NO178923C - Analogifremgangsmåte for fremstilling av terapeutisk aktive 24-homo-vitamin-D-derivater - Google Patents

Analogifremgangsmåte for fremstilling av terapeutisk aktive 24-homo-vitamin-D-derivater

Info

Publication number
NO178923C
NO178923C NO904269A NO904269A NO178923C NO 178923 C NO178923 C NO 178923C NO 904269 A NO904269 A NO 904269A NO 904269 A NO904269 A NO 904269A NO 178923 C NO178923 C NO 178923C
Authority
NO
Norway
Prior art keywords
carbon atoms
derivatives
preparation
therapeutically active
analogous process
Prior art date
Application number
NO904269A
Other languages
English (en)
Other versions
NO904269D0 (no
NO904269L (no
NO178923B (no
Inventor
Gerald Dr Kirsch
Guenter Dr Neef
Katica Schwarz
Matthias Dr Braeutigam
Ruth Dr Thieroff-Eckerdt
Petra Rach
Original Assignee
Schering Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Schering Ag filed Critical Schering Ag
Publication of NO904269D0 publication Critical patent/NO904269D0/no
Publication of NO904269L publication Critical patent/NO904269L/no
Publication of NO178923B publication Critical patent/NO178923B/no
Publication of NO178923C publication Critical patent/NO178923C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C401/00—Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/02—Nutrients, e.g. vitamins, minerals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nutrition Science (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
NO904269A 1989-10-02 1990-10-01 Analogifremgangsmåte for fremstilling av terapeutisk aktive 24-homo-vitamin-D-derivater NO178923C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3933034A DE3933034A1 (de) 1989-10-02 1989-10-02 24-homo-vitamin-d-derivate, verfahren zu ihrer herstellung

Publications (4)

Publication Number Publication Date
NO904269D0 NO904269D0 (no) 1990-10-01
NO904269L NO904269L (no) 1991-04-03
NO178923B NO178923B (no) 1996-03-25
NO178923C true NO178923C (no) 1996-07-03

Family

ID=6390762

Family Applications (1)

Application Number Title Priority Date Filing Date
NO904269A NO178923C (no) 1989-10-02 1990-10-01 Analogifremgangsmåte for fremstilling av terapeutisk aktive 24-homo-vitamin-D-derivater

Country Status (18)

Country Link
US (1) US5665716A (no)
EP (1) EP0421561B1 (no)
JP (1) JPH03246273A (no)
CN (2) CN1031705C (no)
AT (1) ATE103893T1 (no)
AU (1) AU639717B2 (no)
CA (1) CA2026671C (no)
DD (1) DD299178A5 (no)
DE (2) DE3933034A1 (no)
DK (1) DK0421561T3 (no)
ES (1) ES2052166T3 (no)
FI (1) FI93643C (no)
HU (1) HU210032B (no)
IE (1) IE71227B1 (no)
IL (1) IL95872A (no)
NO (1) NO178923C (no)
PT (1) PT95473B (no)
ZA (1) ZA907876B (no)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5260290A (en) * 1990-02-14 1993-11-09 Wisconsin Alumni Research Foundation Homologated vitamin D2 compounds and the corresponding 1α-hydroxylated derivatives
US5030772A (en) * 1990-02-14 1991-07-09 Deluca Hector F Process for preparing vitamin D2 compounds and the corresponding 1 α-hydroxylated derivatives
US20040009958A1 (en) * 1991-01-08 2004-01-15 Bone Care International, Inc. Methods for preparation and use of 1alpha,24(S)-dihydroxyvitamin D2
DE4200783C2 (de) * 1992-01-10 1997-02-06 Schering Ag (5Z,7E,22E)-(1S,3R,24S)-24-Benzyl-9,10-secochola-5,7,10(19),22-tetraen-1,3,24-triol, Verfahren zur Herstellung und Pharmazeutische Präparate
IL107185A (en) * 1992-10-06 1998-02-22 Schering Ag Vitamin d, 25-carboxylic acid derivatives and pharmaceutical compositions containing the same
DE4328217C2 (de) * 1993-08-21 1996-01-11 Lohmann Therapie Syst Lts Therapeutisches System zur Behandlung der Psoriasis
US6242434B1 (en) * 1997-08-08 2001-06-05 Bone Care International, Inc. 24-hydroxyvitamin D, analogs and uses thereof
DE19619036A1 (de) 1996-04-30 1997-11-13 Schering Ag Neue Vitamin D-Derivate mit carbo- oder heterocyclischen Substituenten an C-25, Verfahren zu ihrer Herstellung und die Verwendung zur Herstellung von Arzneimitteln
US5939408A (en) 1996-05-23 1999-08-17 Hoffman-La Roche Inc. Vitamin D3 analogs
US20020128240A1 (en) * 1996-12-30 2002-09-12 Bone Care International, Inc. Treatment of hyperproliferative diseases using active vitamin D analogues
US20030129194A1 (en) * 1997-02-13 2003-07-10 Bone Care International, Inc. Targeted therapeutic delivery of vitamin D compounds
DE19935771A1 (de) 1999-07-23 2001-02-01 Schering Ag Neue Vitamin D-Derivate mit cyclischen Substrukturen in den Seitenketten, Verfahren und Zwischenprodukte zu ihrer Herstellung und die Verwendung zur Herstellung von Arzneimitteln
WO2002006218A2 (en) * 2000-07-18 2002-01-24 Bone Care International, Inc. STABILIZED 1α-HYDROXY VITAMIN D
DE10156596A1 (de) * 2001-11-13 2003-05-28 Schering Ag Vitamin D-Derivate mit Acyloxygruppen in der Seitenkette, Verfahren zu ihrer Herstellung und die Verwendung zur Herstellung von Arzneimitteln
EP1470220B1 (en) * 2002-01-10 2011-10-05 Teva Pharmaceutical Industries, Ltd. Selective enzymatic esterification and solvolysis of epimeric vitamin d analog and separation of the epimers
EP1461314A1 (en) * 2002-06-13 2004-09-29 Teva Pharmaceutical Industries Limited Epimerization of analogs of vitamin d
US7094775B2 (en) 2004-06-30 2006-08-22 Bone Care International, Llc Method of treating breast cancer using a combination of vitamin D analogues and other agents
KR20090039833A (ko) * 2006-08-29 2009-04-22 테바 파마슈티컬 인더스트리즈 리미티드 비타민 ｄ 및 코르티코스테로이드를 포함하는 약학 조성물
US8716334B2 (en) 2008-06-17 2014-05-06 Ben Gurion University Of The Negev Research And Development Authority Substituted cyclohexylidene-ethylidene-octahydro-indene compounds
SG2014006324A (en) 2009-01-27 2014-03-28 Berg Llc Vitamin d3 and analogs thereof for alleviating side effects associated with chemotherapy
CN102655869B (zh) 2009-08-14 2016-08-10 博格有限责任公司 用于治疗脱发的维生素d3及其类似物
HK1222819A1 (zh) 2013-05-29 2017-07-14 博格有限责任公司 使用维生素d预防或减轻化疗诱发的脱发
US10548908B2 (en) 2016-09-15 2020-02-04 Nostopharma, LLC Compositions and methods for preventing and treating heterotopic ossification and pathologic calcification

