NO20013517L - Makrolider med anti-inflammatorisk aktivitet - Google Patents

Makrolider med anti-inflammatorisk aktivitet

Info

Publication number
NO20013517L
NO20013517L NO20013517A NO20013517A NO20013517L NO 20013517 L NO20013517 L NO 20013517L NO 20013517 A NO20013517 A NO 20013517A NO 20013517 A NO20013517 A NO 20013517A NO 20013517 L NO20013517 L NO 20013517L
Authority
NO
Norway
Prior art keywords
macrolides
inflammatory activity
oxyimino
endowed
dimethylamino
Prior art date
Application number
NO20013517A
Other languages
English (en)
Other versions
NO20013517D0 (no
NO318982B1 (no
Inventor
Franco Pellacini
Daniela Botta
Stefano Romagnano
Ermanno Moriggi
Lorenzo Pradella
Original Assignee
Zambon Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon Spa filed Critical Zambon Spa
Publication of NO20013517D0 publication Critical patent/NO20013517D0/no
Publication of NO20013517L publication Critical patent/NO20013517L/no
Publication of NO318982B1 publication Critical patent/NO318982B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Rheumatology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pain & Pain Management (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
NO20013517A 1999-01-15 2001-07-16 Makrolider med anti-inflammatorisk aktivitet, farmasoytisk sammensetning som inneholder disse og anvendelse av 3'-desdimetylamino-3', 4'-dehydroerytromycin A- oksim og 3'-desdimetylamino-3', 4'dehydroerytromycin A-9-O-metyloksim som anti-inflammatoriske forbindelser NO318982B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT1999MI000061A IT1306205B1 (it) 1999-01-15 1999-01-15 Macrolidi ad attivita' antiinfiammatoria.
PCT/EP2000/000163 WO2000042055A2 (en) 1999-01-15 2000-01-12 Macrolides with anti-inflammatory activity

Publications (3)

Publication Number Publication Date
NO20013517D0 NO20013517D0 (no) 2001-07-16
NO20013517L true NO20013517L (no) 2001-07-16
NO318982B1 NO318982B1 (no) 2005-05-30

Family

ID=11381492

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20013517A NO318982B1 (no) 1999-01-15 2001-07-16 Makrolider med anti-inflammatorisk aktivitet, farmasoytisk sammensetning som inneholder disse og anvendelse av 3'-desdimetylamino-3', 4'-dehydroerytromycin A- oksim og 3'-desdimetylamino-3', 4'dehydroerytromycin A-9-O-metyloksim som anti-inflammatoriske forbindelser

Country Status (19)

