NL8700046A - 8 alfa-acylaminoergolinen, werkwijzen voor hun bereiding en farmaceutische preparaten die ze bevatten. - Google Patents

8 alfa-acylaminoergolinen, werkwijzen voor hun bereiding en farmaceutische preparaten die ze bevatten. Download PDF

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Publication number
NL8700046A
NL8700046A NL8700046A NL8700046A NL8700046A NL 8700046 A NL8700046 A NL 8700046A NL 8700046 A NL8700046 A NL 8700046A NL 8700046 A NL8700046 A NL 8700046A NL 8700046 A NL8700046 A NL 8700046A
Authority
NL
Netherlands
Prior art keywords
group
formula
compound
alkyl group
carbon atoms
Prior art date
Application number
NL8700046A
Other languages
English (en)
Dutch (nl)
Original Assignee
Sandoz Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sandoz Ag filed Critical Sandoz Ag
Publication of NL8700046A publication Critical patent/NL8700046A/nl

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D457/00Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/10Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hetero atoms directly attached in position 8
    • C07D457/12Nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/08Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine
NL8700046A 1986-01-24 1987-01-12 8 alfa-acylaminoergolinen, werkwijzen voor hun bereiding en farmaceutische preparaten die ze bevatten. NL8700046A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3602058 1986-01-24
DE3602058 1986-01-24

Publications (1)

Publication Number Publication Date
NL8700046A true NL8700046A (nl) 1987-08-17

Family

ID=6292510

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8700046A NL8700046A (nl) 1986-01-24 1987-01-12 8 alfa-acylaminoergolinen, werkwijzen voor hun bereiding en farmaceutische preparaten die ze bevatten.

Country Status (18)

Country Link
JP (1) JPS62190184A (fr)
KR (1) KR870007175A (fr)
AU (1) AU6791487A (fr)
BE (1) BE1000039A4 (fr)
DK (1) DK35787A (fr)
ES (1) ES2003774A6 (fr)
FI (1) FI870293A (fr)
FR (1) FR2595699A1 (fr)
GB (1) GB2185743A (fr)
GR (1) GR870093B (fr)
HU (1) HUT45248A (fr)
IL (1) IL81355A0 (fr)
IT (1) IT1216783B (fr)
LU (1) LU86743A1 (fr)
NL (1) NL8700046A (fr)
PT (1) PT84184A (fr)
SE (1) SE8700250L (fr)
ZA (1) ZA87520B (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8714767D0 (en) * 1987-06-24 1987-07-29 Erba Farmitalia Egoline derivatives
EP0160842B1 (fr) * 1984-04-09 1994-06-22 Schering Aktiengesellschaft Dérivés d'ergoline substitués sur la position 2, procédés pour leur préparation et leur utilisation comme médicaments
DK338789A (da) * 1988-07-15 1990-01-16 Schering Ag 2-substituerede ergolinylurinstofderivater og fremgangsmaade til fremstilling deraf, deres anvendelse som laegemidler samt mellemprodukter til fremstilling deraf
DE3915950A1 (de) * 1989-05-12 1990-11-15 Schering Ag 8(alpha)-acylamino-ergoline, ihre herstellung und verwendung als arzneimittel
BR112013033339A2 (pt) 2011-06-23 2016-08-16 Map Pharmaceuticals Inc análogos de fluorergolina
EP2793580A4 (fr) * 2011-12-19 2015-05-20 Map Pharmaceuticals Inc Nouveaux dérivés d'iso-ergoline
US9657020B2 (en) 2015-01-20 2017-05-23 Xoc Pharmaceuticals, Inc. Ergoline compounds and uses thereof
JP2018502889A (ja) * 2015-01-20 2018-02-01 エックスオーシー ファーマシューティカルズ インコーポレイテッドXoc Pharmaceuticals, Inc イソエルゴリン化合物およびその使用
BR112019025420A2 (pt) 2017-06-01 2020-06-16 Xoc Pharmaceuticals, Inc. Compostos policíclicos e usos destes

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1517973A (en) * 1974-07-19 1978-07-19 Sandoz Ltd 6-methyl-8alpha-n,n-dimethylsulphamoylaminoergoline i
CH615929A5 (en) * 1975-06-02 1980-02-29 Sandoz Ag Process for the preparation of novel ergoline compounds
CH664568A5 (de) * 1984-01-12 1988-03-15 Sandoz Ag 8-alpha-acylaminoergoline.

Also Published As

Publication number Publication date
FI870293A (fi) 1987-07-25
FI870293A0 (fi) 1987-01-23
HUT45248A (en) 1988-06-28
ES2003774A6 (es) 1988-11-16
IT1216783B (it) 1990-03-14
BE1000039A4 (fr) 1987-12-15
PT84184A (pt) 1987-02-01
FR2595699A1 (fr) 1987-09-18
GB2185743A (en) 1987-07-29
GR870093B (en) 1987-05-25
IT8747551A0 (it) 1987-01-22
IL81355A0 (en) 1987-08-31
ZA87520B (en) 1988-09-28
AU6791487A (en) 1987-07-30
JPS62190184A (ja) 1987-08-20
LU86743A1 (fr) 1987-09-03
DK35787D0 (da) 1987-01-22
GB8701274D0 (en) 1987-02-25
SE8700250D0 (sv) 1987-01-22
KR870007175A (ko) 1987-08-17
DK35787A (da) 1987-07-25
SE8700250L (sv) 1987-07-25

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