NO20006507L - Propenyl kefalosporinderivater - Google Patents
Propenyl kefalosporinderivaterInfo
- Publication number
- NO20006507L NO20006507L NO20006507A NO20006507A NO20006507L NO 20006507 L NO20006507 L NO 20006507L NO 20006507 A NO20006507 A NO 20006507A NO 20006507 A NO20006507 A NO 20006507A NO 20006507 L NO20006507 L NO 20006507L
- Authority
- NO
- Norway
- Prior art keywords
- hydrogen
- carbon
- sulfur
- nitrogen
- exceeding
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/38—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof
- C07D501/40—Methylene radicals, substituted by nitrogen atoms; Lactams thereof with the 2-carboxyl group; Methylene radicals substituted by nitrogen-containing hetero rings attached by the ring nitrogen atom; Quaternary compounds thereof with the 7-amino radical acylated by an aliphatic carboxylic acid, which is substituted by hetero atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cephalosporin Compounds (AREA)
Abstract
Fremlagt er kefalosporinderivater med den generelle forme- len R-S-CH^ CDCH hvori R er en organisk residu med en molekylvekt som ikke overstiger 400 bundet til det tilgrensende svovelatomet via karbon og består av karbon, hydrogen, og valgfritt oksygen, svovel, nitrogen og/eller halogenatomer; R1 er hydrogen, lavere alkyl eller fenyl; og A er et sekundært, tertiært eller kvaternært nitrogen atom bundet direkte til propenylgruppen og er substituert med en organisk residu med en molekylvekt som ikke overstiger 400 og består av karbon, hydrogen, og valgfritt oksygen, svovel, nitrogen og/eller halogenatomer, i tillegg til lett hydrolyserbare estere derav, farmasøytisk akseptable salter av forbindel- sene og hydrater av forbindelsene med formel I og av deres estere og salter. Også fremlagt er en prosess for deres fremstilling, mellomprodukter anvendbare deri. Medikamen- ter inneholdende sluttproduktene og anvendelse av sist- nevnte for behandling og profylakse av infeksjonssykdommer eller for fremstillingen av medikamentene.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP98111415 | 1998-06-22 | ||
EP99108149 | 1999-04-26 | ||
PCT/EP1999/004034 WO1999067255A1 (en) | 1998-06-22 | 1999-06-11 | Propenyl cephalosporin derivatives |
Publications (2)
Publication Number | Publication Date |
---|---|
NO20006507L true NO20006507L (no) | 2000-12-20 |
NO20006507D0 NO20006507D0 (no) | 2000-12-20 |
Family
ID=26149364
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20006507A NO20006507D0 (no) | 1998-06-22 | 2000-12-20 | Propenyl kefalosporinderivater |
Country Status (16)
Country | Link |
---|---|
US (1) | US6583133B1 (no) |
EP (1) | EP1090013A1 (no) |
JP (1) | JP4033630B2 (no) |
KR (1) | KR100414336B1 (no) |
CN (1) | CN1173979C (no) |
AU (1) | AU761450B2 (no) |
BR (1) | BR9911445A (no) |
CA (1) | CA2335288A1 (no) |
HU (1) | HUP0102350A2 (no) |
ID (1) | ID28433A (no) |
IL (1) | IL140010A0 (no) |
MA (1) | MA26657A1 (no) |
NO (1) | NO20006507D0 (no) |
PL (1) | PL345266A1 (no) |
TR (1) | TR200003807T2 (no) |
WO (1) | WO1999067255A1 (no) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR20020085180A (ko) * | 2001-05-07 | 2002-11-16 | 주식회사 엘지생명과학 | 신규 세팔로스포린계 항생제 및 이의 제조 방법 |
KR20020085176A (ko) * | 2001-05-07 | 2002-11-16 | 주식회사 엘지생명과학 | 신규 세팔로스포린계 항생제 및 이의 제조 방법 |
ITRM20020014A1 (it) * | 2002-01-15 | 2003-07-15 | Sigma Tau Ind Farmaceuti | Derivati di acidi a-feniltiocarbossilici e a-fenilossicarbossilici utili per il trattamento di patologie che rispondono all'attivazione del |
KR100693298B1 (ko) * | 2003-06-27 | 2007-03-13 | 영진약품공업주식회사 | 신규한 세팔로스포린계 화합물 및 약제학적으로 허용되는염과 그의 제조 방법 |
