NO161562C - Analogifremgangsmaate for fremstilling av terapeutisk aktive ergolinderivater. - Google Patents

Analogifremgangsmaate for fremstilling av terapeutisk aktive ergolinderivater.

Info

Publication number
NO161562C
NO161562C NO841657A NO841657A NO161562C NO 161562 C NO161562 C NO 161562C NO 841657 A NO841657 A NO 841657A NO 841657 A NO841657 A NO 841657A NO 161562 C NO161562 C NO 161562C
Authority
NO
Norway
Prior art keywords
preparation
therapeutic active
analogy procedure
ergolin
derivatives
Prior art date
Application number
NO841657A
Other languages
English (en)
Norwegian (no)
Other versions
NO161562B (no
NO841657L (no
Inventor
Luigi Bernardi
Laura Chiodini
Sergio Mantegani
Daniela Ruggieri
Aldemio Temperilli
Patricia Salvati
Original Assignee
Erba Carlo Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB838311679A external-priority patent/GB8311679D0/en
Priority claimed from GB838314816A external-priority patent/GB8314816D0/en
Application filed by Erba Carlo Spa filed Critical Erba Carlo Spa
Publication of NO841657L publication Critical patent/NO841657L/no
Publication of NO161562B publication Critical patent/NO161562B/no
Publication of NO161562C publication Critical patent/NO161562C/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D457/00Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D457/00Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/02Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hydrocarbon or substituted hydrocarbon radicals, attached in position 8
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D457/00Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/10Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hetero atoms directly attached in position 8
    • C07D457/12Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO841657A 1983-04-28 1984-04-26 Analogifremgangsmaate for fremstilling av terapeutisk aktive ergolinderivater. NO161562C (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB838311679A GB8311679D0 (en) 1983-04-28 1983-04-28 Ergoline derivatives
GB838314816A GB8314816D0 (en) 1983-05-27 1983-05-27 Ergoline derivatives

Publications (3)

Publication Number Publication Date
NO841657L NO841657L (no) 1984-10-29
NO161562B NO161562B (no) 1989-05-22
NO161562C true NO161562C (no) 1989-08-30

Family

ID=26285978

Family Applications (1)

Application Number Title Priority Date Filing Date
NO841657A NO161562C (no) 1983-04-28 1984-04-26 Analogifremgangsmaate for fremstilling av terapeutisk aktive ergolinderivater.

Country Status (18)

Country Link
US (1) US4690929A (xx)
EP (1) EP0126968B1 (xx)
KR (1) KR900008696B1 (xx)
AU (1) AU556968B2 (xx)
CA (1) CA1205801A (xx)
DE (1) DE3475709D1 (xx)
DK (1) DK162996C (xx)
ES (1) ES531906A0 (xx)
FI (1) FI81349C (xx)
GR (1) GR79575B (xx)
HU (1) HU198713B (xx)
IE (1) IE57240B1 (xx)
IL (1) IL71633A (xx)
NO (1) NO161562C (xx)
PH (1) PH21123A (xx)
PT (1) PT78496B (xx)
SU (1) SU1327788A3 (xx)
YU (1) YU43357B (xx)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8714767D0 (en) * 1987-06-24 1987-07-29 Erba Farmitalia Egoline derivatives
HU196399B (en) * 1983-02-16 1988-11-28 Sandoz Ag Process for producing ergoline derivatives and pharmaceutical compositions comprising such compounds
GB8501078D0 (en) * 1985-01-16 1985-02-20 Erba Farmitalia Piperazin-1-yl-ergo-line derivatives
GB2173189B (en) * 1985-02-21 1988-04-27 Maruko Pharmaceutical Co Ergoline derivatives and salts thereof and pharmaceutical compositions thereof
GB8515528D0 (en) * 1985-06-19 1985-07-24 Erba Farmitalia Ergoline derivatives
US4801712A (en) * 1985-06-24 1989-01-31 Eli Lilly And Company 2-Alkyl(or phenyl)thio-6-n-alkylergolines are dopamine D-1 antagonists without D-2 agonist activity
DE3528576A1 (de) * 1985-08-06 1987-02-19 Schering Ag Verfahren zur herstellung von ergolin-thioharnstoffen
DE3535929A1 (de) * 1985-10-04 1987-04-09 Schering Ag 1,2-disubstituierte ergolinderivate
GB8617907D0 (en) * 1986-07-22 1986-08-28 Erba Farmitalia Tetracyclic indole derivatives
GB8702364D0 (en) * 1987-02-03 1987-03-11 Erba Farmitalia Ergolinyl heterocycles
DK338789A (da) * 1988-07-15 1990-01-16 Schering Ag 2-substituerede ergolinylurinstofderivater og fremgangsmaade til fremstilling deraf, deres anvendelse som laegemidler samt mellemprodukter til fremstilling deraf
RU2074857C1 (ru) * 1990-01-25 1997-03-10 Фармиталиа Карло Эрба С.Р.Л. Способ получения производных эрголина
GB9006772D0 (en) * 1990-03-27 1990-05-23 Erba Carlo Spa 4-piperidinyl-ergoline derivatives
HU220391B (hu) * 1992-12-24 2002-01-28 Farmitalia Carlo Erba S.R.L. Szerotoninerg hatású ergolinszármazékok, e vegyületeket tartalmazó gyógyszerkészítmények és eljárás azok előállítására
DK1401863T3 (da) 2001-06-08 2009-05-25 Ipsen Pharma Kimære somatostatin-dopamin-analoge
TWI523863B (zh) 2012-11-01 2016-03-01 艾普森藥品公司 體抑素-多巴胺嵌合體類似物
JP2016503402A (ja) 2012-11-01 2016-02-04 イプセン ファルマ ソシエテ パール アクシオン サンプリフィエIpsen Pharma S.A.S. ソマトスタチン類似体及びそのダイマー

