NO20000241D0 - Tricykliske vasopressin agonister - Google Patents

Tricykliske vasopressin agonister

Info

Publication number
NO20000241D0
NO20000241D0 NO20000241A NO20000241A NO20000241D0 NO 20000241 D0 NO20000241 D0 NO 20000241D0 NO 20000241 A NO20000241 A NO 20000241A NO 20000241 A NO20000241 A NO 20000241A NO 20000241 D0 NO20000241 D0 NO 20000241D0
Authority
NO
Norway
Prior art keywords
vasopressin agonists
compounds
tricyclic
tricyclic vasopressin
nocturia
Prior art date
Application number
NO20000241A
Other languages
English (en)
Other versions
NO20000241L (no
Inventor
Amedeo Arturo Failli
Jay Scott Shumsky
Robert John Steffan
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Home Prod filed Critical American Home Prod
Publication of NO20000241D0 publication Critical patent/NO20000241D0/no
Publication of NO20000241L publication Critical patent/NO20000241L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO20000241A 1997-07-30 2000-01-18 Trisykliske vasopressin agonister NO20000241L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US94170797A 1997-07-30 1997-07-30
US90337097A 1997-07-30 1997-07-30
PCT/US1998/015487 WO1999006403A1 (en) 1997-07-30 1998-07-24 Tricyclic vasopressin agonists

Publications (2)

Publication Number Publication Date
NO20000241D0 true NO20000241D0 (no) 2000-01-18
NO20000241L NO20000241L (no) 2000-03-06

Family

ID=27129361

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20000241A NO20000241L (no) 1997-07-30 2000-01-18 Trisykliske vasopressin agonister

Country Status (17)

Country Link
EP (1) EP1000059B1 (no)
JP (1) JP2001512120A (no)
KR (1) KR20010022397A (no)
CN (1) CN1162429C (no)
AT (1) ATE277926T1 (no)
AU (1) AU8592598A (no)
BR (1) BR9811559A (no)
CA (1) CA2297407A1 (no)
DE (1) DE69826677T2 (no)
DK (1) DK1000059T3 (no)
ES (1) ES2229523T3 (no)
HU (1) HUP0003394A3 (no)
IL (1) IL133787A0 (no)
NO (1) NO20000241L (no)
NZ (1) NZ502448A (no)
PT (1) PT1000059E (no)
WO (1) WO1999006403A1 (no)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2358895A1 (en) * 1999-02-04 2000-08-10 Wyeth Pyridobenzodiazepine and pyridobenzoxazepine carboxyamide vasopressin agonists
DK1149096T3 (da) * 1999-02-04 2003-04-07 Wyeth Corp Tricykliske pyridin-N-oxider som vasopressinagonister
GB0000079D0 (en) * 2000-01-05 2000-02-23 Ferring Bv Novel antidiuretic agents
GB0015601D0 (en) 2000-06-26 2000-08-16 Ferring Bv Novel antidiuretic agents
WO2002044180A1 (fr) 2000-12-01 2002-06-06 Ajinomoto Co.,Inc. Composes de lactame et leur utilisation medicale
ATE512951T1 (de) 2003-04-28 2011-07-15 Astellas Pharma Inc 4,4-difluor-1,2,3,4-tetrahydro-5h-1- benzazepinderivat oder salz davon
GB201005623D0 (en) 2010-04-01 2010-05-19 Vantia Ltd New polymorph
AR094929A1 (es) 2013-02-28 2015-09-09 Bristol Myers Squibb Co Derivados de fenilpirazol como inhibidores potentes de rock1 y rock2
WO2014134391A1 (en) 2013-02-28 2014-09-04 Bristol-Myers Squibb Company Phenylpyrazole derivatives as potent rock1 and rock2 inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1251767B (de) * 1964-02-28 1968-04-18 Dr Karl Thomae Gesellschaft mit beschrankter Haftung Biberach/Riß Verfahren zur Herstellung von neuen m 6 Stellung substituierten 5 6 Dihydro-5oxo HH pyrido[2,3-b] [l,5]benzodiazepinen
US5512563A (en) * 1993-07-29 1996-04-30 American Cyanamid Company Tricyclic benzazepine vasopressin antagonists
US5420270A (en) * 1993-10-07 1995-05-30 G. D. Searle & Co. Aryl substituted dibenzoxazepine compounds, pharmaceutical compositions and methods of use
AR002459A1 (es) * 1995-01-17 1998-03-25 American Cyanamid Co Antagonistas de vasopresina de benzacepina triciclicos, una composicion farmaceutica que los contiene, un metodo para tratar enfermedades y unprocedimiento para su preparacion.
TW359669B (en) * 1995-12-15 1999-06-01 Otsuka Pharma Co Ltd Benzazepine derivatives