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0197949A1 (en) * 1984-10-04 1986-10-22 Wisconsin Alumni Research Foundation Vitamin d derivatives and methods for preparing same
WO1987003282A1 (fr) * 1985-11-21 1987-06-04 Taisho Pharmaceutical Co., Ltd. Derive de la vitamine d3
US4847012A (en) * 1988-04-29 1989-07-11 Wisconsin Alumni Research Foundation Vitamin D related compounds and processes for their preparation
US4927815A (en) * 1988-04-29 1990-05-22 Wisconsin Alumni Research Foundation Compounds effective in inducing cell differentiation and process for preparing same
US5030772A (en) * 1990-02-14 1991-07-09 Deluca Hector F Process for preparing vitamin D2 compounds and the corresponding 1 α-hydroxylated derivatives
US5260290A (en) * 1990-02-14 1993-11-09 Wisconsin Alumni Research Foundation Homologated vitamin D2 compounds and the corresponding 1α-hydroxylated derivatives

Also Published As

Publication number Publication date
PT95473B (pt) 1997-07-31
DE59005254D1 (de) 1994-05-11
DK0421561T3 (da) 1994-07-25
NO904269D0 (no) 1990-10-01
AU639717B2 (en) 1993-08-05
ES2052166T3 (es) 1994-07-01
DE3933034A1 (de) 1991-04-11
HUT55751A (en) 1991-06-28
CA2026671A1 (en) 1991-04-03
CN1053103C (zh) 2000-06-07
JPH03246273A (ja) 1991-11-01
ATE103893T1 (de) 1994-04-15
ZA907876B (en) 1992-04-29
CN1051907A (zh) 1991-06-05
NO904269L (no) 1991-04-03
IL95872A (en) 1995-03-15
IE903520A1 (en) 1991-04-10
NO178923B (no) 1996-03-25
PT95473A (pt) 1991-06-25
CN1031705C (zh) 1996-05-01
AU6371590A (en) 1991-04-11
EP0421561A3 (en) 1991-06-12
FI904850A0 (fi) 1990-10-02
HU210032B (en) 1995-01-30
US5665716A (en) 1997-09-09
EP0421561A2 (de) 1991-04-10
IE71227B1 (en) 1997-02-12
IL95872A0 (en) 1991-07-18
EP0421561B1 (de) 1994-04-06
HU906284D0 (en) 1991-03-28
CN1106666A (zh) 1995-08-16
FI93643B (fi) 1995-01-31
FI93643C (fi) 1995-05-10
DD299178A5 (de) 1992-04-02
CA2026671C (en) 1998-12-08

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Legal Events

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MM1K Lapsed by not paying the annual fees

Free format text: LAPSED IN APRIL 2001