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE622316A (xx) * 1961-09-11
DK140596B (da) * 1971-05-19 1979-10-08 Sandoz Ag Analogifremgangsmåde til fremstilling af 8beta-(ureidomethyl)-ergolenderivater.
US3996228A (en) * 1973-12-21 1976-12-07 Societa' Farmaceutici Italia S.P.A. Pyrimidinoaminoethyl ergoline derivatives
NL7416120A (nl) * 1973-12-21 1975-06-24 Farmaceutici Italia Werkwijze voor het bereiden van pyrimidinoami- nomethylergolinederivaten.
DE2456930A1 (de) * 1974-12-02 1976-08-12 Tesch Kg E Elektronisches zeitspeicherrelais
CH615181A5 (en) * 1975-05-21 1980-01-15 Sandoz Ag Process for the preparation of novel ergolene derivatives
GB2056437A (en) * 1979-08-07 1981-03-18 Erba Farmitalia Secoergoline derivatives
DE3001752A1 (de) * 1980-01-16 1981-07-30 Schering Ag Berlin Und Bergkamen, 1000 Berlin Verfahren zur herstellung von 8(alpha)-substituierten 6-methylergolinen
DD154897A1 (de) * 1980-12-02 1982-04-28 Seifert Karlheinz Dipl Chem Dr Verfahren zur herstellung von 8-substituierten ergolinen
DE3101535A1 (de) * 1981-01-14 1982-08-12 Schering Ag, 1000 Berlin Und 4619 Bergkamen Neue (2-halogen-ergolinyl)-n'.n'-diethyl-harnstoffderivate, verfahren zu ihrer herstellung und deren verwendung als arzneimittel
GB2112382B (en) * 1981-11-06 1985-03-06 Erba Farmitalia Ergoline derivatives

Also Published As

Publication number Publication date
PT78496A (en) 1984-05-01
HUT34024A (en) 1985-01-28
IE57240B1 (en) 1992-06-17
AU556968B2 (en) 1986-11-27
PH21123A (en) 1987-07-27
KR900008696B1 (ko) 1990-11-27
ES8506031A1 (es) 1985-06-01
EP0126968B1 (en) 1988-12-21
FI841631A0 (xx) 1984-04-25
NO161562B (no) 1989-05-22
CA1205801A (en) 1986-06-10
IL71633A0 (en) 1984-07-31
FI81349C (fi) 1990-10-10
YU43357B (en) 1989-06-30
KR840008353A (ko) 1984-12-14
US4690929A (en) 1987-09-01
FI841631A (xx) 1984-10-29
DK162996C (da) 1992-06-01
PT78496B (en) 1986-07-22
HU198713B (en) 1989-11-28
ES531906A0 (es) 1985-06-01
AU2742184A (en) 1984-11-01
DE3475709D1 (en) 1989-01-26
SU1327788A3 (ru) 1987-07-30
DK212784D0 (da) 1984-04-27
EP0126968A1 (en) 1984-12-05
IL71633A (en) 1987-12-20
NO841657L (no) 1984-10-29
DK162996B (da) 1992-01-06
DK212784A (da) 1984-10-29
FI81349B (fi) 1990-06-29
YU74284A (en) 1986-10-31
GR79575B (xx) 1984-10-30

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