NO20002191L - Dofetilid polymorfer - Google Patents
Dofetilid polymorferInfo
- Publication number
- NO20002191L NO20002191L NO20002191A NO20002191A NO20002191L NO 20002191 L NO20002191 L NO 20002191L NO 20002191 A NO20002191 A NO 20002191A NO 20002191 A NO20002191 A NO 20002191A NO 20002191 L NO20002191 L NO 20002191L
- Authority
- NO
- Norway
- Prior art keywords
- polymorphs
- dofetilide polymorphs
- dofetilide
- processes
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
- C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C311/08—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Cardiology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Heart & Thoracic Surgery (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Steroid Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pyrrole Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
Oppfinnelsen vedrører de hovedsakelige rene dofetilid polymorfer P162, P162a og P143, og fremgangsmåter for fremstillingen av, sammensetninger inneholdende og an-vendelsene av, slike polymorfer.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9722662.5A GB9722662D0 (en) | 1997-10-27 | 1997-10-27 | Polymorphs |
| PCT/EP1998/006641 WO1999021829A1 (en) | 1997-10-27 | 1998-10-09 | Dofetilide polymorphs |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20002191L true NO20002191L (no) | 2000-04-27 |
| NO20002191D0 NO20002191D0 (no) | 2000-04-27 |
| NO325630B1 NO325630B1 (no) | 2008-06-30 |
Family
ID=10821150
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20002191A NO325630B1 (no) | 1997-10-27 | 2000-04-27 | Dofetilidpolymorf, fremgangsmate for fremstilling derav samt anvendelse derav for fremstilling av medikamenter og medisinske preparater. |
Country Status (46)
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10019067C1 (de) * | 2000-04-18 | 2001-10-04 | Lohmann Therapie Syst Lts | Transdermales Therapeutisches System zur Abgabe von Dofetilid und seine Verwendung |
| US7326772B2 (en) * | 2005-05-12 | 2008-02-05 | Penta Biotech, Inc. | Peptide for assaying hERG channel binding |
| CZ2017772A3 (cs) | 2017-12-01 | 2019-05-29 | Farmak, A.S. | Způsob přípravy N-[4-(2-{[2-(4-methansulfonamidofenoxy)ethyl](methyl)amino}ethyl)fenyl]methansulfonamidu (Dofetilidu) |
| US12396970B2 (en) | 2021-08-20 | 2025-08-26 | AltaThera Pharmaceuticals LLC | Anti-arrhythmic compositions and methods |
| US10512620B1 (en) | 2018-08-14 | 2019-12-24 | AltaThera Pharmaceuticals, LLC | Method of initiating and escalating sotalol hydrochloride dosing |
| US11696902B2 (en) | 2018-08-14 | 2023-07-11 | AltaThera Pharmaceuticals, LLC | Method of initiating and escalating sotalol hydrochloride dosing |
| US11610660B1 (en) | 2021-08-20 | 2023-03-21 | AltaThera Pharmaceuticals LLC | Antiarrhythmic drug dosing methods, medical devices, and systems |
| US11344518B2 (en) | 2018-08-14 | 2022-05-31 | AltaThera Pharmaceuticals LLC | Method of converting atrial fibrillation to normal sinus rhythm and loading oral sotalol in a shortened time frame |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EG18188A (en) * | 1986-05-01 | 1992-09-30 | Pfizer Ltd | Process for preparation anti-arhythmia agents |
| EP0898964A1 (en) * | 1997-08-19 | 1999-03-03 | Pfizer Inc. | Method for treating heart failure |
-
1997
- 1997-10-27 GB GBGB9722662.5A patent/GB9722662D0/en not_active Ceased
-
1998
- 1998-09-10 UA UA2000042087A patent/UA67755C2/uk unknown
- 1998-10-08 TW TW087116747A patent/TW449589B/zh not_active IP Right Cessation
- 1998-10-09 KR KR10-2000-7004471A patent/KR100366167B1/ko not_active Expired - Fee Related
- 1998-10-09 ID IDW20000767A patent/ID24658A/id unknown
- 1998-10-09 DE DE69811256T patent/DE69811256T2/de not_active Expired - Fee Related
- 1998-10-09 TR TR2000/01135T patent/TR200001135T2/xx unknown
- 1998-10-09 CN CNB988106213A patent/CN1146537C/zh not_active Expired - Fee Related
- 1998-10-09 AU AU21512/99A patent/AU737668B2/en not_active Ceased
- 1998-10-09 HR HR970680A patent/HRP20000247B1/xx not_active IP Right Cessation
- 1998-10-09 YU YU24000A patent/YU24000A/sh unknown
- 1998-10-09 IL IL13543598A patent/IL135435A0/xx not_active IP Right Cessation
- 1998-10-09 WO PCT/EP1998/006641 patent/WO1999021829A1/en not_active Ceased
- 1998-10-09 CA CA002307121A patent/CA2307121C/en not_active Expired - Fee Related