Also Published As

Publication number Publication date
KR20010022397A (ko) 2001-03-15
EP1000059A1 (en) 2000-05-17
JP2001512120A (ja) 2001-08-21
WO1999006403A1 (en) 1999-02-11
HUP0003394A2 (hu) 2001-08-28
CA2297407A1 (en) 1999-02-11
EP1000059B1 (en) 2004-09-29
CN1162429C (zh) 2004-08-18
HUP0003394A3 (en) 2003-04-28
DE69826677T2 (de) 2005-02-10
ATE277926T1 (de) 2004-10-15
ES2229523T3 (es) 2005-04-16
NO20000241L (no) 2000-03-06
DK1000059T3 (da) 2005-01-10
PT1000059E (pt) 2004-12-31
IL133787A0 (en) 2001-04-30
BR9811559A (pt) 2000-09-12
DE69826677D1 (de) 2004-11-04
NZ502448A (en) 2002-12-20
CN1272110A (zh) 2000-11-01
AU8592598A (en) 1999-02-22

Similar Documents

Publication Publication Date Title
EA200300713A1 (ru) Производные бензимидазола и пиридилимидазола в качестве лигандов рецепторов гамма-аминомасляной кислоты
NO20000242D0 (no) Tricykliske vasopressin agonister
MA25809A1 (fr) Derives d'arylmethylamine pour usage comme inhibiteurs de tryptase
EA200400337A1 (ru) Применение модулятора рецепторов глюкокортикоидов и агониста рецепторов глюкокортикоидов при получении лекарственного средства
BR0208940A (pt) Composto diazepìnico tricìclico, composição farmacêutica compreendendo o mesmo e seu uso
EA200200208A1 (ru) Синергитическая композиция
DE69926806D1 (de) N-ureidoalkylpiperidine als modulatoren der aktivität der chemokinrezeptoren
DE69926919D1 (de) N-ureidoalkylpiperidine als modulatoren der aktivität der chemokinrezeptoren
EA200400466A1 (ru) Производные пиперазина с антагонистической активностью к рецептору ccr1
EA200301142A1 (ru) Производные гетероциклилокси-, -тиокси- и -аминобензазола в качестве лигандов 5-гидрокситриптамина-6
ATE413388T1 (de) Muskarin antagonisten
EA200300716A1 (ru) Гетероциклилалкилиндольные или -азаиндольные соединения в качестве лиганд 5-гидрокситриптамина-6
DK1000059T3 (da) Tricycliske vasopressin-agonister
EA200200132A1 (ru) СЕЛЕКТИВНЫЕ АНТАГОНИСТЫ РЕЦЕПТОРА iGluRДЛЯ ЛЕЧЕНИЯ МИГРЕНИ
BR0011122A (pt) Antagonistas de receptor il-8
IT1293804B1 (it) Diarilalchilpiperazine attive sulle basse vie urinarie
BR0208824A (pt) Composto, métodos de tratamento de distúrbios que são remediados ou aliviados por atividade de agonista de vasopressina em um mamìfero, e de indução de retardamento temporário de urinação em um mamìfero, e, composição farmacêutica
WO2000046224A3 (en) Tricyclic pyridine n-oxides vasopressin agonists
WO2000046225A3 (en) Pyridobenzodiazepine and pyridobenzoxazepine carboxyamide vasopressin agonists
BRPI0415966A (pt) combinações compreendendo antagonistas do receptor ampa para tratamento de esquizofrenia
ATE229528T1 (de) Pyrrolobenzodiazepine carboxamide vasopressin agonisten
DE60117517D1 (de) Indolderivate als mcp-1 rezeptor antagonisten
AR028470A1 (es) Ariltiofeno agonistas de vasopresina, el uso de los mismos para manufactura de un medicamento y composicion farmaceutica

Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application