Country Link
US (1) US6455576B1 (no)
EP (1) EP1144427B1 (no)
JP (1) JP4568433B2 (no)
CN (1) CN1151165C (no)
AT (1) ATE308552T1 (no)
AU (1) AU769006B2 (no)
BR (1) BR0007514A (no)
CA (1) CA2368400C (no)
DE (1) DE60023647T2 (no)
ES (1) ES2251966T3 (no)
HU (1) HU229228B1 (no)
IL (2) IL144044A0 (no)
IT (1) IT1306205B1 (no)
MX (1) MXPA01007164A (no)
NO (1) NO318982B1 (no)
RU (1) RU2243230C2 (no)
SK (1) SK286772B6 (no)
WO (1) WO2000042055A2 (no)
ZA (1) ZA200105748B (no)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HRP20010018A2 (en) 2001-01-09 2002-12-31 Pliva D D Novel anti-inflammatory compounds
AU2003255849A1 (en) * 2002-07-08 2004-01-23 Glaxosmithkline Istrazivacki Centar Zagreb D.O.O. Novel nonsteroidal anti-inflammatory substances, compositions and methods for their use
ATE429441T1 (de) 2002-07-08 2009-05-15 Glaxosmithkline Zagreb Hybridmoleküle von makroliden mit steroidalen/nicht-steroidalen antientzündlich aktiven molekülen
AU2003255851B2 (en) 2002-07-08 2009-07-23 Glaxosmithkline Istrazivacki Centar Zagreb D.O.O. New compounds, compositions and methods for treatment of inflammatory diseases and conditions
ITMI20021726A1 (it) * 2002-08-01 2004-02-02 Zambon Spa Macrolidi ad attivita' antiinfiammatoria.
US7091196B2 (en) 2002-09-26 2006-08-15 Rib-X Pharmaceuticals, Inc. Bifunctional heterocyclic compounds and methods of making and using same
ITMI20022292A1 (it) * 2002-10-29 2004-04-30 Zambon Spa 9a-azalidi ad attivita' antiinfiammatoria.
CA2521462A1 (en) * 2003-04-17 2004-10-28 Sandoz Ag Derivatives of azithromycin
HRP20030324A2 (en) 2003-04-24 2005-02-28 Pliva-Istra�iva�ki institut d.o.o. Compounds of antiinflammatory effect
ITMI20040124A1 (it) * 2004-01-29 2004-04-29 Zambon Spa Macrolidi ad attivita' antiinfiammatoria
WO2006130128A2 (en) * 2004-02-18 2006-12-07 Chiron Corporation Methods of identifying anti-inflammatory macrolides
CN102816194A (zh) 2004-02-27 2012-12-12 瑞伯-X医药品有限公司 大环化合物以及其制作和使用方法
US20080318878A1 (en) * 2004-09-27 2008-12-25 Biswajit Das Antibacterial Agents
MX2007005073A (es) 2004-10-27 2007-06-25 Glaxosmithkline Zagreb Conjugados con actividad antiinflamtoria.
US20080249034A1 (en) * 2005-03-21 2008-10-09 Zambon S.P.A. Use of Macrolides for Treating Intestinal Inflammation
US7582611B2 (en) * 2005-05-24 2009-09-01 Pfizer Inc. Motilide compounds
US20110178287A1 (en) 2010-01-19 2011-07-21 Cerulean Pharma Inc. Cyclodextrin-based polymers for therapeutic delivery
RU2455309C2 (ru) * 2010-07-20 2012-07-10 Открытое Акционерное Общество "Татхимфармпрепараты" Способ получения аморфной формы рокситромицина
GB201608236D0 (en) 2016-05-11 2016-06-22 Fidelta D O O Seco macrolide compounds
AU2021241591A1 (en) 2020-03-24 2022-10-20 Michael W. BURNET Anti-infective and anti-viral compounds and compositions

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3928387A (en) * 1974-02-04 1975-12-23 Hoffmann La Roche Antibiotic 1745A/X and methods for the production thereof
IT1189285B (it) * 1982-05-28 1988-02-04 Nuovo Consor Sanitar Nazionale Sali dell'antibiotico eritromicina e del suo estere propionico con acidi ad attivita' terapeutica coadiuvante
EP0254534A3 (en) * 1986-07-24 1991-04-17 William S. Robinson Erythromycin derivatives and compositions and use for inhibiting virus replication and disease
IT1276901B1 (it) * 1994-12-13 1997-11-03 Zambon Spa Derivati dell'eritromicina a 9-0-ossina dotati di attivita' antibiotica
WO1996027391A1 (fr) * 1995-03-08 1996-09-12 Environmental Research Institute, Inc. Medicament pour le traitement de maladies liees a l'immunite et leur technique d'elaboration

Also Published As

Publication number Publication date
ATE308552T1 (de) 2005-11-15
ES2251966T3 (es) 2006-05-16
JP4568433B2 (ja) 2010-10-27
CA2368400C (en) 2007-06-05
NO20013517D0 (no) 2001-07-16
AU2663600A (en) 2000-08-01
HUP0105105A2 (hu) 2002-04-29
SK286772B6 (sk) 2009-05-07
IT1306205B1 (it) 2001-05-30
HUP0105105A3 (en) 2003-05-28
MXPA01007164A (es) 2002-03-27
EP1144427B1 (en) 2005-11-02
DE60023647D1 (de) 2005-12-08
EP1144427A3 (en) 2002-08-28
BR0007514A (pt) 2001-11-20
ITMI990061A1 (it) 2000-07-15
NO318982B1 (no) 2005-05-30
IL144044A0 (en) 2002-04-21
DE60023647T2 (de) 2006-08-10
CA2368400A1 (en) 2000-07-20
US6455576B1 (en) 2002-09-24
IL144044A (en) 2006-12-31
WO2000042055A3 (en) 2001-09-07
SK9812001A3 (en) 2002-01-07
AU769006B2 (en) 2004-01-15
RU2243230C2 (ru) 2004-12-27
WO2000042055A2 (en) 2000-07-20
JP2002534531A (ja) 2002-10-15
ZA200105748B (en) 2002-10-14
HU229228B1 (en) 2013-09-30
CN1336932A (zh) 2002-02-20
EP1144427A2 (en) 2001-10-17
CN1151165C (zh) 2004-05-26

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