- 1998-10-09 SK SK586-2000A patent/SK5862000A3/sk unknown
- 1998-10-09 JP JP2000517941A patent/JP3569495B2/ja not_active Expired - Fee Related
- 1998-10-09 ES ES98965638T patent/ES2190620T3/es not_active Expired - Lifetime
- 1998-10-09 AT AT98965638T patent/ATE232199T1/de not_active IP Right Cessation
- 1998-10-09 EP EP98965638A patent/EP1027329B1/en not_active Expired - Lifetime
- 1998-10-09 BR BR9813308-0A patent/BR9813308A/pt not_active Application Discontinuation
- 1998-10-09 US US09/423,986 patent/US6124363A/en not_active Expired - Lifetime
- 1998-10-09 SI SI9830347T patent/SI1027329T1/xx unknown
- 1998-10-09 HU HU0004735A patent/HUP0004735A3/hu unknown
- 1998-10-09 DK DK98965638T patent/DK1027329T3/da active
- 1998-10-09 PT PT98965638T patent/PT1027329E/pt unknown
- 1998-10-09 NZ NZ503785A patent/NZ503785A/en unknown
- 1998-10-09 EA EA200000365A patent/EA002656B1/ru not_active IP Right Cessation
- 1998-10-09 PL PL340805A patent/PL197379B1/pl unknown
- 1998-10-22 AP APAP/P/1998/001371A patent/AP906A/en active
- 1998-10-22 PA PA19988462001A patent/PA8462001A1/es unknown
- 1998-10-23 PE PE1998001003A patent/PE122199A1/es not_active Application Discontinuation
- 1998-10-23 MY MYPI98004829A patent/MY123352A/en unknown
- 1998-10-23 AR ARP980105310A patent/AR015193A1/es unknown
- 1998-10-26 TN TNTNSN98193A patent/TNSN98193A1/fr unknown
- 1998-10-26 MA MA25313A patent/MA24683A1/fr unknown
- 1998-10-26 HN HN1998000165A patent/HN1998000165A/es unknown
- 1998-10-26 ZA ZA9809719A patent/ZA989719B/xx unknown
- 1998-10-26 UY UY25222A patent/UY25222A1/es not_active IP Right Cessation
- 1998-10-26 DZ DZ980242A patent/DZ2632A1/xx active
- 1998-10-27 CO CO98062885A patent/CO4970768A1/es unknown
- 1998-10-27 GT GT199800165A patent/GT199800165A/es unknown
- 1998-11-28 SA SA98190834A patent/SA98190834B1/ar unknown
-
1999
- 1999-01-08 UY UY25341A patent/UY25341A1/es not_active IP Right Cessation
-
2000
- 2000-03-31 IS IS5426A patent/IS2179B/is unknown
- 2000-04-20 OA OA1200000117A patent/OA11350A/en unknown
- 2000-04-24 BG BG104373A patent/BG64125B1/bg unknown
- 2000-04-27 NO NO20002191A patent/NO325630B1/no not_active IP Right Cessation
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| TR200001012T2 (tr) | Yeni ariloksi-alkil-dialkilaminler. | |
| PT934325E (pt) | Trisanidridos biciclicos de tetrafosfonato | |
| ES2195970T3 (es) | L-ribavirina y usos de la misma. | |
| IL135536A0 (en) | Ortho-anthranilamide derivatives and pharmaceutical compositions containing the same | |
| BG103485A (en) | Ketobanzamides as calpain inhibitors | |
| MY113806A (en) | Antiparasitic marcfortines and paraherquamides | |
| NZ503308A (en) | Alpha-ketoamide multicatalytic protease inhibitors | |
| MX9804588A (es) | Uso de composiciones que comprenden blanqueador de halogeno para suavidad mejorada a la piel. | |
| IL109720A (en) | N-alkylthio polyamine derivatives and radioprotective compositions containing them | |
| BG99177A (bg) | Нови 7 бета-заместени-4-аза-5 алфа-холестанони като инхибитори на 5 алфа-редуктаза | |
| YU2500A (sh) | Alatrofloksacin parenteralni preparati | |
| NO20002191L (no) | Dofetilid polymorfer | |
| HU9500559D0 (en) | New mercapto-acetamide tricyclic derivatives as enkephalinase-inhibitors | |
| CA2166692A1 (en) | Novel 9-n-bicyclic nucleoside agents useful as selective inhibitors of proinflammatory cytokines | |
| MX9801190A (es) | Inhibidores de prolil endopeptidasa. | |
| SE9604582D0 (sv) | Novel compounds | |
| BG100248A (bg) | Инхибитори на скваленсинтетаза | |
| MY127474A (en) | Naphthyl compounds, intermediates, compositions, and methods of use | |
| GR3034406T3 (en) | Intermediates for the preparation of 2-imidazoline-5-ones | |
| MX9602767A (es) | Dimaleato de n,n-dietil-8,8-dipropil-2-azaspiro[4,5]decano-2-propanamina. | |
| SE9603726D0 (sv) | Novel compounds | |
| TW282449B (no) | ||
| IL119412A (en) | Gonadotropins and pharmaceutical compositions containing them | |
| ECSP982713A (es) | Polimorfos de dofetilida | |
| ES2151820A1 (es) | Herbicidas a base de derivados de 1,3-oxazin-4-ona, composiciones que los contienen y procedimiento para su preparacion. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM1K | Lapsed by not paying the annual fees |