JP3928086B2 (ja) * | 2005-03-29 | 2007-06-13 | 塩野義製薬株式会社 | 3−プロペニルセフェム誘導体 |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3983113A (en) * | 1975-08-15 | 1976-09-28 | Syntex (U.S.A.) Inc. | Cephalosporin type antibacterials |
US4486586A (en) | 1983-02-10 | 1984-12-04 | Bristol-Myers Company | Cephalosporin derivatives |
US4751295A (en) | 1984-04-09 | 1988-06-14 | Bristol-Myers Company | Cephalosporin derivatives |
CA1276929C (en) | 1984-04-09 | 1990-11-27 | Masahisa Oka | Cephalosporin antibacterial agents |
FR2622585B1 (fr) | 1987-11-03 | 1991-04-19 | Roussel Uclaf | Nouvelles cephalosporines comportant en position 3 un radical vinyle substitue, leur procede de preparation, leur application comme medicaments, les compositions les renfermant et les nouveaux intermediaires obtenus |
EP0764648B1 (en) * | 1988-03-16 | 2002-01-16 | Eisai Co., Ltd. | Cephem derivatives and process for the preparation thereof |
DE69231815T2 (de) | 1991-03-08 | 2001-09-27 | Biochemie Ges.M.B.H., Kundl | Verfahren zur Herstellung von Cephalosporinen und Zwischenprodukte in diesem Verfahren |
AT396108B (de) * | 1991-08-21 | 1993-06-25 | Biochemie Gmbh | Neues verfahren und neue zwischenprodukte zur herstellung von 7-aminocephalosporansaeurederivaten |
US5523400A (en) * | 1993-04-16 | 1996-06-04 | Hoffmann-La Roche Inc. | Cephalosporin antibiotics |
CA2143519A1 (en) * | 1994-03-11 | 1995-09-12 | Markus Bohringer | Beta-lactams |
CZ251896A3 (en) * | 1995-09-12 | 1997-04-16 | Hoffmann Ka Roche Ag F | Cephalosporin derivatives |
DK0841339T3 (da) | 1996-11-06 | 2007-07-02 | Basilea Pharmaceutica Ag | Vinylpyrrolidinon-cephalosporinderivater |
US6150350A (en) * | 1997-09-15 | 2000-11-21 | Hoffman-La Roche Inc. | Antimicrobial compositions |
-
1999
- 1999-06-11 EP EP99929182A patent/EP1090013A1/en not_active Withdrawn
- 1999-06-11 TR TR2000/03807T patent/TR200003807T2/xx unknown
- 1999-06-11 CN CNB998077682A patent/CN1173979C/zh not_active Expired - Fee Related
- 1999-06-11 PL PL99345266A patent/PL345266A1/xx unknown
- 1999-06-11 HU HU0102350A patent/HUP0102350A2/hu unknown
- 1999-06-11 JP JP2000555907A patent/JP4033630B2/ja not_active Expired - Fee Related
- 1999-06-11 IL IL14001099A patent/IL140010A0/xx unknown
- 1999-06-11 BR BR9911445-3A patent/BR9911445A/pt not_active IP Right Cessation
- 1999-06-11 CA CA002335288A patent/CA2335288A1/en not_active Abandoned
- 1999-06-11 ID IDW20010140A patent/ID28433A/id unknown
- 1999-06-11 KR KR10-2000-7014573A patent/KR100414336B1/ko not_active IP Right Cessation
- 1999-06-11 AU AU46081/99A patent/AU761450B2/en not_active Ceased
- 1999-06-11 WO PCT/EP1999/004034 patent/WO1999067255A1/en active IP Right Grant
- 1999-06-21 MA MA25640A patent/MA26657A1/fr unknown
- 1999-06-22 US US09/337,908 patent/US6583133B1/en not_active Expired - Fee Related
-
2000
- 2000-12-20 NO NO20006507A patent/NO20006507D0/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
WO1999067255A1 (en) | 1999-12-29 |
CN1306536A (zh) | 2001-08-01 |
NO20006507D0 (no) | 2000-12-20 |
JP4033630B2 (ja) | 2008-01-16 |
PL345266A1 (en) | 2001-12-03 |
CA2335288A1 (en) | 1999-12-29 |
BR9911445A (pt) | 2001-03-20 |
KR100414336B1 (ko) | 2004-01-07 |
ID28433A (id) | 2001-05-24 |
EP1090013A1 (en) | 2001-04-11 |
CN1173979C (zh) | 2004-11-03 |
JP2002518505A (ja) | 2002-06-25 |
IL140010A0 (en) | 2002-02-10 |
AU4608199A (en) | 2000-01-10 |
AU761450B2 (en) | 2003-06-05 |
TR200003807T2 (tr) | 2001-06-21 |
HUP0102350A2 (hu) | 2001-11-28 |
MA26657A1 (fr) | 2004-12-20 |
US6583133B1 (en) | 2003-06-24 |
KR20010053092A (ko) | 2001-06-25 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |