP2004506664A (ja) 2004-03-04
ZA200301384B (en) 2004-04-02
US20030139583A1 (en) 2003-07-24
AU2001280000A1 (en) 2002-03-04
NO20030772L (no) 2003-04-22
EP1313749A2 (en) 2003-05-28
US7414114B2 (en) 2008-08-19
EP1313749A4 (en) 2004-01-21
EP1313749B1 (en) 2005-10-12
DE60114028D1 (de) 2006-02-23
DE60114028T2 (de) 2006-07-13
WO2002015842A3 (en) 2002-10-31
US20090018090A1 (en) 2009-01-15

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